Contents

Medicinal Chemistry, Volume 7 - Number 6

Analysis of the α-Glucosidase Inhibitory Activity of Chromenone Derivatives Based on their Molecular Features: A Computational Study

, 7(6): 526 - 533

N. S. Hari Narayana Moorthy, Maria J. Ramos and Pedro A. Fernandes


DOI: 10.2174/157340611797928389




Synthesis and Bioactivities of 2-Azetidinone Derivatives as Cholesterol Absorption Inhibitors

, 7(6): 534 - 542

Yubin Wang, Hai Qian, Jinpei Zhou, Huibin Zhang, Jianfeng Ji and Wenlong Huang


DOI: 10.2174/157340611797928271




3D-QSAR of Novel Phosphodiesterase-4 Inhibitors by Genetic Function Approximation

, 7(6): 543 - 552

Anand V. Raichurkar, Ujashkumar A. Shah and Vithal M. Kulkarni


DOI: 10.2174/157340611797928352




A QSAR Study on Some Series of HIV-1 Integrase Inhibitors

, 7(6): 553 - 560

Shikha Kaushik, Satya P. Gupta, P. K. Sharma and Zaihra Anwar


DOI: 10.2174/157340611797928361




Syntheses of 2,3-Diarylated 2H-Benzo[e][1,2]Thiazine 1,1-Dioxides and their 3,4-Dihydro Derivatives, and Assessment of their Inhibitory Activity Against MCF-7 Breast Cancer Cells

, 7(6): 561 - 571

Yuan-Yuan Shan, Cheng-Mei Zhang, Long-Qiang Tang, Zhao-Peng Liu, Nicole R. Bearss, Jeffrey G. Sarver, Amarjit Luniwal and Paul W. Erhardt


DOI: 10.2174/157340611797928307




Synthesis of 2,4,6-Trichlorophenyl Hydrazones and their Inhibitory Potential Against Glycation of Protein

, 7(6): 572 - 580

Khalid Mohammed Khan, Zarbad Shah, Viqar Uddin Ahmad, Momin Khan, Muhammad Taha, Fazal Rahim, Humera Jahan, Shahnaz Perveen and M. Iqbal Choudhary


DOI: 10.2174/157340611797928415




Pharmacophoric Modeling and Atom-Based 3D-QSAR of Novel 1-Aryl-3-(1-acylpiperidin-4-yl) Urea as Human Soluble Epoxide Hydrolase Inhibitors (sEHIs)

, 7(6): 581 - 592

Nirupam Das, Meenakshi Dhanawat, Akanksha Kulshrestha and Sushant K. Shrivastava


DOI: 10.2174/157340611797928479




Synergism from Combination of Cisplatin and Multicentred Platinums Coded as DH6Cl and TH1 in the Human Ovarian Tumour Models

, 7(6): 593 - 598

Ali Alshehri, Philip Beale, Jun Qing Yu and Fazlul Huq


DOI: 10.2174/157340611797928316




Synthesis and Antitumoral Evaluation of 7-chloro-4-quinolinylhydrazones Derivatives

, 7(6): 599 - 604

Raquel Carvalho Montenegro, Leticia Veras Lotufo, Manoel Odorico de Moraes, Claudia do O Pessoa, Felipe Augusto Rocha Rodrigues, Marcelle de Lima Ferreira Bispo, Laura Nogueira de Faria Cardoso, Carlos Roland Kaiser and Marcus Vinicius Nora de Souza


DOI: 10.2174/157340611797928299




Novel 3-(2-(3-methyl-5-substituted-phenyl-4,5-dihydropyrazol-1-yl)-2-oxoethoxy)-2-substituted-phenyl-4H-chromen-4-one: Synthesis and Anticancer Activity

, 7(6): 605 - 610

Xin-Hua Liu, Jun Li, Fan-Rong Wu, Bao-An Song, Pinaki S. Bhadury and Lei Shi


DOI: 10.2174/157340611797928442




Synthesis and Antitubercular Activity of New L-serinyl Hydrazone Derivatives

, 7(6): 611 - 623

Alessandra Campbell Pinheiro, Carlos Roland Kaiser, Thais Cristina Mendonca Nogueira, Samir Aquino Carvalho, Edson Ferreira da Silva, Larisse de Oliveira Feitosa, Maria das Gracas Muller de Oliveira Henriques, Andre Luis Peixoto Candea, Maria Cristina Silva Lourenco and Marcus Vinicius Nora de Souza


