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Endorsements

"Medicinal Chemistry is an invaluable journal, which contains the latest outstanding developments in medicinal chemistry. It is recommended to all scientists working in this field."

Michael Kassiou
University of Sydney, Australia

Authors' Comments
Thank you for your mail. I am very delighted to be the author of this article in your esteemed journal (Medicinal Chemistry, Bentham science publishers ). Glad to say that the quality of your service is very nice. I will surely contribute new research publication to this esteemed journal soon.

Sreekanth Thota
(National Institute for Science and Technology on Innovation on Neglected Diseases (INCT/IDN), Center for Technological Development in Health (CDTS), Fiocruz, Rio de Janeiro, Brazil)


Medicinal Chemistry

,

Volume 14

-

Number 4



Biography   Open Access





Research Article

The Synthesis of Chalcones as Anticancer Prodrugs and their Bioactivation in CYP1 Expressing Breast Cancer Cells

, 14(4): 322 - 332

Ketan C. Ruparelia*, Keti Zeka, Taeeba Ijaz, Dyan N. Ankrett, Nicola E. Wilsher, Paul C. Butler, Hoon L. Tan, Sabahat Lodhi, Avninder S. Bhambra, Gerard A. Potter, Randolph R.J. Arroo and Kenneth J.M. Beresford


DOI: 10.2174/1573406414666180112120134






Research Article





Research Article





Research Article





Research Article

Synthesis and in vitro Antioxidant Activity Study of Some Novel Substituted Piperazinyl Flavone Compounds

, 14(4): 372 - 386

Elmas Sari, Pawel Berczynski, Aleksandra Kladna, Irena Kruk, Oya Bozdag Dundar, Monika Szymanska and Hassan Y. Aboul-Enein*


DOI: 10.2174/1573406414666171204105000






Research Article

A Novel Method to Synthesize Phosphocreatine and Phosphocreatine Prodrugs

, 14(4): 387 - 393

Maria Arkel, Patrizia Garbati, Annalisa Salis, Gianluca Damonte, Nara Liessi, Enrico Adriano, Umberto Benatti, Maurizio Balestrino and Enrico Millo*


DOI: 10.2174/1573406413666171120164702






Research Article

Activity of Rifabutin and Hemi-synthetic Derivatives Against Mycobacterium abscessus

, 14(4): 394 - 399

Ivy B. Ramis*, Ricardo Figueiredo, Daniela F. Ramos, Priscila C.B. Halicki, Andrea von Groll, Miguel Viveiros, Maria do Ceu Costa and Pedro E.A. da Silva


DOI: 10.2174/1573406414666171204102633






Design of Bactericidal Peptides Against Escherichia coli O157:H7, Pseudomonas aeruginosa and methicillin-resistant Staphylococcus aureus


Jenniffer Cruz, Paola Rondon , Rodrigo Torres, Mauricio Urquiza, Fanny Guzman, Claudio Alvarez, Maria Angeles Abengozar, Daniel A. Sierra, Luis Rivas, Roberto Fernandez-Lafuente and Claudia Ortiz*


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Synthetic Diethyl 2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylates Induce Apoptosis


Seunghyun Ahn, Youngshim Lee, Jihyun Park, Junho Lee, Soon Young-Shin, Young Han Lee, Dongsoo Koh* and Yoongho Lim*


View Abstract View on PubMed


Synthesis and Antibacterial Activity Against MRSA of Pleuromutilin Derivatives Possessing a Mercaptoethylamine Linker


Zhao-Sheng Zhang, Yun-Zhen Huang, Jian Luo, Bing-Feng Wang, Zhen Jin, Ya-Hong Liu and You-Zhi Tang*


View Abstract View on PubMed


Evaluation of Trypanocidal and Antioxidant Activities of a Selected Series of 3-amidocoumarins


Mauricio Moncada-Basualto, Michel Lapier, Juan Diego Maya, Betty Matsuhiro, Claudio Olea-Azar*, Giovanna L. Delogu, Eugenio Uriarte, Lourdes Santana and Maria Joao Matose


View Abstract View on PubMed


Diclofenac 1,3,4-Oxadiazole Derivatives; Biology-Oriented Drug Synthesis (BIODS) in Search of Better Non-Steroidal, Non-Acid Antiinflammatory Agents


