Contents

Medicinal Chemistry, Volume 4 - Number 5

Synthesis and Antimalarial Activity of New Amino Analogues of Amodiaquine

, 4(5): 407 - 425

E. Paunescu, S. Susplugas, E. Boll, R. A. Varga, E. Mouray, P. Grellier and P. Melnyk


DOI: 10.2174/157340608785700153




Dihydroethanoanthracene Derivatives Reverse In Vitro Quinoline Resistance in Plasmodium falciparum Malaria

, 4(5): 426 - 437

Maud Henry, Sandrine Alibert, Meili Baragatti, Joel Mosnier, Eric Baret, Remy Amalvict, Eric Legrand, Thierry Fusai, Jacques Barbe, Christophe Rogier, Jean-Marie Pages and Bruno Pradines


DOI: 10.2174/157340608785700234




N,N-Bis(trifluoromethylquinolin-4-yl)diamino Alkanes: Synthesis and Antimalarial Activity

, 4(5): 438 - 445

Joseph L. Kgokong, Gilbert M. Matsabisa, Peter P. Smith and Jaco C. Breytenbach


DOI: 10.2174/157340608785700216




Synthesis and Antimalarial Activity of Novel Side Chain Modified Antimalarial Agents Derived from 4-Aminoquinoline

, 4(5): 446 - 456

V. Raja Solomon, W. Haq, M. Smilkstein, Kumkum Srivastava, S. Rajakumar, Sunil K. Puri and S. B. Katti


DOI: 10.2174/157340608785700207




Synthesis of 2-Methyl N10-Substituted Acridones as Selective Inhibitors of Multidrug Resistance (MDR) Associated Protein in Cancer Cells

, 4(5): 457 - 465

Y. C. Mayur, Osman Ahmad, V. V.S. Rajendra Prasad, M. N. Purohit, N. Srinivasulu and S. M. Shanta Kumar


DOI: 10.2174/157340608785700180




Synthesis and Evaluation of 1-Benzhydryl-sulfonyl-piperazine Derivatives as Inhibitors of Tumor Growth and Tumor Angiogenesis of Mouse Ehrlich Ascites Tumor In Vivo

, 4(5): 466 - 472

C. S. Ananda Kumar, H. Chandru, A. C. Sharada, N. R. Thimmegowda, S. B. Benaka Prasad, M. Karuna Kumar and K. S. Rangappa


DOI: 10.2174/157340608785700171




Dibenzoylmethane Activates Nrf2-Dependent Detoxification Pathway and Inhibits Benzo(a)pyrene Induced DNA Adducts in Lungs

, 4(5): 473 - 481

R. K. Thimmulappa, T. Rangasamy, J. Alam and S. Biswal


DOI: 10.2174/157340608785700199




Synthesis, Antimycobacterial Activities and Phototoxic Evaluation of 5H-thiazolo[3,2-a]quinoline-4-carboxylic Acid Derivatives

, 4(5): 482 - 491

Murugesan Dinakaran, Palaniappan Senthilkumar, Perumal Yogeeswari, Arnab China, Valakunja Nagaraja and Dharmarajan Sriram


DOI: 10.2174/157340608785700225




Synthesis and Biological Evaluation of Naphthalene-1,4-dione Derivatives as Potent Antimycobacterial Agents

, 4(5): 492 - 497

A. Mital, V. S. Negi and U. Ramachandran


DOI: 10.2174/157340608785700243




Structure-Activity Relationship Study of a Series of N-Substituted Piperazinyl-Fluoroquinolones as Anti-Helicobacter pylori Agents

, 4(5): 498 - 502

A. Foroumadi, M. Safavi, S. Emami, F. Siavoshi, S. Najjari, F. Safari and A. Shafiee


DOI: 10.2174/157340608785700162




Synthesis of N3-Substituted Thymidine Analogues for Measurement of Cellular Kinase Activity

, 4(5): 503 - 512

P. Ghosh, A. Pal, A. Shavrin, W. Bornmann, J. G. Gelovani and M. M. Alauddin


DOI: 10.2174/157340608785700252




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