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[1]
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[http://dx.doi.org/10.1021/ja044996f] [PMID: 15547999]
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Qian, L.; Zhang, C-J.; Wu, J.; Yao, S.Q. Fused bicyclic caspase-1 inhibitors assembled by copper-free strain-promoted alkyne-azide cycloaddition (SPAAC). Chemistry, 2017, 23(2), 360-369.
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Kim, E.; Koo, H. Biomedical applications of copper-free click chemistry: in vitro, in vivo, and ex vivo. Chem. Sci. (Camb.), 2019, 10(34), 7835-7851.
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Barrow, A.S.; Smedley, C.J.; Zheng, Q.; Li, S.; Dong, J.; Moses, J.E. The growing applications of SuFEx click chemistry. Chem. Soc. Rev., 2019, 48(17), 4731-4758.
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[http://dx.doi.org/10.1039/C8CS00960K] [PMID: 31364998]
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Liu, Z.; Li, J.; Li, S.; Li, G.; Sharpless, K.B.; Wu, P. SuFEx click chemistry enabled late-stage drug functionalization. J. Am. Chem. Soc., 2018, 140(8), 2919-2925.
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Dai, H.; Huang, M.; Qian, J.; Liu, J.; Meng, C.; Li, Y.; Ming, G.; Zhang, T.; Wang, S.; Shi, Y.; Yao, Y.; Ge, S.; Zhang, Y.; Ling, Y. Excellent antitumor and antimetastatic activities based on novel coumarin/pyrazole oxime hybrids. Eur. J. Med. Chem., 2019, 166, 470-479.
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[http://dx.doi.org/10.1016/j.ejmech.2019.01.070] [PMID: 30739827]
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Sutanto, F.; Shaabani, S.; Oerlemans, R.; Eris, D.; Patil, P.; Hadian, M.; Wang, M.; Sharpe, M.E.; Groves, M.R.; Dömling, A. Combining high-throughput synthesis and high-throughput protein crystallography for accelerated hit identification. Angew. Chem. Int. Ed. Engl., 2021, 60(33), 18231-18239.
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Sutanto, F.; Shaabani, S.; Neochoritis, C.G.; Zarganes-Tzitzikas, T.; Patil, P.; Ghonchepour, E.; Dömling, A. Multicomponent reaction-derived covalent inhibitor space. Sci. Adv., 2021, 7(6), ,eabd9307.
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[http://dx.doi.org/10.1126/sciadv.abd9307] [PMID: 33536213]
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