Contents

Medicinal Chemistry, Volume 9 - Number 5

Graphical Abstracts:

, 9(5): i - v


DOI: 10.2174/1573406411309050001




Cinnamic Acid Derivatives Induce Cell Cycle Arrest in Carcinoma Cell Lines

, 9(5): 633 - 641

Matej Sova, Zeljko Zizak, Jelena A. Antic Stankovic, Matevz Prijatelj, Samo Turk, Zorica D. Juranic, Irena Mlinaric-Rascan and Stanislav Gobec


DOI: 10.2174/1573406411309050002




Structure Activity Relationship of Arylidene Pyrrolo and Pyrido [2,1-b] Quinazolones as Cytotoxic Agents: Synthesis, SAR Studies, Biological Evaluation and Docking Studies

, 9(5): 642 - 650

Veenu Mangla, Kunal Nepali, Gagandip Singh, Jagjeet Singh, Santosh Guru, Manish Kumar Gupta, Priya Mahajan, Ajit Kumar Saxena and Kanaya Lal Dhar


DOI: 10.2174/1573406411309050003




Synthesis, DNA Binding Ability and Anticancer Activity of 2-heteroaryl Substituted Benzimidazoles Linked Pyrrolo[2,1-c][1,4]benzodiazepine Conjugates

, 9(5): 651 - 659

Ahmed Kamal, Praveen Kumar Pogula, Mohammed Naseer Ahmed Khan, Bobburi Naga Seshadri and Kokkonda Sreekanth


DOI: 10.2174/1573406411309050004




Peptidomimetics as Potent and Selective PTP1B Inhibitors

, 9(5): 660 - 671

Dipam Patel, Mukul Jain, Shailesh R. Shah, Rajesh Bahekar, Pradip Jadav, Kiran Shah, Amit Joharapurkar, Mubeen Shaikh and Kalapatapu V.V.M. Sairam


DOI: 10.2174/1573406411309050005




Modified Silica Matrices for Controlled Release of Cephalexin

, 9(5): 672 - 680

María S. Legnoverde, Ignacio Jiménez-Morales, Alberto Jimenez-Morales, Enrique Rodriguez- Castellon and Elena I. Basaldella


DOI: 10.2174/1573406411309050006




Oxindole Derivatives: Synthesis and Antiglycation Activity

, 9(5): 681 - 688

Khalid Mohammed Khan, Momin Khan, Nida Ambreen, Muhammad Taha, Fazal Rahim, Saima Rasheed, Sumayya Saied, Humaira Shafi, Shahnaz Perveen and Muhammad Iqbal Choudhary


DOI: 10.2174/1573406411309050007




Structure-Activity Relationship for the Reactivators of Acetylcholinesterase Inhibited by Nerve Agent VX

, 9(5): 689 - 693

Kamil Kuca, Kamil Musilek, Daniel Jun, Jana Karasova, Ondrej Soukup, Jaroslav Pejchal and Martina Hrabinova


DOI: 10.2174/1573406411309050008




Synthesis and Evaluation of Substituted 4-methyl-2-oxo-2H-chromen-7-yl Phenyl Carbamates as Potent Acetylcholinesterase Inhibitors and Anti- Amnestic Agents

, 9(5): 694 - 702

Preet Anand and Baldev Singh


DOI: 10.2174/1573406411309050009




6-Acetyl-5H-thiazolo[3,2-a]pyrimidine Derivatives as the Novel Acetylcholinesterase Inhibitors: Design, Synthesis, and Biological Activity

, 9(5): 703 - 709

Hui Zhi, Can Zhang, Zhixin Cheng, Zhe Jin, Erfang Huang, Shuo Li, Huangquan Lin, David Chicheong Wan and Chun Hu


DOI: 10.2174/1573406411309050010




Synthesis, Characterization of (Z)-N-(1-(2-(2-amino-3-(dimethylamino) methyl)phenyl)-5-phenyl-1,3,4, oxadiazol-3(2H)-yl)ethanone Analogs as Potent Antimicrobial and Hydrogen Peroxide Scavenging Agents

, 9(5): 710 - 717

Manav Malhotra, Vikramdeep Monga, Rajiv Sharma, Kapendra Sahu, Gaurav Sharma, Jainendra Jain and Aakash Deep


DOI: 10.2174/1573406411309050011




Design, Synthesis and Molecular Docking Study of Some Substituted 4,5- dihydro-2H-indazole Derivatives as Potential Anti-inflammatory Agents

, 9(5): 718 - 730

Mona H. Badr, Rasha Y. Elbayaa and Ibrahim M. El-Ashmawy


DOI: 10.2174/1573406411309050012




3-Methyl-6-(prop-1-en-2-yl)cyclohex-3-ene-1,2-diol: the Importance of Functional Groups for Antiparkinsonian Activity

, 9(5): 731 - 739

Oleg V. Ardashov, Alla V. Pavlova, Dina V. Korchagina, Konstantin P. Volcho, Tat’ yana G. Tolstikova and Nariman F. Salakhutdinov


DOI: 10.2174/1573406411309050013




Synthesis and Evaluation of Water-Soluble Etoposide Esters of Malic Acid as Prodrugs

, 9(5): 740 - 747

Jing Chen and Wenting Du


DOI: 10.2174/1573406411309050014




Synthesis of Aminoalkoxy Substituted 4,5-Diphenylisoxazole Derivatives as Potential Anti-osteoporotic Agents

, 9(5): 748 - 755

Yeh-Long Chen, Chih-Hua Tseng, You-Chih Lo, Ru-Wei Lin, Chain-Fu Chen, Gwo-Jaw Wang, Mei-Ling Ho and Cherng-Chyi Tzeng


DOI: 10.2174/1573406411309050015




Antibacterial Activity of Phenyl Isothiocyanate on Escherichia coli and Staphylococcus aureus

, 9(5): 756 - 761

Ana Cristina Abreu, Anabela Borges, Lucia Chaves Simoes, Maria Jose Saavedra and Manuel Simoes


DOI: 10.2174/1573406411309050016




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