Contents

Letters in Drug Design & Discovery, Volume 9 - Number 5

Graphical Abstracts

, 9(5): i - v


DOI: 10.2174/157018012800389278




Synthesis of Phenanthroindolizidine Alkaloids with an Acyloxy Group at the C3 Position and their Antitumor Activities and Toxicities

, 9(5): 447 - 453

Takashi Ikeda, Takashi Yaegashi, Takeshi Matsuzaki, Ryuta Yamazaki, Satoshi Ueno, Syusuke Hashimoto and Seigo Sawada


DOI: 10.2174/157018012800389232




An Efficient One Pot Three Component Synthesis of N-(Methylene-4-oxo coumarinyl)anilines; Their Z,E-Isomeric Product Distribution Determination From 1HNMR and their Antibacterial Studies

, 9(5): 454 - 458

Abdul Rauf, Hamish McNab and Ashfaq Mahmood Qureshi


DOI: 10.2174/157018012800389377




Synthesis and Antitumor Activities of 4H-Pyrano[3,2-h]quinoline-3-carbonitrile, 7H-Pyrimido[4',5':6,5]pyrano[3,2-h]quinoline, and 14HPyrimido[4',5':6,5]pyrano[3,2-h][1,2,4]triazolo[1,5-c]quinoline Derivatives

, 9(5): 459 - 470

Abdullah Megbas Al-Ghamdi, Ashraf Hassan Fekry Abd El-Wahab, Hany Mostafa Mohamed and Ahmed Mohamed El-Agrody


DOI: 10.2174/157018012800389331




An Efficient Synthesis, Characterization and Antimicrobial Screening of N-substituted 2-(piperidin-4-yl)-2H-benzo[d] [1, 2, 3] Triazoles

, 9(5): 471 - 478

Jalapathi Pochampalli, Devender Mandala, Nalla Umapathireddy and Pompu Rajakomuraiah


DOI: 10.2174/157018012800389304




Design, Synthesis and Evaluation of Chalcone Derivatives as Anti- Inflammatory, Antioxidant and Antiulcer Agents

, 9(5): 479 - 488

Alka N. Choudhary, Arun Kumar and Vijay Juy


DOI: 10.2174/157018012800389368




Synthesis and Biological Evaluation of Berberine Derivatives as IBS Modulator

, 9(5): 489 - 493

Xin Deng, Xinxin Zhao, Jing Han, Jingjie Wang, Wenlong Huang, Hai Qian and Liang Ge


DOI: 10.2174/157018012800389386




Deformable Surfactant Vesicles Loading Ammonium Glycyrrhizinate: Characterization and In Vitro Permeation Studies

, 9(5): 494 - 499

Luisa Di Marzio, Carlotta Marianecci, Federica Rinaldi, Sara Esposito and Maria Carafa


DOI: 10.2174/157018012800389287




CNS Cancer Cell Line Cytotoxicity Profiles of Some 2, 6, 9-Substituted Purines: A Comparative Five-Dose Testing Study

, 9(5): 500 - 504

Tien N. Banh, Nageswara R. Kode and Shashikan Phadtare


DOI: 10.2174/157018012800389241




Enhanced Oral Bioavailability of Oleanolic Acid in Rats with Phospholipid Complex

, 9(5): 505 - 512

Feng Cao, Yahan Gao, Zhi Yin and Qineng Ping


DOI: 10.2174/157018012800389340




The Analgesic Activity of 8-(Trifluoromethyl)-1,2,3,4,5-benzopentathiepine- 6-amine and Its Hydrochloride

, 9(5): 513 - 516

Tatyana G. Tolstikova, Alla V. Pavlova, Ekaterina A. Morozova, Tatyana M. Khomenko, Konstantin P. Volcho and Nariman F. Salakhutdin


DOI: 10.2174/157018012800389296




In Vivo Applied Positively Charged FITC-Labeled Peptide Conjugates Show Artificial Relocation in Frozen Sections

, 9(5): 517 - 526

Alexander Sturzu, Sumbla Sheikh, Ulrich Vogel, Hartmut Echner, Alireza Gharabaghi, Alexander Beck, Thomas Nagele, Ulrike Ernemann and Stefan Heckl


DOI: 10.2174/157018012800389313




In Silico Methods Applied in Food Chemistry: A Short Review with Bitter and Mutagenic Compounds

, 9(5): 527 - 534

Luciana Scotti, Hamilton Ishiki, Marcelo J.P. Ferreira, Francisco J.B.M. Junior, Vicente de P. Emerenciano, Marcelo S. Silva and Marcus T. Scotti


DOI: 10.2174/157018012800389269




Small Molecules Antileishmanials: A Review

, 9(5): 535 - 548

Akanksha Kulshrestha, Meenakshi Dhanawat, Nirupam Das and Sushant K. Shrivastava


DOI: 10.2174/157018012800389359




A Study on the Biological Activity of 2-thioxo-imidazolidin-4-ones

, 9(5): 549 - 555

Sudha Vengurlekar, Rajesh Sharma and Piyush Trivedi


DOI: 10.2174/157018012800389322




Retraction Notice: Solubilization and Amorphization of Non Steroidal Anti-Inflammatory Drug with Low Molecular Weight Chitosan for a New Guar-Based Colon Delivery Formulation

, 9(5): 556


DOI: 10.2174/1570180811209050556




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