Contents

Medicinal Chemistry, Volume 9 - Number 1

Graphical Abstract

Graphical Abstracts

, 9(1): i - vi


DOI: 10.2174/157340641130901000i




Foreword

, 9(1): vii

Atta-ur-Rahman


DOI: 10.2174/1573406411309010vii




Synthesis and Opioid Activity of Novel 6-ketolevorphanol Derivatives

, 9(1): 1 - 10

Zsuzsanna Gyulai, Antal Udvardy, Attila Cs. Bényei, Jakub Fichna, Katarzyna Gach, Martin Storr, Géza Tóth, Sándor Antus, Sándor Berényi, Anna Janecka and Attila Siposa


DOI: 10.2174/1573406411309010001




Syntheses, DNA Binding and Anticancer Profiles of L-Glutamic Acid Ligand and its Copper(II) and Ruthenium(III) Complexes

, 9(1): 11 - 21

Imran Ali, Waseem A. Wani, Kishwar Saleem and Diana Wesselinova


DOI: 10.2174/1573406411309010011




Identification of Structural and Electronic Features for a Series of MCH1R Antagonists

, 9(1): 22 - 31

Danielle C. Silva, Adriano D. Andricopulo, Emmanuela F. de Lima and Káthia M. Honório


DOI: 10.2174/1573406411309010022




Predicting the Activity of Antimicrobial Peptides with Amino Acid Topological Information

, 9(1): 32 - 44

Mao Shu, Rui Yu, Yunru Zhang, Juan Wang, Li Yang, Li Wang and Zhihua Lin


DOI: 10.2174/1573406411309010032




Design, Synthesis and Antimicrobial Properties of Novel 3,3a,4,5,6,7- Hexahydroindazole and Arylthiazolylpyrazoline Derivatives

, 9(1): 45 - 52

Abha Bishnoi, Suruchi Singh, Anil K. Tiwari, Arun Sethi and Chandrakant Mani Tripathi


DOI: 10.2174/1573406411309010045




Synthesis, Antimycobacterial, Antiviral, Antimicrobial Activity and QSAR Studies of N2-acyl isonicotinic Acid Hydrazide Derivatives

, 9(1): 53 - 76

Vikramjeet Judge, Balasubramanian Narasimhan, Munish Ahuja, Dharmarajan Sriram, Perumal Yogeeswari, Erik De Clercq, Christophe Pannecouque and Jan Balzarini


DOI: 10.2174/1573406411309010053




Novel 2-hydrazino-pyrimidin-4(3H)-one Derivatives with Pseudofunctional- Similarity to Siderophores as Potential Antimycobacterial Agents

, 9(1): 77 - 83

Ranjeet Bairwa, Nilesh R. Tawari, Amruta Alate, Swapnil Anam, Mariam S. Degani, Muktikant Ray and Ramakrishna M. G. Rajan


DOI: 10.2174/1573406411309010077




5-Arylidene-4-Thiazolidinone Derivatives Active as Antidegenerative Agents on Human Chondrocyte Cultures

, 9(1): 84 - 90

Annamaria Panico, Rosanna Maccari, Venera Cardile, Lucia Crascì, Simone Ronsisvalle and Rosaria Ottanà


DOI: 10.2174/1573406411309010084




Synthesis, p38 Kinase Inhibitory and Anti-inflammatory Activity of New Substituted Benzimidazole Derivatives

, 9(1): 91 - 99

Ravindra G. Kulkarnia, Stefan A. Laufer, Chandrashekhar V. M and Achaiah Garlapati


DOI: 10.2174/1573406411309010091




Novel C-9, 9'-O-acyl Esters of (-)-Carinol as Free-radical Scavengers and Xanthine Oxidase Enzyme Inhibitors: Synthesis and Biological Evaluation

, 9(1): 100 - 103

Praveen Kumar Suryadevara, Hari Babu Tatipaka, Rama Subba Rao Vidadala, Ashok k Tiwari, Janaswamy Madhusudana Rao and Katragadda Suresh Babu


DOI: 10.2174/1573406411309010100




Design, Synthesis and In-vivo Hypoglycemic Evaluation of Novel Non - TZD’S in a Type - 2 Diabetic Model

, 9(1): 104 - 111

Rupali Jadhav, Ranu Gupta-Rajoria, Tanushree Pal and Ramaa Chelakara Subramanian


DOI: 10.2174/1573406411309010104




Synthesis and In-vitro Photodynamic Studies of the Superparamagnetic Chitosan Hydrogel/Chlorin E6 Nanocarriers

, 9(1): 112 - 117

Mohammad Reza Saboktakin, Roya M. Tabatabaie, Fahimeh Satarzade Amini, Abel Maharramov and Mohammad Ali Ramazanov


DOI: 10.2174/1573406411309010112




Synthesis and Biological Evaluation of Novel Pentacyclic Triterpene Derivatives as Potential PPARγ Agonists

, 9(1): 118 - 125

Liying Zhang, Jizhe Dong, Jun Liu, Luyong Zhang, Lingyi Kong, Hequan Yao and Hongbin Sun


DOI: 10.2174/1573406411309010118




Discovering the Binding Modes of Natural Products with Histone Deacetylase 1

, 9(1): 126 - 132

Lei Zhang, Minyong Li, Lihui Zhang and Wenfang Xu


DOI: 10.2174/1573406411309010126




Prediction of Allergenic Proteins by Means of the Concept of Chou’s Pseudo Amino Acid Composition and a Machine Learning Approach

, 9(1): 133 - 137

Hassan Mohabatkara, Majid Mohammad Beigib, Kolsoum Abdolahic and Sasan Mohsenzadeh


DOI: 10.2174/1573406411309010133




Exploring the Biological Potential of Urea Derivatives Against mPGES-1: A Combination of Quantum Mechanics, Pharmacophore Modelling and QSAR Analyses

, 9(1): 138 - 151

Malkeet Singh Bahia and Om Silakari


DOI: 10.2174/1573406411309010138




QSAR and Pharmacophore Study of Dyrk1A Inhibitory Meridianin Analogs as Potential Agents for Treatment of Neurodegenerative Diseases

, 9(1): 152 - 161

Sandip B. Bharate, Rammohan R. Yadav and Ram A. Vishwakarma


DOI: 10.2174/1573406411309010152




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