Contents

Letters in Drug Design & Discovery, Volume 8 - Number 9

Graphical Abstracts

, 8(9): i - v


DOI: 10.2174/157018011797200885




Rapid and Facile Synthesis of N-Benzenesulfonyl Derivatives of Heterocycles and their Antimicrobial Properties

, 8(9): 778 - 791

Romina J. Pagliero, Reesa Mercado, Vance McCracken, Maria R. Mazzieri and Marcelo J. Nieto


DOI: 10.2174/157018011797200803




Isonicotinic Acid Hydrazide Derivatives: Synthesis, Antimycobacterial, Antiviral, Antimicrobial Activity and QSAR Studies

, 8(9): 792 - 810

Vikramjeet Judge, Balasubramanian Narasimhan, Munish Ahuja, Dharmarajan Sriram and Perumal Yogeeswar


DOI: 10.2174/157018011797200795




Synthesis, Antibacterial and Antifungal Activities of Some Carbazole Dithiocarbamate Derivatives

, 8(9): 811 - 815

Ahmet Cagri Karaburun, Zafer Asim Kaplancikli, Nalan Gundogdu-Karaburun and Fatih Demirci


DOI: 10.2174/157018011797200858




Synthesis and Biological Evaluation of Andrographolide Derivatives as Potent Antibacterial Agents

, 8(9): 816 - 821

Chunlei Tang, Wenjie Zhang, Xinyang Wang, Bin Wang, Xiaoyun Zhu, Dandan Huang, Xiaoyong Du, Hai Qian, Wenlong Huang and Jing Li


DOI: 10.2174/157018011797200740




Synthesis and In Vitro Antiviral Evaluation of Novel 1-Arylpyrazoles and Their N- and S-Glycosides

, 8(9): 822 - 829

Emad M. El-Telbani, Sara M. Ghanem, Farrag A. El-Essawy and Aly F. El-Sayed


DOI: 10.2174/1570180811108090822




Synthesis of Some Benzothiazole Based Piperazine-Dithiocarbamate Derivatives and Evaluation of Their Anticancer Activities

, 8(9): 830 - 837

Gulhan Turan-Zitouni, Yusuf Ozkay, Ahmet Ozdemir, Zafer Asim Kaplancikli and Mehlika Dilek Altintop


DOI: 10.2174/157018011797200786




Thiazole Containing Nitrogen Mustards: Synthesis, Structural Evaluation, Cytotoxicity and DNA Binding Studies

, 8(9): 838 - 842

Nulgulmnalli Manjunathiah Raghavendra, Surampudi Renuka, Sayan Dutta Gupta and Pingili Divya


DOI: 10.2174/157018011797200830




Synthesis and In Vitro Antitumor Activity of Novel Fluorine Containing Pyrazoles and Pyrazolines

, 8(9): 843 - 849

Ashish Sharma, Tabreskhan Pathan, Rhea Mohan and C. S. Ramaa


DOI: 10.2174/157018011797200812




Use of Physicochemical and Topological Parameters in Estimating Anti-Cancer Activity of Benzothiazole Derivatives

, 8(9): 850 - 856

Deepali Gupta, Basheerulla Shaik, Jyoti Singh, Neelu Singh and Vijay K. Agrawal


DOI: 10.2174/157018011797200759




Cytotoxicity Study on Some Synthetic Aromatic Esters of 4-Demethyl-4-deoxypodophyllotoxin

, 8(9): 857 - 860

Juan-Juan Wang, Hong-Jin Han, Guang-Zhi Zeng, Hui Xu and Ning-Hua Tan


DOI: 10.2174/157018011797200849




Doxorubicin Sensitizes the Non-Small Cell Lung Cancer Cells to Tumor Necrosis Factor-Related Apoptosis-Inducing Ligand-Mediated (TRAIL) Apoptosis In Vitro but not In Vivo

, 8(9): 861 - 867

Li Fan, Liangran Guo, Jinfeng Ren, Yulong Ren, Zhiqing Pang and Xinguo Jiang


DOI: 10.2174/157018011797200867




A QSAR Analysis of Coumarin Derivatives as TNF-α Inhibitor - A Rational Approach to Anticancer Drug Design

, 8(9): 868 - 876

Malleshappa N. Noolvi, Harun M. Patel and Tarandeep Kaur


DOI: 10.2174/157018011797200768




A Comparative Molecular Field (CoMFA) Studies on Carbonic Anhydrase Inhibitor hCA IX-Tumor-Associated (Hypoxia)

, 8(9): 877 - 883

Shalini Singh


DOI: 10.2174/157018011797200777




Synthesis, Crystal Structure and Biological Evaluation of 4, 5, 6, 7-tetrahydropravastatin as HMG-CoA Reductase Inhibitor

, 8(9): 884 - 888

Jing Li, Huan Li and Lei Zhang


DOI: 10.2174/157018011797200876




Molecular Modelling, Design, Synthesis and Biochemical Evaluation of a Range of Non-Steroidal Thiosemicarbazone-Based Inhibitors of Estrone Sulfatase (ES) - A Potential Insight into the Action of a Range of Allosteric Inhibitors of ES

, 8(9): 889 - 896

Amit Kumar, Sukriti Singh, Balkrishna Bhamare, Kruti Shah, Pallav S. Shah and Sabbir Ahmed


DOI: 10.2174/157018011797200821




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