Letters in Drug Design & Discovery, Volume 9 - Number 1

Graphical Abstracts

, 9(1): i - v

DOI: 10.2174/157018012798192964


, 9(1): 1


DOI: 10.2174/157018012798192937

Design and Synthesis of 3-Arylisoxazoline-5-Carboxamide and 3-Arylisoxazoline-5-Acetamide Libraries as Potential Factor Xa Inhibitors

, 9(1): 2 - 7

John F. Quinn, Brian T. Gregg, Douglas B. Kitchen, Robert M. Lewis, Dana A. Razzano, Lauren E. Kayser, Levon J. Schilling and Kathryn C. Golden

DOI: 10.2174/157018012798193035

Antioxidant Activity of Resveratrol Analogs

, 9(1): 8 - 11

Natalia Oliveira Calil, Gustavo Senra Goncalves de Carvalho, Danielle Cristina Zimmermann Franco, Adilson David da Silva and Nadia Rezende Barbosa Raposo

DOI: 10.2174/157018012798192928

Semi-Automatic Synthesis of Distamycin Analogues and their DNA Binding Properties

, 9(1): 12 - 16

Danuta Drozdowska and Jakub Szerszenowicz

DOI: 10.2174/157018012798192919

Ligand and Structure-Based Pharmacophore Modeling for the Discovery of Potential Human HNMT Inhibitors

, 9(1): 17 - 29

Pavadai Elumalai, Hsuan-Liang Liu, Zheng-Li Zhou, Jian-Hua Zhao, Wilson Chen, Chih-Kuang Chuang, Wei-Bor Tsai and Yih Ho

DOI: 10.2174/157018012798192955

Synthesis and Anti-Paracoccidioides Activity of Calix[n]arenes

, 9(1): 30 - 36

Marcilene Coimbra de Oliveira, Fabiano Souza Reis, Angelo de Fatima, Thais Furtado Ferreira Magalhaes, Danielle Leticia da Silva, Raphael Rodrigues Porto, Giselle Almeida Watanabe, Cleide Viviane Buzanello Martins, Daniel Leite da Silva, Ana Lucia Tasca Gois Ruiz, Sergio Antonio Fernandes, Joao Ernesto de Carvalho and Maria Aparecida de Resende-Stoianoff

DOI: 10.2174/157018012798192991

Preliminary Evaluation of Anticonvulsant Activity of Some Aminoalkanol and Amino Acid Cinnamic Acid Derivatives

, 9(1): 37 - 43

Agnieszka Gunia, Anna M. Waszkielewicz, Marek Cegla and Henryk Marona

DOI: 10.2174/157018012798192982

Discovery of 5,6-Dihydro-indolo[1,2-a]quinoxaline Derivatives as New HIV-1 Inhibitors In Vitro

, 9(1): 44 - 47

Ling-Ling Fan, Ning Huang, Rui-Ge Yang, Shu-Zhen He, Liu-Meng Yang, Hui Xu and Yong-Tang Zheng

DOI: 10.2174/157018012798193026

Evaluation of the Radioprotective Potential of the Polyphenol Norbadione A

, 9(1): 48 - 53

Antoine Le Roux, Elodie Josset, Sami Benzina, Brice Nadal, Marine Desage-El Murr, Benoit Heurtaux, Frederic Taran, Jean-Marc Denis, Thierry Le Gall, Stephane Meunier and Pierre Bischoff

DOI: 10.2174/157018012798192900

Lobeline Docking on AChBP and Nicotinic Receptors: Discriminating Importance of the Pocket Geometry and of the Ligand Configuration

, 9(1): 54 - 62

Claire Colas, Xavier Brotel, Nathalie Duclert-Savatier, Michael Nilges, Delphine Joseph and Therese E. Malliavin

DOI: 10.2174/157018012798193017

Synthesis and Biological Evaluation of Some Novel Thiazolylhydrazinomethylideneferrocenes as Antimicrobial Agents

, 9(1): 63 - 68

Navneet Chandak, Pawan Kumar, Chetan Sharma, Kamal R. Aneja and Pawan K. Sharma

DOI: 10.2174/157018012798192973

Synthesis, Biochemical Evaluation and Rationalisation of a Series of (3-O-Sulfonate) Derivatives of Estrone (E1) as Probes of the Active Site of Type 3 of the 17β-Hydroxysteroid Dehydrogenase (17β-HSD) Family of Enzymes

, 9(1): 69 - 76

Mohsen Akbarzadeh, Moniola S. Olusanjo and Sabbir Ahmed

DOI: 10.2174/157018012798193044

Pramipexole Tachyphylaxis and its Management in Bipolar Depression

, 9(1): 77

Verinder Sharma

DOI: 10.2174/157018012798193008

Design, Synthesis and Biological Evaluation of Scutellarein Derivatives as Potential Anti-Alzheimers Disease Candidates Based on Metabolic Mechanism

, 9(1): 78 - 83

Shu-Lin Song, Nian-Guang Li, Yu-Ping Tang, Zhen-Jiang Wang, Li-Hua Qian, Hao Tang and Jin-Ao Duan

DOI: 10.2174/157018012798192946

Small Molecule Tyrosine Kinase Inhibitors: The New Dawn for Cancer Therapy

, 9(1): 84 - 125

Malleshappa N. Noolvi and Harun M. Patel

DOI: 10.2174/157018012798192892

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