Shazia Shah, Arshia, Nida Siraj Kazmi, Almas Jabeen, Aisha Faheem, Nida Dastagir, Tariq Ahmed, Khalid Mohammed Khan*, Shakil Ahmed, Abeer Raza and Shahnaz Perveen


View Abstract View on PubMed


Benzoin Schiff Bases: Design, Synthesis, and Biological Evaluation as Potential Antitumor Agents


Dima A. Sabbah*, Fatima Al-Tarawneh, Wamidh H. Talib, Kamal Sweidan, Sanaa K. Bardaweel, Eveen Al-Shalabi, Haizhen A. Zhong, Ghassan Abu Sheikha, Reema Abu Khalaf and Mohammad S. Mubarak


View Abstract View on PubMed


Construction of an M1GS Ribozyme for Targeted and Rapid mRNA Cleavage; Application on the Ets-2 Oncogene


Chrisavgi Toumpeki, Dimitrios Anastasakis, Ioannis Panagoulias, Vassiliki Stamatopoulou, Tassos Georgakopoulos, Sofia Kallia-Raftopoulos, Athanasia Mouzaki* and Denis Drainas*


View Abstract View on PubMed


2-Oxo-1,2,3,4-tetrahydropyrimidines as potent β-Glucuronidase Inhibitors: One-pot Synthesis, In vitro and In silico Studies


Sarosh Iqbal*, Nimra Naveed Shaikh, Khalid Mohammed Khan*, Sehrish Naz, Zaheer-Ul-Haq Qasmi , Shahnaz Perveen and M. Iqbal Choudhary*


View Abstract


Neuropharmacological screening of chiral and non-chiral phthalimidecontaining compounds in mice: in vivo and in silico experiments


Carolina Campos-Rodriguez, Jose G. Trujillo-Ferrara*, Ameyali Alvarez-Guerra, Iran M. Cumbres Vargas, Roberto I. Cuevas-Hernandez, Erik Andrade-Jorge, Sergio Zamudio and Eduardo Ramirez-San Juan*


View Abstract


4-Hydroxy-2-pyridone derivatives and the δ-pyrone isostere as novel agents against Mycobacterium smegmatis biofilm inhibitors


Maheshkumar R. Borkar, Santosh Nandan*, M N Harish Kumar , Jayashree Puttur, M Jisha , Dipankar Chatterji and Evans C. Coutinho *


View Abstract


Crystal Structure of Mistletoe Lectin I (ML-I) from Viscum album in Complex with 4-N-Furfurylcytosine at 2.85 Å Resolution


Malik Shoaib Ahmad*, Saima Rasheed, Sven Falke, Binish Khaliq, Markus Perbandt, M. Iqbal Choudhary, Wojciech T. Markiewicz, Jan Barciszewski and Christian Betzel*


View Abstract


Synthesis and biological evaluation of novel 2,3-disubstituted benzofuran analogues of GABA as neurotropic agents


Arturo Coaviche-Yoval, Hector Luna, Ricardo Tovar-Miranda, Marvin Antonio Soriano-Ursua and Jose G. Trujillo-Ferrara*


View Abstract


Inhibition of Mutated Isocitrate Dehydrogenase 1 in Cancer


Fangrui Wu, Gang Cheng, Yuan Yao, Mari Kogiso, Hong Jiang, Xiao-Nan Li and Yongcheng Song*


View Abstract


Pyrazole and imidazo[1,2-b]pyrazole derivatives as new potential anti-tuberculosis agents


Elda Meta, Chiara Brullo*, Michele Tonelli, Scott G. Franzblau, Yuehong Wang, Rui Ma, Wan Baojie , Beatrice Silvia Orena, Maria Rosalia Pasca and Olga Bruno


View Abstract


Antimicrobial evaluation of erythrinan alkaloids from Erythrina crista-galli L.


Janaina M. de Avila, Ionara I. Dalcol*, Alessandra O. Pereira, Eveline W. Santos, Adriano Ferraz, Maura Z. Santos, Marco Aurelio Mostardeiro and Ademir F. Morel


View Abstract


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