ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)


Volume 14, 12 Issues, 2017


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Letters in Drug Design & Discovery

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Editor-in-Chief:
G. Perry
University of Texas
San Antonio, TX
USA


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Abstracts Ahead of Print

2-Amino analogues of alkynyl substituted 1,4-dihydropyrimidine: Their synthesis and evaluation as potential antimicrobial / cytotoxic agents


V. Mallikarjuna Rao , P. Ravi Kumar , S. Shobha Rani , A. Srinivasa Rao and Manojit Pal *.


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Charting the Bromodomain BRD4: Towards the Identification of Novel Inhibitors with Molecular Similarity and Receptor Mapping


Fernando D. Prieto-Martinez and Jose L Medina-Franco*.


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Barbaterpene and barbatusterol, new constituents from Plectranthus barbatus growing in Saudi Arabia


Musarat Amina *, Nawal M. Al Musayeib , Mansour S Al-Said , Rania A Al-Zaharni , Sabrin R.M. Ibrahim and Gamal A Mohamed.


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Unveiling the Accuracy of Homology Modeling to Elucidate the Structure of GPCRs-HIV Co-receptor-CCR5 as a Case Study


Vadivelu Aanand , Rajendran Anitha , Somarathinam Kanagasabai , Gunalan Seshan , Changdev G Gadhe and Gugan Kothandan *.


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2-Indolinone Derivatives as Potent Urease Inhibitors


Momin Khan *, Muhammad Yousaf , Abdul Wadood , Zahid Hussain, Muhammad Naeem , Khalid Mohammed Khan and Shahnaz Perveen.


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The Possible Potency of Ocimum basilicum New Constituent on Glucose-stimulated Insulin Secretion In vitro and β-cell Function In vivo


Huma Aslam Bhatti , Kiran Maryam , Rizwana S. Waraich , Abdul Hameed and Rahman M Hafizur.


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Synthesis, surface properties and antimicrobial effect of hydroxymethyl-substituted pyridinium salts


Kamil Kuca*.


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Rational design, synthesis and biological evaluation of novel derivatives based on in vivo metabolism of natural product β-elemene


Renren Bai*, Xiaokang Jie , Eric Salgado , Jian Sun, Yao Zhu, Thomas Pickel , Yuanyuan Xie, Jichao Chen and Jinyi Xu.


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Theoretical modeling and systemic analysis of various active dipeptides and analogues with 3D-QSAR methods


Guanghui Tang, Ya Zhang, Cheng Chen, Yuping Zhang, Zhihua Lin* and Yuanqiang Wang.


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Antihelmintic Activity of Some 2-Substituted Thieno[2,3-d]pyrimidine-4-ones


Anelia Mavrova, Stefan Dimov, Dimitar Vutchev, Kameliya Anichina and Denitsa Yancheva*.


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Synthesis, Characterization, Biological activity of novel 1H-benzo[f]-chromene and 12H-benzo[f]chromeno[2,3-d]pyrimidine derivatives


Heba K. Abd El-Mawgoud, Hebat Allah M. Radwan, Fatma El-Mariah and Ahmed M El-Agrody *.


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Efficient Synthesis of Ibandronate in the Presence of an Ionic Liquid


David Illes Nagy, Alajos Grun, Oliver Pavela, Sandor Garadnay, Istvan Greiner and Gyorgy Keglevich*.


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3D-QSAR modeling of some S-trityl-L-Cysteine analogues as inhibitors of mitotic kinesin Eg5 by CoMFA, CoMSIA and H-QSAR methodologies


Fatemeh Mousavi* and Mohammad Hossein Fatemi*.


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Enhanced Antibacterial Activity of endo-nortropine substituted (C-7) Fluoroquinolones against V. cholerae, S. aureus and B. subtilis


Ramkrushna Ashok Salunke, Chandni Sidhu, Ashok Rana, Anil Kumar Pinnaka, Baldev Raj Bansal and Manmohan Chhibber*.


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4-Acetamidobenzaldehyde derivatives as biological active candidates; Synthesis, anti-oxidant, anti-Alzheimer and DNA binding studies


Shahzad Murtaza* and Adina Tatheer.


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Synthesis, Biological Evaluation and Docking studies of N-(2-benzamido feruloyl) Aryl hydrazone Analogues


M. Soujanya * and G Rajitha.


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Molecular and cellular mechanism of cutaneous injuries due to exposure to sulfur mustard


Yunes Panahi , Seyyed Mahdi Rajaee and Amirhossein Sahebkar*.


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Synthesis, biological evaluation and computational study of new quinoline hybrids as antitubercular agent


Zahid Zaheer*, Sameer I. Shaikh, Santosh N. Mokale and Deepak K Lokwani.


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Reactivation Potential of Novel More Lipophilic Pralidoxime Analogs


Martina Hrabinova, Jan Misik, Daniel Jun and Kamil Kuca.


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Novel Hybrid Molecules Of Quinazoline Chalcone Derivatives: Synthesis And Study Of Invitro Cytotoxic Activities


Arunkumar Thiriveedhi*, Ratnakaram Venkata Nadh, Navuluri Srinivasu and Kishore Kaushal.


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Inhibitory effects of 1,4-disubstituted thiosemicarbazide derivatives on Streptococcus mutans and Streptococcus sanguinis mono-species biofilms


Malgorzata Miazga-Karska, Maciej Wos, Agnieszka A. Kaczor, Anna Pachuta-Stec, Grazyna Ginalska and Monika Pitucha*.


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Synthesis and biological activity of new Schiff bases of benzylideneamine bearing thiophene, 1,2,4-triazolone, 1,3,4-oxadiazole , morpholine moieties


Yasemin Unver* and Ersan Bektas.


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Synthesis, Pharmacological Evaluation and Docking Study of a New Modulator of Microtubule Polymerization


Teiliane R. Carneiro, Daniel N. do Amaral, Harold H. Fokoue, Carlos M.R. Sant`Anna, Maria L.G. Porras, Cláudia Pessoa, Augusto C.A. Oliveira, Eliezer J Barreiro, Bruno C. Cavalcanti and Lidia Moreira Lima.


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Synthesis, aqueous solubility, metabolic stability and pharmacological profile of simplified urea derivatives


Raquel de Oliveira Lopes, Roberta Olmo Pinheiro, Cristina Setim Freitas, Fernando Q Cunha, Eliezer J. Barreiro* and Lídia Moreira Lima.


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Review of medicinal plants and their compounds for aldose reductase inhibitory activity


Saliha Bouknana, Mohamed Bouhrim, Hayat Ouassou and Mohamed Bnouham*.


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Antimicrobial Activities of Synthetic Arylidine Nicotinic and Isonicotinic Hydrazones


Muhammad Hayat, Khalid Mohammed Khan*, Sumayya Saeed, Uzma Salar, Momin Khan, Taimoor Baig, Aqeel Ahmad, Shahnaz Perveen and Muhammad Taha.


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