Contents

Mini-Reviews in Medicinal Chemistry, Volume 4 - Number 6

Preface [Hot Topic: Arachidonic Acid Cascade Modulators: The Cyclooxygenase Pathway (Executive Editors: Jean-Michel Dogné / Xavier de Leval)]

, 4(6): i

Jean-Michel Dogne and Xavier de Leval


DOI: 10.2174/1389557043403774




First and Second Generations of COX-2 Selective Inhibitors

, 4(6): 597 - 601

Xavier de Leval, Fabien Julemont, Valerie Benoit, Michel Frederich, Bernard Pirotte and Jean-Michel Dogne


DOI: 10.2174/1389557043403693




Structural Approach for COX-2 Inhibition

, 4(6): 603 - 615

C. Michaux and C. Charlier


DOI: 10.2174/1389557043403756




The Second Generation of COX-2 Inhibitors: Clinical Pharmacological Point of View

, 4(6): 617 - 624

D. O. Stichtenoth


DOI: 10.2174/1389557043403783




COX-2 Selective Inhibitors, Carbonic Anhydrase Inhibition and Anticancer Properties of Sulfonamides Belonging to This Class of Pharmacological Agents

, 4(6): 625 - 632

Claudiu T. Supuran, Angela Casini, Antonio Mastrolorenzo and Andrea Scozzafava


DOI: 10.2174/1389557043403792




Recent Development in the Field of Dual COX / 5-LOX Inhibitors

, 4(6): 633 - 638

Fabien Julemont, Jean-Michel Dogne, Bernard Pirotte and Xavier de Leval


DOI: 10.2174/1389557043403747




Advance in Understanding the Biosynthesis of Prostacyclin and Thromboxane A2 in the Endoplasmic Reticulum Membrane via the Cyclooxygenase Pathway

, 4(6): 639 - 647

Ke-He Ruan


DOI: 10.2174/1389557043403710




New Developments on Thromboxane Modulators

, 4(6): 649 - 657

Jean-Michel Dogne, Julien Hanson, Xavier de Leval, Bernard Masereel, Philippe Kolh and Bernard Pirotte


DOI: 10.2174/1389557043403684




Modulation of the Arachidonic Cascade with ω3 Fatty Acids or Analogues: Potential Therapeutic Benefits

, 4(6): 659 - 668

Isabelle Roland, Xavier de Leval, Brigitte Evrard, Bernard Pirotte, Jean-Michel Dogne and Luc Delattre


DOI: 10.2174/1389557043403738




“Dipeptoids”: From the Chemical Structure of the Endogenous Peptide to the Design of Peptidomimetics

, 4(6): 669 - 680

Mercedes Martin-Martinez, Rosario Patino-Molina, M. Teresa Garcia-Lopez and Rosario Gonzalez-Muniz


DOI: 10.2174/1389557043403701




Predicting Synthetic Accessibility: Application in Drug Discovery and Development

, 4(6): 681 - 692

J. C. Baber and M. Feher


DOI: 10.2174/1389557043403765




The Development of Inhibitors of Heparanase, a Key Enzyme Involved in Tumour Metastasis, Angiogenesis and Inflammation

, 4(6): 693 - 702

Vito Ferro, Edward Hammond and Jon K. Fairweather


DOI: 10.2174/1389557043403729




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