Contents

Medicinal Chemistry, Volume 10 - Number 1

Graphical Abstract

Graphical Abstracts

, 10(1): i - iv


DOI: 10.2174/157340641001131226100523




Foreword

, 10(1): 1

Atta-ur-Rahman


DOI: 10.2174/157340641001131226101323




Bioavailability of Endomorphins and the Blood-brain Barrier- A Review

, 10(1): 2 - 17

Renata Perlikowska and Anna Janecka


DOI: 10.2174/15734064113099990040




Ramoplanin Imaging Conjugates – Synthesis and Evaluation

, 10(1): 18 - 26

Sumbla Sheikh, Alexander Sturzu, Hubert Kalbacher, Uwe Klose, Thomas Nagele, Bushra Amin, Martin Deeg, Marius Horger, Ulrike Ernemann and Stefan Heckl


DOI: 10.2174/157340641001131226121133




Anti-Neoplastic Activity of 1,3-Diaza-2-Functionalized-Adamantan-6-One Compounds Against Melanoma Cells

, 10(1): 27 - 37

Yifat Sharabi-Ronen, Shlomo Levinger, Miri Ben-Dahan Lellouche and Amnon Albeck


DOI: 10.2174/15734064113099900002




Design, Synthesis and Biological Evaluation of Novel Non-peptide Boronic Acid Derivatives as Proteasome Inhibitors

, 10(1): 38 - 45

Jiankang Zhang, Luqing Shen, Jincheng Wang, Peihua Luo and Yongzhou Hu


DOI: 10.2174/15734064113099990006




Structural Elucidation of Unique Inhibitory Activities of Two Thiazolo[ 4,5-d]pyrimidines Against Epidermal Growth Factor Receptor (EGFR): Implications for Successful Drug Design

, 10(1): 46 - 58

Petar M. Mitrasinovic


DOI: 10.2174/157340641001131226122124




Effect of Stilbene and Chalcone Scaffolds Incorporation in Clofibric Acid on PPARα Agonistic Activity

, 10(1): 59 - 65

Letizia Giampietro, Alessandra D’Angelo, Antonella Giancristofaro, Alessandra Ammazzalorso, Barbara De Filippis, Mauro DiMatteo, Marialuigia Fantacuzzi, Pasquale Linciano, Cristina Maccallini and Rosa Amoroso


DOI: 10.2174/157340641001131226123613




Computer-aided Design, Synthesis, and Biological Evaluation of 5- Substituted Aminomethylenepyrimidine-2,4,6-Triones as H1 Antihistaminic Agents (Part2)

, 10(1): 66 - 73

Rasha Y. Elbayaa


DOI: 10.2174/15734064113099990032




Alkyl Caffeates as Anti-Helicobacter Pylori and Scavenger of Oxidants Produced by Neutrophils

, 10(1): 74 - 80

Luana Chiquetto Paracatu, Cibele Bonacorsi, Carolina Maria Quinello Gomes de Farias, Ana Carolina Nazaré, Maicon Segalla Petrônio, Luiz Octávio Regasini, Dulce Helena Siqueira Silva, Maria Stella Gonçalves Raddi, Luiz Marcos da Fonseca and Valdecir Farias Ximenes


DOI: 10.2174/157340641001131226125042




Ligustrazine Derivatives. Part 8: Design, Synthesis, and Preliminary Biological Evaluation of Novel Ligustrazinyl Amides as Cardiovascular Agents

, 10(1): 81 - 89

Zhenyu Li, Fang Yu, Lei Cui, Wenmin Chen, Shouxun Wang, Peng Zhan, Yuemao Shen and Xinyong Liu


DOI: 10.2174/157340641130900042




Approaches to a Multitargeting Drug Development: First Profiled 3- Ethoxycarbonyl-1-aza-9-oxafluorenes Representing a Perspective Compound Class Targeting Alzheimer Disease Relevant Kinases CDK1, CDK5 and GSK-3 β

, 10(1): 90 - 97

Andreas Hilgeroth, Volkmar Tell, Steffi Kramer, Frank Totzke and Christoph Schachtele


DOI: 10.2174/157340641001131226141606




A Comprehensive Ligand Based Mapping of the σ2 Receptor Binding Pocket

, 10(1): 98 - 121

Derek J. Rhoades, David H. Kinder and Tarek M. Mahfouz


DOI: 10.2174/1573406409999131119103621




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