Contents

Medicinal Chemistry, Volume 11 - Number 1



Synthesis and First Evaluation of [18F]Fluorocyano- and [18F]Fluoronitroquinoxalinedione as Putative AMPA Receptor Antagonists

, 11(1): 13 - 20

Sebastian Olma, Johannes Ermert, Wiebke Sihver and Heinz H. Coenen


DOI: 10.2174/1573406410666140428151318



Preparation, In Vitro Screening and Molecular Modelling of Monoquaternary Compounds Related to the Selective Acetylcholinesterase Inhibitor BW284c51

, 11(1): 21 - 29

Ondrej Benek, Kamil Musilek, Anna Horova, Vlastimil Dohnal, Rafael Dolezal and Kamil Kuca


DOI: 10.2174/1573406410666140428153110



N-Valproyl-L-Phenylalanine as New Potential Antiepileptic Drug: Synthesis, Characterization and In Vitro Studies on Stability, Toxicity and Anticonvulsant Efficacy

, 11(1): 30 - 40

Viviana De Caro, Anna Lisa Scaturro, Flavia Maria Sutera, Giuseppe Avellone, Gabriella Schiera, Evelina Ferrantelli, Maria Carafa, Valerio Rizzo, Fabio Carletti, Pierangelo Sardo and Libero Italo Giannola


DOI: 10.2174/1573406410666140507094954



Synthesis, Anticonvulsant and Antimicrobial Activities of Some New [1-(2-Naphthyl)-2-(pyrazol-1-yl)ethanone]oxime Ethers

, 11(1): 41 - 49

Zeynep Ozdemir, Arzu Karakurt, Unsal Calis, Selami Gunal, Samil Isik, Z. Sibel Sahin and Sevim Dalkara


DOI: 10.2174/1573406410666140428150358



Synthesis of New Thiazolo[4,5-d]pyrimidines as Corticotropin Releasing Factor Modulators

, 11(1): 50 - 59

Bhimanna Kuppast, Katerina Spyridaki, Christophina Lynch, Yueshan Hu, George Liapakis, Gareth E. Davies and Hesham Fahmy


DOI: 10.2174/1573406410666140724115627



Antiglycation Activity of Quinoline Derivatives- A New Therapeutic Class for the Management of Type 2 Diabetes Complications

, 11(1): 60 - 68

Bilquees Bano, Sanaullah Abbasi, Jalaluddin A. J. Khan, Shafqat Hussain, Saima Rasheed, Shahnaz Perveen, Khalid Mohammed Khan and M. Iqbal Choudhary


DOI: 10.2174/1573406410666140526151254



Synthesis and Evaluation of Anti-inflammatory and Analgesic Activities of New 1,2,4-triazole Derivatives

, 11(1): 69 - 76

Fatemeh Ahmadi, Mohsen Rezayan Ghayahbashi, Mohammad Sharifzadeh, Eskandar Alipoiur, Seyed Nasser Ostad, Mohsen Vosooghi, Hamid Reza khademi and Mohsen Amini


DOI: 10.2174/1573406410666140613154507



Electronic-Topological and Neural Network Approaches to the Structure- Antimycobacterial Activity Relationships Study On Hydrazones Derivatives

, 11(1): 77 - 85

Fatma Kandemirli, Can Dogan Vurdu, Murat Alper Basaran, Hakan Sezgin Sayiner, Nathaly Shvets, Anatholy Dimoglo, Vasyl Kovalish and Turgay Polat


DOI: 10.2174/1573406410666140428144334



Functionalization of Tetracycline and Evaluation of Its Antibacterial Activity Including Against Resistant Bacteria

, 11(1): 86 - 93

Priyanka Dogra and Ghanshyam S. Chauhan


DOI: 10.2174/1573406410666140507094435



Seeds of Peganum Harmala L. Chemical Analysis, Antimalarial and Antioxidant Activities, and Cytotoxicity Against Human Breast Cancer Cells

, 11(1): 94 - 101

Naziha Chabir, Hany Ibrahim, Mehrez Romdhane, Alexis Valentin, Beatrice Moukarzel, Mohamed Mars and Jalloul Bouajila


DOI: 10.2174/1573406410666140613152434




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