Medicinal Chemistry, Volume 9 - Number 3

Graphical Abstract

Graphical Abstracts

, 9(3): i - vi

DOI: 10.2174/1573406411309030001

Structural and Molecular Docking Studies of 4-Benzyl-3-[(1-methylpyrrol- 2-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one with Anticancer Activity

, 9(3): 313 - 328

Agnieszka A. Kaczor, Monika Pitucha, Zbigniew Karczmarzyk, Waldemar Wysocki, Jolanta Rzymowska and Dariusz Matosiuk

DOI: 10.2174/1573406411309030002

Synthesis, Topoisomerase I Inhibitory and Cytotoxic Activities of Chromone Derivatives

, 9(3): 329 - 339

Chirattikan Maicheen, Jiraphun Jittikoon, Opa Vajragupta and Jiraporn Ungwitayatorn

DOI: 10.2174/1573406411309030003

Design, Synthesis, and In vitro Antitumor Evaluation of Novel Phenylaminopyrimidine Derivatives

, 9(3): 340 - 350

Youguang Zheng, Ming Zheng, Yi Liu, Yunsheng Xue, Ling Zhang, Lin An, Ling Liu and Min Ji

DOI: 10.2174/1573406411309030004

Synthesis, Cytotoxicity, Antibacterial and Antileishmanial Activities of Imidazolidine and Hexahydropyrimidine Derivatives

, 9(3): 351 - 359

Gustavo S. G. de Carvalho, Rafael M. P. Dias, Fernando R. Pavan, Clarice Q. F. Leite, Vania L. Silva, Claudio G. Diniz, Daniela T. S. de Paula, Elaine S. Coimbra, Pascal Retailleau and Adilson D. da Silva

DOI: 10.2174/1573406411309030005

A Combination of 3D-QSAR Modeling and Molecular Docking Approach for the Discovery of Potential HIF Prolyl Hydroxylase Inhibitors

, 9(3): 360 - 370

Mahesh Kumar Teli and Rajanikant Golgodu Krishnamurthy

DOI: 10.2174/1573406411309030006

Synthesis, Molecular Docking and Antiamnesic Activity of Selected 2- Naphthyloxy Derivatives

, 9(3): 371 - 378

Poonam Piplani, Paramveer Singh and Anuradha Sharma

DOI: 10.2174/1573406411309030007

Synthesis and Antimalarial Activity Study of Some New Mannich Bases of 7-Chloro-4-Aminoquinoline

, 9(3): 379 - 383

Susanta Roy, Dipak Chetia, Mithun Rudrapal and Anil Prakash

DOI: 10.2174/1573406411309030008

Synthesis, Antifungal Activity, and Molecular Docking Studies of Novel Triazole Derivatives

, 9(3): 384 - 388

Nan Wang, Xiaoyun Chai, Ying Chen, Lei Zhang, Wenjuan Li, Yijun Gao, Yi Bi, Shichong Yu and Qingguo Meng

DOI: 10.2174/1573406411309030009

CoMFA and CoMSIA 3D QSAR Models for a Series of Some Condensed Thieno[2,3-d]pyrimidin-4(3H)-ones with Antihistaminic (H1) Activity

, 9(3): 389 - 401

Meenakshi Singh, Sushil K. Singh, Mahesh T. Chhabria, Kamala Vasu and Dhaivat Pandya

DOI: 10.2174/1573406411309030010

Modeling of LIM-Kinase 2 Inhibitory Activity of Pyrrolopyrimidine Analogues: Useful in Treatment of Ocular Hypertension and Glaucoma

, 9(3): 402 - 409

Gagandip Singh, Manish K. Gupta, Viney Kumar and Yenamandra S. Prabhakar

DOI: 10.2174/1573406411309030011

Quantitative Structure-Activity Relationship Study of Aromatic Inhibitors Against Rat Lens Aldose Reductase Activity Using Variable Selections

, 9(3): 410 - 419

Mankil Jung, Yongnam Lee, Minjoo Shim, Eunyoung Lim, Eun Jig Lee and Hyun Chul Lee

DOI: 10.2174/1573406411309030012

Insight into the Binding Mode between HIV-1 Integrase and Pyrimidone Analogue Inhibitors with MD Simulation and 3D-QSAR

, 9(3): 420 - 433

Songyao Ma, Wei Ye, Dingjue Ji and Hai-Feng Chen

DOI: 10.2174/1573406411309030013

Quantitative Structure-activity Relationships of Imidazole-containing Farnesyltransferase Inhibitors Using Different Chemometric Methods

, 9(3): 434 - 448

Ali Shayanfar, Saeed Ghasemi, Somaieh Soltani, Karim Asadpour-Zeynali, Robert J. Doerksen and Abolghasem Jouyban

DOI: 10.2174/1573406411309030014

Chondromodulating Chimeric Prodrugs of Diacetylrhein: Synthesis and Evaluation in Monoiodoacetate-induced Hyperalgesia

, 9(3): 449 - 458

Suneela Dhaneshwar and Dipmala Patil

DOI: 10.2174/1573406411309030015

Synthesis, Antifungal Evaluation and Molecular Docking Studies on 2- thioxoimidazolidin-4-one Derivatives

, 9(3): 459 - 473

Sudha Vengurlekar, Rajesh Sharma and Piyush Trivedi

DOI: 10.2174/1573406411309030016

Synthesis and QSAR Modeling of Novel Benzimidazolo Thiazolidinones, Thiazinones and 5-arylidene-2-imino Thiazolidinones as Antibacterial Agents

, 9(3): 474 - 485

Manjunath Ghate, Praveena Devi, Jignesh Parikh and Vivek K. Vyas

DOI: 10.2174/1573406411309030017

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