Contents

Mini-Reviews in Medicinal Chemistry, Volume 4 - Number 3

Preface [Hot topic: New Insights in Protein Kinase Inhibitors: Chemogenomics, Phosphoproteomics, Structural Based Approaches and the Emergence of Resistance Executive Editor: Doriano Fabbro ]

, 4(3): i

Doriano Fabbro


DOI: 10.2174/1389557043487358




Kinase Chemogenomics: Targeting the Human Kinome for Target Validation and Drug Discovery

, 4(3): 235 - 253

E. ter Haar, W. P. Walters, S. Pazhanisamy, P. Taslimi, A. C. Pierce, G. W. Bemis, F. G. Salituro and S. L. Harbeson


DOI: 10.2174/1389557043487367




Targeting FLT3 Kinase in Acute Myelogenous Leukemia: Progress, Perils, and Prospects

, 4(3): 255 - 271

Michael C. Heinrich


DOI: 10.2174/1389557043487394




Therapeutically Targeted Anticancer Agents: Inhibitors of Receptor Tyrosine Kinases

, 4(3): 273 - 283

Carlos Garcia-Echeverria and Doriano Fabbro


DOI: 10.2174/1389557043487349




Imatinib (STI571) Resistance in Chronic Myelogenous Leukemia: Molecular Basis of the Underlying Mechanisms and Potential Strategies for Treatment

, 4(3): 285 - 299

Sandra W. Cowan-Jacob, Valerie Guez, Gabriele Fendrich, James D. Griffin, Doriano Fabbro, Pascal Furet, Janis Liebetanz, Jurgen Mestan and Paul W. Manley


DOI: 10.2174/1389557043487321




New Lead Generation Strategies for Protein Kinase Inhibitors - Fragment Based Screening Approaches

, 4(3): 301 - 311

Adrian Gill


DOI: 10.2174/1389557043487385




Exploring the Phosphoproteome with Mass Spectrometry

, 4(3): 313 - 324

Eric C. Peters, Ansgar Brock and Scott B. Ficarro


DOI: 10.2174/1389557043487330




The Emergence of Selective 5-HT2B Antagonists Structures, Activities and Potential Therapeutic Applications [General Reviews]

, 4(3): 325 - 330

G. Poissonnet, J. G. Parmentier, J. A. Boutin and S. Goldstein


DOI: 10.2174/1389557043487312




Small Molecule Antagonists of the Tachykinin NK2 Receptor [General Reviews]

, 4(3): 331 - 340

Daniela Fattori, Maria Altamura and Carlo Alberto Maggi


DOI: 10.2174/1389557043487376




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