Contents

Medicinal Chemistry, Volume 3 - Number 6

Synthesis and Biological Evaluation of 2-amino-3-(3, 4, 5-trimethoxyphenylsulfonyl)-5-aryl thiophenes as a New Class of Antitubulin Agents

, 3(6): 507 - 512

Romeo Romagnoli, Pier Giovanni Baraldi, Vincent Remusat, Maria Dora Carrion, Carlota Lopez Cara, Olga Cruz-Lopez, Delia Preti, Francesca Fruttarolo, Mojgan Aghazadeh Tabrizi, Jan Balzarini and Ernest Hamel


DOI: 10.2174/157340607782360380




Design, Synthesis and Biological Evaluation of a Series of Thioamides as Non-Nucleoside Reverse Transcriptase Inhibitors

, 3(6): 513 - 519

Ahmed S. Mehanna, Jitendra D. Belani, Charles J. Kelley and Luke A. Pallansch


DOI: 10.2174/157340607782360344




Synthesis and Anti-Picornaviridae In Vitro Activity of a New Class of Helicase Inhibitors the N,N-bis[4-(1H(2H)-benzotriazol-1(2)-yl)phenyl] alkyldicarboxamides

, 3(6): 520 - 532

A. Carta, M. Loriga, S. Piras, G. Paglietti, M. Ferrone, M. Fermeglia, S. Pricl, P. La Colla, G. Collu, T. Sanna and R. Loddo


DOI: 10.2174/157340607782360308




Design, Synthesis and Pharmacological Evaluation of HIV-1 Reverse Transcriptase Inhibition of New Indolin-2-Ones

, 3(6): 533 - 542

Nubia Boechat, W. Bruce Kover, Vera Bongertz, Monica M. Bastos, Nelilma C. Romeiro, Maria L.G. Azevedo and Wagner Wollinger


DOI: 10.2174/157340607782360326




The Preparation and Human Muscarinic Receptor Profiling of Oxybutynin and N-Desethyloxybutynin Enantiomers

, 3(6): 543 - 545

Allen B. Reitz, Suneel K. Gupta, Yifang Huang, Michael H. Parker and Richard R. Ryan


DOI: 10.2174/157340607782360353




A Salicylic Acid-Based Analogue Discovered from Virtual Screening as a Potent Inhibitor of Human 20α-Hydroxysteroid Dehydrogenase

, 3(6): 546 - 550

Urmi Dhagat, Vincenzo Carbone, Roland P.-T. Chung, Toshihiro Matsunaga, Satoshi Endo, Akira Hara and Ossama El-Kabbani


DOI: 10.2174/157340607782360399




Synthesis of 1,2,4-triazole Derivatives: Binding Properties on Endothelin Receptors

, 3(6): 551 - 560

L. Salerno, F. Guerrera, M. Modica, G. Romeo, V. Pittala, M. A. Siracusa, I. Mereghetti, A. Cagnotto and T. Mennini


DOI: 10.2174/157340607782360281




Design and Synthesis of New N-OMe Fluoro-Indole Melatoninergics

, 3(6): 561 - 571

A. Tsotinis, J. Gourgourinis, A. Eleutheriades, K. Davidson and D. Sugden


DOI: 10.2174/157340607782360335




New Steroidal Anti-Inflammatory Antedrugs: 21-Thioalkylether Derivatives of Methyl 16-Prednisolone Carboxylates

, 3(6): 572 - 575

M. Omar F. Khan, Kwan K. Park, Sharye N. Glynn and Henry J. Lee


DOI: 10.2174/157340607782360317




Computational Approach to Drug Design for Oxazolidinones as Antibacterial Agents

, 3(6): 576 - 582

Yun Li, Dong-Qing Wei, Wei-Na Gao, Hui Gao, Bing-Ni Liu, Chang-Jiang Huang, Wei-Ren Xu, Deng-Ke Liu, Hai-Feng Chen and Kuo-Chen Chou


DOI: 10.2174/157340607782360362




Synthesis of Opioidmimetics, 3-[H-Dmt-NH(CH2)m]-6-[H-Dmt-NH(CH2)n]-2(1H)-pyrazinones, and Studies on Structure-Activity Relationships

, 3(6): 583 - 598

Kimitaka Shiotani, Anna Miyazaki, Tingyou Li, Yuko Tsuda, Toshio Yokoi, Akihiro Ambo, Yusuke Sasaki, Sharon D. Bryant, Yunden Jinsmaa, Lawrence H. Lazarus and Yoshio Okada


DOI: 10.2174/157340607782360272




In Vitro Binding Receptors Study by Valeriana adscendens, Iresine herbstii and Brugmansia arborea Extracts

, 3(6): 599 - 604

Anna Capasso and Vincenzo De Feo


DOI: 10.2174/157340607782360290




Peptide-Based Soft Materials as Potential Drug Delivery Vehicles

, 3(6): 605 - 611

Sandeep Verma, K. B. Joshi and Surajit Ghosh


DOI: 10.2174/157340607782360371




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