Contents

Letters in Drug Design & Discovery, Volume 9 - Number 3

Graphical Abstracts

, 9(3): i - vi


DOI: 10.2174/157018012799129819




Editorial [ Hot Topic :Recent Developments in the Discovery of Anticancer Agents (Guest Editors: Ahmed Kamal and Y.V.D.Nageswar)]

, 9(3): 225

Ahmed Kamal


DOI: 10.2174/157018012799129855




Manipulating the Ability of Substituted Titanocene Derivatives to Induce Apoptosis in Castrate-Resistant Prostate Cancer Cells

, 9(3): 226 - 233

Catherine M. Dowling, Sandra Cuffe, Matthias Tacke, Anthony Deally, Megan Hogan, John M. Fitzpatrick and R. William G. Watson


DOI: 10.2174/157018012799129891




Synthesis, DNA Binding and Anticancer Activity of Pyridylimidazolidinone Linked Pyrrolo[2,1-c][1,4]benzodiazepine Conjugates

, 9(3): 234 - 241

Ahmed Kamal, B. Ashwini Kumar and Paidakula Suresh


DOI: 10.2174/157018012799129927




Synthesis, Anticancer Activity and Inhibition of Tubulin Polymerization of Bisindole Sulfonates

, 9(3): 242 - 250

Ahmed Kamal, Y. V.V. Srikanth, M. Naseer Ahmed Khan, Md. Ashraf, Thokhir Basha Shaik and Shasi V. Kalivendi


DOI: 10.2174/157018012799129774




Cytotoxic Activity of Polysubstituted 7-chloro-4-quinolinylhydrazone Derivatives

, 9(3): 251 - 256

Raquel Carvalho Montenegro, Leticia Veras Lotufo, Manoel Odorico de Moraes, Claudia do O Pessoa, Felipe Augusto Rocha Rodrigues, Marcelle de Lima Ferreira Bispo, Bruna Abreu Freire, Carlos Roland Kaiser and Marcus Vinicius Nora de Souza


DOI: 10.2174/157018012799129837




Synthesis and Antitumoral Evaluation of Benzyl (1S)-2-[2-(monosubstituted-benzylidene)hydrazino]-1-(hydroxymethyl)-2-oxoethylcarbamate

, 9(3): 257 - 262

Raquel Carvalho Montenegro, Leticia Veras Costa Lotufo, Manoel Odorico de Moraes, Claudia do O Pessoa, Felipe Augusto Rocha Rodrigues, Alessandra Campbell Pinheiro, Thais Cristina Mendonça Nogueira and Marcus Vinicius Nora de Souza


DOI: 10.2174/157018012799129800




Carbohydrate Based Blood Antigens in Cancer: Current Status and Future Perspectives

, 9(3): 263 - 275

Syed Khalid Yousuf, Debaraj Mukherjee and Subhash Chandra Taneja


DOI: 10.2174/157018012799129783




Synthesis of New S-alkylated-3-mercapto-1,2,4-triazole Derivatives Bearing Cyclic Amine Moiety as Potent Anticancer Agents

, 9(3): 276 - 281

M. S.R. Murty, Kesur R. Ram, Rayudu Venkateswara Rao, J. S. Yadav, Janapala Venkateswara Rao and L. R. Velatooru


DOI: 10.2174/157018012799129882




Metal Complexes of Uracil Derivatives with Cytotoxicity and Superoxide Scavenging Activity

, 9(3): 282 - 287

Supaluk Prachayasittikul, Apilak Worachartcheewan, Ratchanok Pingaew, Thummaruk Suksrichavalit, Chartchalerm Isarankura-Na-Ayudhya, Somsak Ruchirawat and Virapong Prachayasittikul


DOI: 10.2174/157018012799129918




The Chemometric Evaluation of Antitumor Activity of Novel Benzensulfonamide Derivatives Based on their Physiochemical Properties

, 9(3): 288 - 294

Mariusz Belka, Lucyna Konieczna, Piotr Kawczak, Tomasz Ciesielski, Jaroslaw Slawinski and Tomasz Baczek


DOI: 10.2174/157018012799129945




Design, Synthesis and Biochemical Evaluation of Estrogen Receptor Ligand Conjugates as Tumour Targeting Agents

, 9(3): 295 - 304

Niall O. Keely, Daniela M. Zisterer and Mary J. Meegan


DOI: 10.2174/157018012799129864




One Pot Synthesis and In Vitro Antitumor Activity of some Bipyrazolic Tripodal Derivatives

, 9(3): 305 - 309

Smaail Radi, Yahya Toubi, Nihed Draoui, Olivier Feron and Olivier Riant


DOI: 10.2174/157018012799129792




Synthesis and Biological Evaluation of Some Hydrazone Derivatives as Anti-inflammatory Agents

, 9(3): 310 - 315

Zafer Asim Kaplancikli, Mehlika Dilek Altintop, Ahmet Ozdemir, Gulhan Turan-Zitouni, Shabana I. Khan and Nurhayat Tabanca


DOI: 10.2174/157018012799129828




Synthesis and In Vitro Antibacterial Screening of some New 2,4,6-Trisubstituted-1,3,5-Triazine Derivatives

, 9(3): 316 - 321

Ravi Bhushan Singh, Nirupam Das, Srabanti Jana and Aparoop Das


DOI: 10.2174/157018012799129936




Calcium Level Controlling Activities of Novel Derivatives of Amlodipine,Riodipine and Cerebrocrast

, 9(3): 322 - 328

R. Vilskersts, B. Vigante, Z. Neidere, A. Krauze, I. Domracheva, L. Bekere, I. Shestakova, G. Duburs and M. Dambrova


DOI: 10.2174/157018012799129909




Design, Facile Synthesis, Antibacterial Activity and Structure-Activity Relationship of Novel Di- and Tri-Substituted 1,3,5-Triazines

, 9(3): 329 - 335

Surajit Kumar Ghosh, Ashmita Saha, Bornali Hazarika, Udaya Pratap Singh, Hans Raj Bhat and Prashant Gahtori


DOI: 10.2174/157018012799129846




Optimization and Evaluation of Micromeritic and Release Properties of High Dose Flutamide Liquisolid Systems

, 9(3): 336 - 344

Kadria A. Elkhodairy and Wael M. Samy


DOI: 10.2174/157018012799129873




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