Contents

Medicinal Chemistry, Volume 9 - Number 3

Graphical Abstract

Graphical Abstracts

, 9(3): i - vi


DOI: 10.2174/1573406411309030001




Structural and Molecular Docking Studies of 4-Benzyl-3-[(1-methylpyrrol- 2-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one with Anticancer Activity

, 9(3): 313 - 328

Agnieszka A. Kaczor, Monika Pitucha, Zbigniew Karczmarzyk, Waldemar Wysocki, Jolanta Rzymowska and Dariusz Matosiuk


DOI: 10.2174/1573406411309030002




Synthesis, Topoisomerase I Inhibitory and Cytotoxic Activities of Chromone Derivatives

, 9(3): 329 - 339

Chirattikan Maicheen, Jiraphun Jittikoon, Opa Vajragupta and Jiraporn Ungwitayatorn


DOI: 10.2174/1573406411309030003




Design, Synthesis, and In vitro Antitumor Evaluation of Novel Phenylaminopyrimidine Derivatives

, 9(3): 340 - 350

Youguang Zheng, Ming Zheng, Yi Liu, Yunsheng Xue, Ling Zhang, Lin An, Ling Liu and Min Ji


DOI: 10.2174/1573406411309030004




Synthesis, Cytotoxicity, Antibacterial and Antileishmanial Activities of Imidazolidine and Hexahydropyrimidine Derivatives

, 9(3): 351 - 359

Gustavo S. G. de Carvalho, Rafael M. P. Dias, Fernando R. Pavan, Clarice Q. F. Leite, Vania L. Silva, Claudio G. Diniz, Daniela T. S. de Paula, Elaine S. Coimbra, Pascal Retailleau and Adilson D. da Silva


DOI: 10.2174/1573406411309030005




A Combination of 3D-QSAR Modeling and Molecular Docking Approach for the Discovery of Potential HIF Prolyl Hydroxylase Inhibitors

, 9(3): 360 - 370

Mahesh Kumar Teli and Rajanikant Golgodu Krishnamurthy


DOI: 10.2174/1573406411309030006




Synthesis, Molecular Docking and Antiamnesic Activity of Selected 2- Naphthyloxy Derivatives

, 9(3): 371 - 378

Poonam Piplani, Paramveer Singh and Anuradha Sharma


DOI: 10.2174/1573406411309030007




Synthesis and Antimalarial Activity Study of Some New Mannich Bases of 7-Chloro-4-Aminoquinoline

, 9(3): 379 - 383

Susanta Roy, Dipak Chetia, Mithun Rudrapal and Anil Prakash


DOI: 10.2174/1573406411309030008




Synthesis, Antifungal Activity, and Molecular Docking Studies of Novel Triazole Derivatives

, 9(3): 384 - 388

Nan Wang, Xiaoyun Chai, Ying Chen, Lei Zhang, Wenjuan Li, Yijun Gao, Yi Bi, Shichong Yu and Qingguo Meng


DOI: 10.2174/1573406411309030009




CoMFA and CoMSIA 3D QSAR Models for a Series of Some Condensed Thieno[2,3-d]pyrimidin-4(3H)-ones with Antihistaminic (H1) Activity

, 9(3): 389 - 401

Meenakshi Singh, Sushil K. Singh, Mahesh T. Chhabria, Kamala Vasu and Dhaivat Pandya


DOI: 10.2174/1573406411309030010




Modeling of LIM-Kinase 2 Inhibitory Activity of Pyrrolopyrimidine Analogues: Useful in Treatment of Ocular Hypertension and Glaucoma

, 9(3): 402 - 409

Gagandip Singh, Manish K. Gupta, Viney Kumar and Yenamandra S. Prabhakar


DOI: 10.2174/1573406411309030011




Quantitative Structure-Activity Relationship Study of Aromatic Inhibitors Against Rat Lens Aldose Reductase Activity Using Variable Selections

, 9(3): 410 - 419

Mankil Jung, Yongnam Lee, Minjoo Shim, Eunyoung Lim, Eun Jig Lee and Hyun Chul Lee


DOI: 10.2174/1573406411309030012




Insight into the Binding Mode between HIV-1 Integrase and Pyrimidone Analogue Inhibitors with MD Simulation and 3D-QSAR

, 9(3): 420 - 433

Songyao Ma, Wei Ye, Dingjue Ji and Hai-Feng Chen


DOI: 10.2174/1573406411309030013




Quantitative Structure-activity Relationships of Imidazole-containing Farnesyltransferase Inhibitors Using Different Chemometric Methods

, 9(3): 434 - 448

Ali Shayanfar, Saeed Ghasemi, Somaieh Soltani, Karim Asadpour-Zeynali, Robert J. Doerksen and Abolghasem Jouyban


DOI: 10.2174/1573406411309030014




Chondromodulating Chimeric Prodrugs of Diacetylrhein: Synthesis and Evaluation in Monoiodoacetate-induced Hyperalgesia

, 9(3): 449 - 458

Suneela Dhaneshwar and Dipmala Patil


DOI: 10.2174/1573406411309030015




Synthesis, Antifungal Evaluation and Molecular Docking Studies on 2- thioxoimidazolidin-4-one Derivatives

, 9(3): 459 - 473

Sudha Vengurlekar, Rajesh Sharma and Piyush Trivedi


DOI: 10.2174/1573406411309030016




Synthesis and QSAR Modeling of Novel Benzimidazolo Thiazolidinones, Thiazinones and 5-arylidene-2-imino Thiazolidinones as Antibacterial Agents

, 9(3): 474 - 485

Manjunath Ghate, Praveena Devi, Jignesh Parikh and Vivek K. Vyas


DOI: 10.2174/1573406411309030017




Webmaster Contact: info@benthamscience.org
Copyright © 2018 Bentham Science