Title: New and Efficient Synthesis of 2-Alkoxyapomorphines
Volume: 4
Issue: 1
Author(s): Sandor Berenyi, Csaba Csutoras, Attila Sipos and Zsuzsanna Gyulai
Affiliation:
Keywords:
2-Alkoxyapomorphines, oripavine, acid-catalyzed rearrangement, O-demethylation, dopamine receptor binding affinity
Abstract: A novel synthetic route has been developed for the preparation of pharmacologically remarkable (R)- (-)-2-methoxyapomorphine (2) and other 2-alkoxyapomorphines 8-10.
