Contents

Medicinal Chemistry, Volume 2 - Number 4

Design, Synthesis and In Vitro Evaluation of 4-Androstene-3,17-dione/Adenosine Hybrid Compounds as Bisubstrate Inhibitors of Type 3 17β-Hydroxysteroid Dehydrogenase

, 2(4): 329 - 347

Marie Berube, Yannick Laplante and Donald Poirier


DOI: 10.2174/157340606777724086




New Substrate Analogue Inhibitors of Factor Xa Containing 4-Amidinobenzylamide as P1 Residue: Part 1

, 2(4): 349 - 361

Torsten Steinmetzer, Jorg Sturzebecher, Oliver Schuster, Uta Sturzebecher, Andrea Schweinitz and Anne Sturzebecher


DOI: 10.2174/157340606777724040




Classical QSAR Study on Chromene Derivatives as Lanosterol 14α -Demethylase Inhibitor: A Non Azole Antifungal Target

, 2(4): 363 - 367

S. G. Kaskhedikar, M. A. Babu, M. Lakshmi and P. Vasanthanathan


DOI: 10.2174/157340606777724004




Medicinal Chemistry of Probimane and MST-16: Comparison of Anticancer Effects Between Bisdioxopiperazines

, 2(4): 369 - 375

Bin Xu, Jian Ding, Hong Zhu, Cheng-Hui Xu, Min Huang and Da-Yong Lu


DOI: 10.2174/157340606777724095




Cytoprotective Effects of 5 Benzophenones and a Xanthone from Hypericum annulatum in Models of Epirubicin-Induced Cytotoxicity: SARAnalysis and Mechanistic Investigations

, 2(4): 377 - 384

Margarita Karaivanova, Ulrich Girreser, Tzvetomira Tzanova, Gerassim M. Kitanov, Dimitrina Zh.Zheleva-Dimitrova, Paraskev T. Nedialkov and Georgi Momekov


DOI: 10.2174/157340606777724103




Physico-Chemical Profiling of Antidepressive Sertraline: Solubility,Ionisation, Lipophilicity

, 2(4): 385 - 389

Karoly Tihanyi, Bela Noszal, Krisztina Takacs-Novak and Katalin Deak


DOI: 10.2174/157340606777723997




Cyclosporin-A in the Treatment of Nephrotic Syndrome: The Importance of Monitoring C0 (Trough) and C2 (Two Hours After its Administration) Blood Levels

, 2(4): 391 - 393

John G. Vlachojannis, Irene Savidaki, Pantelitsa Kalliakmani, Sotiris Tsakas and D. S. Goumenos


DOI: 10.2174/157340606777724068




A Novel Family of Minimal PMRI Cyclic Peptides as Versatile Scaffolds for Generating New Molecular Topology

, 2(4): 395 - 400

Cristina Tiozzo, Federico Squassabia, Alessandra Tolomelli, Luca Gentilucci and Giuliana Cardillo


DOI: 10.2174/157340606777724077




Molecular Interactions Between Human Cytochrome P450 1A2 and Flavone Derivatives

, 2(4): 401 - 406

Maria Joao Ramos, Francesco Iori, Maria Cristina Menziani, Andre Melo and Rute da Fonseca


DOI: 10.2174/157340606777723988




Folic Acid as a Fenton-modulator: Possible Physiological Implication

, 2(4): 407 - 413

Subrata Chattopadhyay, Birija S. Patro, Soumyakanti Adhikari and Tulsi Mukherjee


DOI: 10.2174/157340606777724059




The Structure - Antituberculosis Activity Relationships Study in a Series of 5-(4-Aminophenyl)-4-Substituted-2,4-Dihydro-3h-1,2,4-Triazole-3-Thione Derivatives. A Combined Electronic-Topological and Neural Networks Approach

, 2(4): 415 - 422

Fatma Kandemirli, Nathali Shvets, Seda Unsalan, Ilkay Kucukguzel, Sevim Rollas, Vasyl Kovalishyn and Anatholy Dimoglo


DOI: 10.2174/157340606777724013




Does the Septic Shock Interfere Experimental Acute Pancreatitis in Rats?

, 2(4): 423 - 429

S. Hac, M. Dobosz, J. J. Kaczor, S. Dobrowolski, J. Krajewski, R. Rzepko, Z. Gruca and Z. Sledzinski


DOI: 10.2174/157340606777724031




Retinoids in Clinical Use

, 2(4): 431 - 438

Vincent C. O. Njar, Lalji Gediya, Puranik Purushottamachar, Panka Chopra, Aashvini Belosay and Jyoti B. Patel


DOI: 10.2174/157340606777724022




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