DOI: 10.2174/157340611797928325




Design, Synthesis and Antitumor Activity of Novel D-Glucuronic Acid Derivatives

, 7(6): 624 - 638

Ahmed O. H. El-Nezhawy, Frady G. Adly, Ahmed F. Eweas, Atef G. Hanna, Yehya M. El-Kholy, Shahenaz H. El-Syed and Tarek B. A. El-Naggar


DOI: 10.2174/157340611797928398




Free Radical Scanvenging and Antioxidant Effects of Some Anthraquinone Derivatives

, 7(6): 639 - 644

Abderrahmane Baghiani, Noureddine Charef, Meriem Djarmouni, Haythem A. Saadeh, Lekhmici Arrar and Mohammad S. Mubarak


DOI: 10.2174/157340611797928424




MIA-QSAR Coupled to Different Regression Methods for the Modeling of Antimalarial Activities of 2-aziridinyl and 2,3-bis-(aziridinyl)-1,4-naphtoquinonyl Sulfate and Acylate Derivatives

, 7(6): 645 - 654

Mohammad Goodarzi and Matheus P. Freitas


DOI: 10.2174/157340611797928343




In silico Designing and Screening of Lead Compounds to NS5-Methyltransferase of Dengue Viruses

, 7(6): 655 - 662

Dakshinamurthy Sivakumar and Thirunavukkarasu Sivaraman


DOI: 10.2174/157340611797928451




Synthesis of Novel 8-Hydroxy Quinolin Based 1,3,4-oxadiazoles and S-substituted 1,2,4-triazole Derivatives and Evaluation of their Anti-inflammatory, Analgesic, Ulcerogenic and Anti-Microbial Activities

, 7(6): 663 - 673

Mohammad Mahboob Alam, Mohammad Shaharyar, Hinna Hamid, Syed Nazreen, Saqlain Haider and Mohammad Sarwar Alam


DOI: 10.2174/157340611797928334




Antibacterial Activity of Thyme and Lavender Essential Oils

, 7(6): 674 - 689

Monika Sienkiewicz, Monika Lysakowska, Julita Ciecwierz, Pawel Denys and Edward Kowalczyk


DOI: 10.2174/157340611797928488




Antimicrobial Activity and SAR Study of Some Novel Thiosemicarbazide Derivatives Bearing Piperidine Moiety

, 7(6): 690 - 696

Agata Siwek and Joanna Stefanska


DOI: 10.2174/157340611797928406




Synthesis, Structure and Antibacterial Evaluation of Some N-substituted 3-amino-5-hydroxy-4-phenyl-1H-pyrazole-1-carboxamides

, 7(6): 697 - 703

Monika Pitucha, Urszula Kosikowska, Liliana Urszula and Anna Malm


DOI: 10.2174/157340611797928433




Synthesis and in vitro Leishmanicidal Activity of Disulfide Derivatives

, 7(6): 704 - 710

Khalid Mohammed Khan, Muhammad Taha, Farzana Naz, Momin Khan, Fazal Rahim, Samreen, Shahnaz Perveen and M. Iqbal Choudhary


DOI: 10.2174/157340611797928460




Novel Hexahydropyridoindole Derivative as Prospective Agent Against Oxidative Damage in Pancreatic βCells

, 7(6): 711 - 717

Lucia Rackova, Ahmet Cumaoglu, E. Umit Bagrιacιk, Milan Stefek, Pierre Maechler and Cimen Karasu


DOI: 10.2174/157340611797928370




Cloning, Expression and Characterization of Mouse (Mus musculus) Nicotinamide 5-Mononucleotide Adenylyltransferase-2

, 7(6): 718 - 726

David W. Raches, Suhong Xiao, Praveen Kusumanchi, Joel Yalowitz, Paresh Sanghani, Eric C. Long, Asok C. Antony and Hiremagalur N. Jayaram


DOI: 10.2174/157340611797928262




Synthesis and Evaluation of Biological Activities of a Series of (6-substitutedbenzothiazol-2-yl)acrylamides

, 7(6): 727 - 731

Nguyen-Hai Nam, Phan Thi Phuong Dung, Doan Thanh Hieu, Le Hoang, Tran Thi Hien, Tran The Cuong and Phan Dinh Chau


DOI: 10.2174/157340611797928280




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