Contents

Medicinal Chemistry, Volume 9 - Number 8

Graphical Abstract

Graphical Abstracts:

, 9(8): i - v


DOI: 10.2174/1573406411309080001




The Metabolism of Carbadox, Olaquindox, Mequindox, Quinocetone and Cyadox: An Overview

, 9(8): 1017 - 1027

Zhao-Ying Liu and Zhi-Liang Sun


DOI: 10.2174/1573406411309080002




Hemisynthesis of Selected Embelin Analogs and Investigation of their Proapoptotic Activity Against Cancer Cells

, 9(8): 1028 - 1034

Guillaume Viault, Katragadda Suresh Babu, Fabien Gautier, Sophie Barillé-Nion, Philippe Juin, Olivier Tasseau and René Grée


DOI: 10.2174/1573406411309080003




Synthesis and Inhibitory Effects of Some Novel 1,3-diarylprop-2-en-1-one Analogues in Foxp3 Expression: A Novel Class of Anti-cancer Candidates

, 9(8): 1035 - 1040

Mayank Kinger, Jeong Hoon Park, Min Goo Hur, Sang Wook Kim and Seung Dae Yang


DOI: 10.2174/15734064113099990029




The Evaluation of Multivariate Adaptive Regression Splines for the Prediction of Antitumor Activity of Acridinone Derivatives

, 9(8): 1041 - 1050

Marcin Koba and Tomasz Bączek


DOI: 10.2174/1573406411309080005




New Benzothiazole/thiazole-Containing Hydroxamic Acids as Potent Histone Deacetylase Inhibitors and Antitumor Agents

, 9(8): 1051 - 1057

Truong Thanh Tung, Dao Thi Kim Oanh, Phan Thi Phuong Dung, Van Thi My Hue, Sang Ho Park, Byung Woo Han, Youngsoo Kim, Jin-Tae Hong, Sang-Bae Han and Nguyen-Hai Nam


DOI: 10.2174/15734064113099990027




Synthesis and Anti-tumor Activity Evaluation of Gallic Acid-mangiferin Hybrid Molecule

, 9(8): 1058 - 1062

Xiang-yu Hu, Jia-gang Deng, Lin Wang and Ye-fei Yuan


DOI: 10.2174/1573406411309080007




Synthesis and in vitro Cytotoxicity Studies of Certain Novel Heterocycles Derived from Bis 1, 2, 4-Triazoles and their DNA Damage Studies

, 9(8): 1063 - 1072

Madhusudan N. Purohit, Chandrashekhar Venkaraddi Mangannavar and Mayur C. Yergeri


DOI: 10.2174/1573406411309080008




QSAR and Docking Based Semi-synthesis and in vitro Evaluation of 18 β-glycyrrhetinic Acid Derivatives Against Human Lung Cancer Cell Line A-549

, 9(8): 1073 - 1084

Dharmendra Kumar Yadav, Komal Kalani, Feroz Khan and Santosh Kumar Srivastava


DOI: 10.2174/1573406411309080009




Synthesis of 1H-1,2,3-triazoles and Study of their Antifungal and Cytotoxicity Activities

, 9(8): 1085 - 1090

Iara F. da Silva, Prisicila R.C. Martins, Emanuelly G. da Silva, Sabrina B. Ferreira, Vitor F. Ferreira, Karen Regina C. da Costa, Marne C. de Vasconcellos, Emerson S. Lima and Fernando de C. da Silva


DOI: 10.2174/1573406411309080010




Synthesis and Effects of Pyrazolines and Isoxazoles on the Phagocytic Chemotaxis and Release of Reactive Oxygen Species by Zymosan Stimulated Human Neutrophils

, 9(8): 1091 - 1098

Syed Nasir Abbas Bukhari, Ibrahim Jantan, Lam Kok Wai, Nordin Haji Lajis, Faridah Abbas and Malina Jasamai


DOI: 10.2174/1573406411309080011




Synthesis and Biological Evaluation of Some Novel Thieno[2,3-d] pyrimidine Derivatives as Potential Anti-inflammatory and Analgesic Agents

, 9(8): 1099 - 1112

Alaa A. El-Tombary, Soad A.M. El-Hawash, Nargues S. Habib, Raafat Soliman, Ibrahim M. El-Ashmawy and Omaima G. Shaaban


DOI: 10.2174/1573406411309080012




Design, Synthesis, and Bioactivity of Pyrazole Acid Derivatives as Endothelin Receptor Antagonists

, 9(8): 1113 - 1122

Jin Cai, Ligang Liu, Junqing Chen, Meng Cao and Min Ji


DOI: 10.2174/1573406411309080013




Effect of Stabilizers on Bioactivity of Peptide-24 in PLGA Microspheres

, 9(8): 1123 - 1128

Mingbo Wang, XiaoDong Guo, Rongwei Tan, Zhending She and Qingling Feng


DOI: 10.2174/1573406411309080014




Synthesis and in vitro Antibacterial Activity of 5-Halogenomethylsulfonyl- Benzimidazole and Benzotriazole Derivatives

, 9(8): 1129 - 1136

Zbigniew Ochal, Maria Bretner, Renata Wolinowska and Stefan Tyski


DOI: 10.2174/1573406411309080015




ACKNOWLEDGEMENT TO REVIEWERS:

, 9(8): 1137


DOI: 10.2174/1573406411309080016




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