Contents

Medicinal Chemistry, Volume 8 - Number 6

Selective Inhibition of Inducible Nitric Oxide Synthase by Derivatives of Acetamidine

, 8(6): 991 - 995

Cristina Maccallini, Antonia Patruno, Alessandra Ammazzalorso, Barbara De Filippis, Marialuigia Fantacuzzi, Sara Franceschelli, Letizia Giampietro, Simona Masella, Maria Luisa Tricca and Rosa Amoroso


DOI: 10.2174/1573406411208060991


Transient Injury-Dependent Up-Regulation of CD105 and its Specific Targeting with an Anti-Vascular Anti-Mouse Endoglin-Nigrin b Immunotoxin

, 8(6): 996 - 1002

Raquel Munoz, Yolanda Arias, Jose Miguel Ferreras, Pilar Jimenez, Maria Angeles Rojo, Carmelo Bernabeu, Damian Cordoba-Diaz and Tomas Girbes


DOI: 10.2174/1573406411208060996



Synthesis, SAR and Biological Evaluation of Natural and Non-natural Hydroxylated and Prenylated Xanthones as Antitumor Agents

, 8(6): 1012 - 1025

Xiaojin Zhang, Xiang Li, Suofu Ye, Yu Zhang, Lei Tao, Yuan Gao, Dandan Gong, Meiyang Xi, Huyan Meng, Mingqian Zhang, Wenlei Gao, Xiaoli Xu, Qinglong Guo and Qidong You


DOI: 10.2174/1573406411208061012



Impact of Clozapine, N-Desmethylclozapine and Chlorpromazine on Thromboxane Production in Vitro

, 8(6): 1032 - 1038

Hubertus Himmerich, Luise Schmidt, Susen Becker, Linda Kortz, Jeremias Schonherr, Roland Mergl, Katrin Bauer, Ulrich Sack, Abigail J. Sheldrick, Joachim Thiery and Uta Ceglarek


DOI: 10.2174/1573406411208061032


Synthesis and Biological Evaluation of New Sulfonamide Derivatives as Potential Anti-Trypanosoma cruzi Agents

, 8(6): 1039 - 1044

Virgilio Bocanegra-Garcia, Juan Carlos Villalobos-Rocha, Benjamin Nogueda-Torres, Maria Edith Lemus- Hernandez, Argelia Camargo-Ordonez, Ninfa Maria Rosas-Garcia and Gildardo Rivera


DOI: 10.2174/1573406411208061039


Molecular Features for Antitrypanosomal Activity of Thiosemicarbazones Revealed by OPS-PLS QSAR Studies

, 8(6): 1045 - 1056

Norka Beatriz Huaman Lozano, Vinicius Goncalves Maltarollo, Karen Cacilda Weber, Kathia Maria Honorio, Rafael Victorio Carvalho Guido, Adriano Defini Andricopulo and Alberico Borges Ferreira Da Silva


DOI: 10.2174/1573406411208061045









3D QSAR Pharmacophore Modeling for c-Met Kinase Inhibitors

, 8(6): 1117 - 1125

Dandan Huang, Xiaoyun Zhu, Chunlei Tang, Yicheng Mei, Wei Chen, Baowei Yang, Jing Han, Hai Qian and Wenlong Huang


DOI: 10.2174/1573406411208061117




Looking for New Targets: Simple Coumarins as Antibacterial Agents

, 8(6): 1140 - 1145

Maria Joao Matos, Saleta Vazquez-Rodriguez, Lourdes Santana, Eugenio Uriarte, Cristina Fuentes-Edfuf, Ysabel Santos and Angeles Munoz-Crego


DOI: 10.2174/1573406411208061140


New Cathepsin D Inhibitor Library Utilizing Hydroxyethyl Isosteres with Cyclic Tertiary Amines

, 8(6): 1146 - 1154

Rose M. McConnell, Kalyani Inapudi, Naveen Kadasala, Karthika Yarlagadda, Priya Velusamy, Matthew S. McConnell, Adam Green, Carol Trana, Kelley Sayyar and James S. McConnell


DOI: 10.2174/1573406411208061146


In Silico Prediction of Novel Inhibitors of the DNA Binding Activity of FoxG1

, 8(6): 1155 - 1162

Syam Bhuvanachandran Nair, Shaik Mahammad Abdul Fayaz and Rajanikant Golgodu Krishnamurthy


DOI: 10.2174/1573406411208061155


Evaluating the Diagnostic and Chemotherapeutic Potential of Vancomycin- Derived Imaging Conjugates

, 8(6): 1163 - 1170

Sumbla Sheikh, Alexander Sturzu, Uwe Klose, Hartmut Echner, Martin Deeg, Thomas Nagele, Marius Horger, Christian Schwentner, Ulrike Ernemann, Wolfgang Voelter and Stefan Heckl


DOI: 10.2174/1573406411208061163



Description of High Purity and High Specific Activity of [11C]Choline Synthesis Using TRACERlab FXc Module, and Detailed Report of Quality Controls

, 8(6): 1182 - 1189

Giorgio Biasiotto, Francesco Bertagna, Ugo Biasiotto, Carlo Rodella, Giovanni Bosio, Luigi Caimi, Giovanni Bettinsoli and Raffaele Giubbini


DOI: 10.2174/1573406411208061182




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