Contents

Medicinal Chemistry, Volume 12 - Number 7


Research Article

Synthesis, Cytotoxic Activity on Leukemia Cell Lines and Quantitative Structure-Activity Relationships (QSAR) Studies of Morita-Baylis-Hillman Adducts

, 12(7): 602 - 612

Claudio G. Lima–Junior, Gláucia V. Faheina–Martins, Caio C. B. Bomfim, Bruna B. Dantas, Everton P. Silva, Demetrius A. M. de Araújo, Edilson B. A. Filho and Mário L. A. A. Vasconcellos


DOI: 10.2174/1573406412666160506150924



Research Article

Integrated In Silico-In Vitro Discovery of Lung Cancer-related Tumor Pyruvate Kinase M2 (PKM2) Inhibitors

, 12(7): 613 - 620

Xiangyun Ye, Yinjia Sun, Yunhua Xu, Zhiwei Chen and Shun Lu


DOI: 10.2174/1573406412666160307151535



Research Article

Design, Synthesis, and Cytotoxicity of Novel 2,4,6-Trisubstituted 1,3,5- triazines Bearing Aryl Hydrazone Moiety as Potent Antitumor Agent

, 12(7): 621 - 630

Limei Wang, Sijia Zhao, Guanglong Bao, Yu Zhang, Shuancheng Xi, Guolin Zhou, Xin Zhai and Ping Gong


DOI: 10.2174/1573406412666160106154551



Research Article

Synthesis and Biological Evaluation of Novel 1,3,4-thiadiazole Derivatives Incorporating Benzisoselenazolone Scaffold as Potential Antitumor Agents

, 12(7): 631 - 639

Xiaoyun Fu, Sha Li, Fen Jing, Xuefeng Wang, Baolin Li, Jijun Zhao, Yuming Liu and Baoquan Chen


DOI: 10.2174/1573406412666160201120806



Research Article

Synthesis and Antifungal Activity of Some 4,6-Dimethylisoxazolo[3,4- b]pyridin-3(1H)-one Derivatives

, 12(7): 640 - 646

Jaroslaw Saczewski, Joanna Fedorowicz, Anna Kedzia, Marta Ziolkowska-Klinkosz and Aleksandra Jalinska


DOI: 10.2174/1573406412666160517122925



Research Article

Synthesis of Cyclic Imides (Methylphtalimides, Carboxylic Acid Phtalimides and Itaconimides) and Evaluation of their Antifungal Potential

, 12(7): 647 - 654

Dorimar Stiz, Rogério Corrêa, Felicia D. D'Auria, Giovanna Simonetti and Valdir Cechinel-Filho


DOI: 10.2174/1573406412666160229150833



Research Article

Antiplasmodial Limonoids from Trichilia rubescens (Meliaceae)

, 12(7): 655 - 661

Tsamo T. Armelle, Nangmo K. Pamela, Mkounga Pierre, Ingrid B. Müller, Kirk Marat, Gabriele Sass and Nkengfack A. Ephrem


DOI: 10.2174/1573406412666160106154357



Research Article

Three Arachidonoylamide Derivatives Inhibit Pro-Inflammatory Genes Expression by Modulating NF-κB and AP1 Activities

, 12(7): 662 - 673

Alex Gregorelli, Anna Sgarbossa, Shahbaz Khan, Annunziata Soriente, Margherita De Rosa, Carmela Saturnino and Marta Menegazzi


DOI: 10.2174/1573406412666160502154936



Research Article

Synthesis, in vivo Anticoagulant Evaluation and Molecular Docking Studies of Bicoumarins Obtained from Furocoumarin Peucedanin

, 12(7): 674 - 683

Alla V. Lipeeva, Mikhail V. Khvostov, Dmitry S. Baev, Makhmut M. Shakirov, Tatijana G. Tolstikova and Elvira E. Shults


DOI: 10.2174/1573406412666160129105115



Research Article

Biologically Active New N, N', N''-Tri-Substituted Ferrocenyl Phenylguanidines and their Characterization

, 12(7): 684 - 698

Rukhsana Gul, Ataf A. Altaf, Amin Badshah, Afzal Shah, Zia ur Rehman, Rabia Naz, Muhammad N. Tahir and Asif Junaid


DOI: 10.2174/1573406412666160129104817




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