Contents

Medicinal Chemistry, Volume 4 - Number 1

Synthesis and Pharmacological Evaluation of 4-Phenoxy-1,2,3,4- Tetrahydroisoquinolines and 4,5,6,6a-Tetrahydrochromeno [2,3,4-de]isoquinolines

, 4(1): 1 - 10

G. Giorgioni, S. Ruggieri, F. Claudi, A. Di Stefano, E. Ljung and T. Carlsson


DOI: 10.2174/157340608783331506




Insight into the Bioreductive Mode of Action of Antitrypanosomal 5- Nitrofuryl Containing Thiosemicarbazones

, 4(1): 11 - 17

D. Gambino, L. Otero, J. D. Maya, A. Morello, C. Rigol, G. Barriga, J. Rodriguez, C. Folch, E. Norambuena, M. Gonzalez, C. Olea Azar and H. Cerecetto


DOI: 10.2174/157340608783331470




Synthesis, Molecular Docking and PTP1B Inhibitory Activity of Functionalized 4,5-Dihydronaphthofurans and Dibenzofurans

, 4(1): 18 - 24

Atul Goel, Manish Dixit, Uzma Saeed, Amit Kumar, Mohammad Imran Siddiqi, Akhilesh K. Tamrakar and Arvind K. Srivastava


DOI: 10.2174/157340608783331515




Synthesis and Theoretical Calculations of 5-Aminosalicylic Acid Derivatives as Potential Analgesic Agents

, 4(1): 25 - 29

Trujillo-Ferrara Jose, Correa-Basurto Jose, M. C. Rosales-Hernandez, Ramirez-San Juan Eduardo, Badillo Abigail, Z. Gomez-Castro Carlos and L. H. Fabila-Castillo


DOI: 10.2174/157340608783331489




Estimation of Human Carbonic Anhydrase II Inhibition Using Topological Indices and their Combination with Quantum-Theoretical Descriptors

, 4(1): 30 - 66

Padmakar V. Khadikar, Jyoti Singh, Shalini Singh, Rajika Mishra, Claudiu T. Supuran, Brian W. Clare and Meenakshi Lakhwani


DOI: 10.2174/157340608783331461




Studies on the Structure-Activity Relationship of the Basic Amine of Phenylpiperazines as Melanocortin-4 Receptor Antagonists

, 4(1): 67 - 74

Chen Chen, Joe A. Tran, Melissa Arellano, Beth A. Fleck, Joseph Pontillo, Dragan Marinkovic, Fabio C. Tucci, Jenny Wen and John Saunders


DOI: 10.2174/157340608783331498




HIV Protease Inhibitors Impact on Apoptosis

, 4(1): 75 - 79

Stacey A. Rizza and Andrew D. Badley


DOI: 10.2174/157340608783331443




Simulation of Sequential Screening Experiments Using Emerging Chemical Patterns

, 4(1): 80 - 90

Jurgen Bajorath and Jens Auer


DOI: 10.2174/157340608783331452




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