Contents

Letters in Drug Design & Discovery, Volume 9 - Number 10

Graphical Abstract

Graphical Abstracts

, 9(10): i - iv


DOI: 10.2174/157018081120905000i




Acknowledgement

, 9(10): v


DOI: 10.2174/157018081120905000v




Novel Non-Competitive Antagonists of Kainate GluK1/GluK2 Receptors

, 9(10): 891 - 898

Agnieszka Anna Kaczor, Christiane Kronbach, Klaus Unverferth, Kalevi Pihlaja, Kirsti Wiinamaki, Jari Sinkkonen, Urszula Kijkowska-Murak, Tomasz Wrobel, Tomasz Stachal and Dariusz Matosiuk


DOI: 10.2174/1570180811209050891




Pharmacophore Generation and 3D-QSAR of Novel 2-(quinazolin-4- ylamino)-[1,4] Benzoquinone Derivatives as VEGFR-2 Inhibitors

, 9(10): 899 - 914

Mahesh Kumar Teli, Pradeep Hanumanthappa and Rajanikant G. Krishnamurthy


DOI: 10.2174/1570180811209050899




QSAR Studies of PTP1B Inhibitors: 1, 2-Naphthoquinone Derivatives

, 9(10): 915 - 925

Feng Luan, Xuan Xu, Huitao Liu, Maria Natalia Dias Soeiro Cordeiro and Xiaoyun Zhang


DOI: 10.2174/1570180811209050915




3-(Adamantan-1-yl)-4-hydroxybenzyl Substituted Purines and Pyrimidines: Synthesis and Cytotoxic Activity

, 9(10): 926 - 933

Nageswara Rao Kode, Dakshinamurthy Devangachinta and Shashikant Phadtare


DOI: 10.2174/1570180811209050926




Microwave Assisted Synthesis, Characterization of Some New Isatin and Thiophene Derivatives as Cytotoxic and Chemopreventive Agents

, 9(10): 934 - 941

Kiran Gangarapu, Sarangapani Manda, Sreekanth Thota, Rajeshwar Yerra, Subhas S. Karki, Jan Balzarini, Erik De Clercq and Harukuni Tokuda


DOI: 10.2174/1570180811209050934




Synthesis and Cytotoxicity Evaluation of Some Novel 3,5-disubstituted- 1,2,4-Oxadiazoles

, 9(10): 942 - 946

M. Siva Nagi Reddy, B. Sailaja Kumari and B. Hari Babu


DOI: 10.2174/1570180811209050942




Halogen Substituents as an Effective Modulators of Antibacterial Activity of Substituted 1,2,4-triazole-3-thiones

, 9(10): 947 - 952

Tomasz Plech, Monika Wujec, Urszula Kosikowska and Anna Malm


DOI: 10.2174/1570180811209050947




Antimycobacterial Agents: Synthesis and Biological Evaluation of Novel 4-(Substituted-phenyl)-6-methyl-2-oxo-N-(pyridin-2-yl)-1,2,3,4-tetrahydropyrimidine- 5-carboxamide Derivatives by Using One-pot Multicomponent Method

, 9(10): 953 - 957

Abdulrahman I. Almansour, Mohamed Ashraf Ali, Sadath Ali, Ang Chee Wei, Yeong Keng Yoon, Rusli Ismail, Tan Soo Choon, Suresh Pandian, Raju Suresh Kumar, Natarajan Arumugam and Hasnah Osman


DOI: 10.2174/1570180811209050953




Exploring Nitrostyrene as a Scaffold for a New Class a of Monoamine Oxidase Inhibitors

, 9(10): 958 - 961

Joana Reis, Catarina Oliveira, Nuno Milhazes, Dolores Vina and Fernanda Borges


DOI: 10.2174/1570180811209050958




Synthesis of 3,4–Dihydropyrimidin–2-ones (DHPMs) Using Highly Efficient Recyclable Silica Supported Rhodium Chloride as Heterogeneous Catalyst and their Anti-Neuroinflammatory Activity

, 9(10): 962 - 966

Shobha Donthabhakthuni, Adharvana Chari Murugulla, Prabhakara Chari Murugulla and Kim SunYeou


DOI: 10.2174/1570180811209050962




Hydroxysafflor Yellow A Attenuates Renal Ischemia- Reperfusion Injury in a Rat Model

, 9(10): 967 - 972

Weiran Chai, Wenhui Zhang, Zhu Jin, Yanqian Zheng, Peiyao Jin, Qiaoyan Zhang and Jianming Zhi


DOI: 10.2174/1570180811209050967




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