Articles Ahead of Print

Synthesis and Structural Elucidation of Novel Benzothiazole Derivatives as Anti-tubercular Agents: In-silico Screening for Possible Target Identification


Katharigatta N. Venugopala*, Sandeep Chandrashekharappa, Melendhran Pillay, Subhrajyoti Bhandary, Mahmoud Kandeel, Fawzi M. Mahomoodally , Mohamed A. Morsy, Deepak Chopra , Bandar E. Aldhubiab, Mahesh Attimarad, Osama I. Alwassil , Sree Harsha and Koleka Mlisana


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Neuropharmacological Screening of Chiral and Non-chiral Phthalimide- Containing Compounds in Mice: in vivo and in silico Experiments


Carolina Campos-Rodriguez, Jose G. Trujillo-Ferrara*, Ameyali Alvarez-Guerra, Iran M. Cumbres Vargas, Roberto I. Cuevas-Hernandez, Erik Andrade-Jorge, Sergio Zamudio and Eduardo Ramirez-San Juan*


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Synthesis and Biological Evaluation of Novel 2,3-disubstituted Benzofuran Analogues of GABA as Neurotropic Agents


Arturo Coaviche-Yoval, Hector Luna, Ricardo Tovar-Miranda, Marvin Antonio Soriano-Ursua and Jose G. Trujillo-Ferrara*


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Novel Hydroxamic Acids Incorporating 1-((1H-1,2,3-Triazol-4-yl)methyl)- 3-substituted-2-oxoindolines: Synthesis, Biological Evaluation and SAR Analysis


Do Thi Mai Dung, Nguyen Van Huan, Do Manh Cam, Dao Cam Hieu, Pham-The Hai, Le-Thi-Thu Huong, Jisung Kim, Jeong Eun Choi, Jong Soon Kang, Sang-Bae Han* and Nguyen-Hai Nam*


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The Evaluation of Metal Co-ordinating Bis-Thiosemicarbazones as Potential Anti-malarial Agents


Fady N. Akladios, Scott D. Andrew, Samantha J. Boog, Carmen de Kock, Richard K. Haynes and Christopher J. Parkinson*


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2-Oxo-1,2,3,4-tetrahydropyrimidines as Potent β-Glucuronidase Inhibitors: One-pot Synthesis, In vitro and In silico Studies


Sarosh Iqbal*, Nimra Naveed Shaikh, Khalid Mohammed Khan*, Sehrish Naz, Zaheer Ul-Haq Qasmi, Shahnaz Perveen and M. Iqbal Choudhary*


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Pyrano[3,2-c]quinoline Derivatives as New Class of α-glucosidase Inhibitors to Treat Type 2 Diabetes: Synthesis, in vitro Biological Evaluation and Kinetic Study


Zahra Heydari, Maryam Mohammadi-Khanaposhtani, Somaye Imanparast, Mohammad Ali Faramarzi, Mohammad Mahdavi *, Parviz Rashidi Ranjbar* and Bagher Larijani


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4-Hydroxy-2-pyridone Derivatives and the δ-pyrone Isostere as Novel Agents Against Mycobacterium smegmatis Biofilm Inhibitors


Maheshkumar R. Borkar, Santosh Nandan*, M N Harish Kumar , Jayashree Puttur, M Jisha , Dipankar Chatterji and Evans C. Coutinho *


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Design, Synthesis and Biological Evaluation of 1H-1,2,3-Triazole-Linked- 1H


Carolina S. Bortolot, Luana da S. M. Forezi, Roberta K. F. Marra, Marcelo I. P. Reis, Barbara V. F. e Sa, Ricardo Imbroisi Filho, Zeinab Ghasemishahrestani, Mauro Sola-Penna, Patricia Zancan, Vitor F. Ferreira* and Fernando de C. da Silva*


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Design, Synthesis and Investigation of New Diphenyl Substituted Pyridazinone Derivatives as Both Cholinesterase and Aβ-Aggregation Inhibitors


Burcu Kilic, Merve Erdogan, Hayrettin O. Gulcan, Fatma Aksakal, Nihan Oruklu, E. Umit Bagriacik and Deniz S. Dogruer*


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Exploration of (hetero)aryl Derived Thienylchalcones for Antiviral and Anticancer Activities


Vikrant Patil, Siddappa A. Patil*, Renukadevi Patil, Alejandro Bugarin, Kenneth Beaman and Shivaputra A. Patil*


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Antimicrobial Evaluation of Erythrinan Alkaloids from Erythrina cristagalli L.


Janaina M. de Avila, Ionara I. Dalcol*, Alessandra O. Pereira, Eveline W. Santos, Adriano Ferraz, Maura Z. Santos, Marco Aurelio Mostardeiro and Ademir F. Morel


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Sorbinil, an Aldolase Reductase Inhibitor, in Fighting Against Diabetic Complications


Qi Huang, Qiong Liu and Dongsheng Ouyang*


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Synthesis of Nucleosides and Non-nucleosides Based 4,6-disubstituted-2- oxo-dihydropyridine-3-carbonitriles as Antiviral Agents


Tarek S. Ibrahim, Hassan A. El-Sayed, Maan T. Khayat, Amany M.M. AL-Mahmoudy, Ahmed H. Moustafa, Ayat K. Saad El-Deen, Sherif A.F. Rostom and Siva S. Panda*


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Crystal Structure of Mistletoe Lectin I (ML-I) from Viscum album in Complex with 4-N-Furfurylcytosine at 2.85 Å Resolution


Malik Shoaib Ahmad*, Saima Rasheed, Sven Falke, Binish Khaliq, Markus Perbandt, M. Iqbal Choudhary, Wojciech T. Markiewicz, Jan Barciszewski and Christian Betzel*


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Pyrazole and imidazo[1,2-b]pyrazole Derivatives as New Potential Antituberculosis Agents


Elda Meta, Chiara Brullo*, Michele Tonelli, Scott G. Franzblau, Yuehong Wang, Rui Ma, Wan Baojie , Beatrice Silvia Orena, Maria Rosalia Pasca and Olga Bruno


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Synthetic Diethyl 2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylates Induce Apoptosis


Seunghyun Ahn, Youngshim Lee, Jihyun Park, Junho Lee, Soon Young-Shin, Young Han Lee, Dongsoo Koh* and Yoongho Lim*


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Synthesis and Biological Evaluation of 12N-substituted Tricyclic Matrinic Derivatives as a Novel Family of Anti-Influenza Agents


Sheng Tang, Yu-Huan Li , Xin–Yue Cheng, Jin–Qiu Yin , Ying–Hong Li , Dan–Qing Song , Yan–Xiang Wang * and Zhan–Dong Liu


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Identification of New Chromenone Derivatives as Cholinesterase Inhibitors and Molecular Docking Studies


Jamshed Iqbal *, Muhammad Shakeel Ahmad Abbasi, Sumera Zaib , Saifullah Afridi, Norbert Furtmann, Jurgen Bajorath and Peter Langer


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