Contents

Letters in Drug Design & Discovery, Volume 9 - Number 1

Graphical Abstracts

, 9(1): i - v


DOI: 10.2174/157018012798192964




Editorial

, 9(1): 1

Atta-ur-Rahman


DOI: 10.2174/157018012798192937




Design and Synthesis of 3-Arylisoxazoline-5-Carboxamide and 3-Arylisoxazoline-5-Acetamide Libraries as Potential Factor Xa Inhibitors

, 9(1): 2 - 7

John F. Quinn, Brian T. Gregg, Douglas B. Kitchen, Robert M. Lewis, Dana A. Razzano, Lauren E. Kayser, Levon J. Schilling and Kathryn C. Golden


DOI: 10.2174/157018012798193035




Antioxidant Activity of Resveratrol Analogs

, 9(1): 8 - 11

Natalia Oliveira Calil, Gustavo Senra Goncalves de Carvalho, Danielle Cristina Zimmermann Franco, Adilson David da Silva and Nadia Rezende Barbosa Raposo


DOI: 10.2174/157018012798192928




Semi-Automatic Synthesis of Distamycin Analogues and their DNA Binding Properties

, 9(1): 12 - 16

Danuta Drozdowska and Jakub Szerszenowicz


DOI: 10.2174/157018012798192919




Ligand and Structure-Based Pharmacophore Modeling for the Discovery of Potential Human HNMT Inhibitors

, 9(1): 17 - 29

Pavadai Elumalai, Hsuan-Liang Liu, Zheng-Li Zhou, Jian-Hua Zhao, Wilson Chen, Chih-Kuang Chuang, Wei-Bor Tsai and Yih Ho


DOI: 10.2174/157018012798192955




Synthesis and Anti-Paracoccidioides Activity of Calix[n]arenes

, 9(1): 30 - 36

Marcilene Coimbra de Oliveira, Fabiano Souza Reis, Angelo de Fatima, Thais Furtado Ferreira Magalhaes, Danielle Leticia da Silva, Raphael Rodrigues Porto, Giselle Almeida Watanabe, Cleide Viviane Buzanello Martins, Daniel Leite da Silva, Ana Lucia Tasca Gois Ruiz, Sergio Antonio Fernandes, Joao Ernesto de Carvalho and Maria Aparecida de Resende-Stoianoff


DOI: 10.2174/157018012798192991




Preliminary Evaluation of Anticonvulsant Activity of Some Aminoalkanol and Amino Acid Cinnamic Acid Derivatives

, 9(1): 37 - 43

Agnieszka Gunia, Anna M. Waszkielewicz, Marek Cegla and Henryk Marona


DOI: 10.2174/157018012798192982




Discovery of 5,6-Dihydro-indolo[1,2-a]quinoxaline Derivatives as New HIV-1 Inhibitors In Vitro

, 9(1): 44 - 47

Ling-Ling Fan, Ning Huang, Rui-Ge Yang, Shu-Zhen He, Liu-Meng Yang, Hui Xu and Yong-Tang Zheng


DOI: 10.2174/157018012798193026




Evaluation of the Radioprotective Potential of the Polyphenol Norbadione A

, 9(1): 48 - 53

Antoine Le Roux, Elodie Josset, Sami Benzina, Brice Nadal, Marine Desage-El Murr, Benoit Heurtaux, Frederic Taran, Jean-Marc Denis, Thierry Le Gall, Stephane Meunier and Pierre Bischoff


DOI: 10.2174/157018012798192900




Lobeline Docking on AChBP and Nicotinic Receptors: Discriminating Importance of the Pocket Geometry and of the Ligand Configuration

, 9(1): 54 - 62

Claire Colas, Xavier Brotel, Nathalie Duclert-Savatier, Michael Nilges, Delphine Joseph and Therese E. Malliavin


DOI: 10.2174/157018012798193017




Synthesis and Biological Evaluation of Some Novel Thiazolylhydrazinomethylideneferrocenes as Antimicrobial Agents

, 9(1): 63 - 68

Navneet Chandak, Pawan Kumar, Chetan Sharma, Kamal R. Aneja and Pawan K. Sharma


DOI: 10.2174/157018012798192973




Synthesis, Biochemical Evaluation and Rationalisation of a Series of (3-O-Sulfonate) Derivatives of Estrone (E1) as Probes of the Active Site of Type 3 of the 17β-Hydroxysteroid Dehydrogenase (17β-HSD) Family of Enzymes

, 9(1): 69 - 76

Mohsen Akbarzadeh, Moniola S. Olusanjo and Sabbir Ahmed


DOI: 10.2174/157018012798193044




Pramipexole Tachyphylaxis and its Management in Bipolar Depression

, 9(1): 77

Verinder Sharma


DOI: 10.2174/157018012798193008




Design, Synthesis and Biological Evaluation of Scutellarein Derivatives as Potential Anti-Alzheimers Disease Candidates Based on Metabolic Mechanism

, 9(1): 78 - 83

Shu-Lin Song, Nian-Guang Li, Yu-Ping Tang, Zhen-Jiang Wang, Li-Hua Qian, Hao Tang and Jin-Ao Duan


DOI: 10.2174/157018012798192946




Small Molecule Tyrosine Kinase Inhibitors: The New Dawn for Cancer Therapy

, 9(1): 84 - 125

Malleshappa N. Noolvi and Harun M. Patel


DOI: 10.2174/157018012798192892




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