Contents

Letters in Drug Design & Discovery, Volume 8 - Number 8

Graphical Abstracts

, 8(8): i - v


DOI: 10.2174/157018011796576042




DNA Polymerase β Specific Inhibitors, a Loliolide Derivative and Pubinernoid A, Isolated from the Brown Algae Laminaria sp.

, 8(8): 671 - 677

Yoshiyuki Mizushina, Toshifumi Takeuchi, Isoko Kuriyama, Yoshihiro Takahashi, So Maezawa, Takuro Matsumoto, Osamu Koiwai, Fumio Sugawara and Hiromi Yoshida


DOI: 10.2174/157018011796576024




Characterization of Carbonic Anhydrase Isozyme Specific Inhibition by Sulfamated 2-Ethylestra Compounds

, 8(8): 678 - 684

Katherine H. Sippel, Andre Stander, Chingkuang Tu, Balasubramanian Venkatakrishnan, Arthur H. Robbins, Mavis Agbandje-McKenna, Fourie Joubert, Annie M. Joubert and Robert McKenna


DOI: 10.2174/157018011796576105




Structure-Activity Evaluation of N-benzyl-5-substituted Indole-3-imine Derivatives and their Amine Congeners as Bovine Testicular Hyaluronidase (BTH) Inhibitor

, 8(8): 685 - 690

S. Olgen, A. Kaessler, Z. Kilic Kurt and J. Jose


DOI: 10.2174/157018011796576079




Prevention of VP-16 Resistance by a Disiloxane, SILA409: Effects of SILA409 on the Expression of GRP78 in NCI-H446 Human Small Cell Lung Cancer Cells

, 8(8): 691 - 697

Encheng Li, Jinhui Zhang, Jiarui Wang, Fei Gao, Zhonghai Yang, Qiang Meng, Qianqian Zhang, Na Li, Ming Huang, Gabriella Spengler, Joseph Molnar and Qi Wang


DOI: 10.2174/157018011796575971




Synthesis and Anti – Tumour Activity of Novel Camptothecin – Bile Acid Analogues

, 8(8): 698 - 703

Q.-Y. Li, Y. Gao, W. Qiu, Y.-G. Zu, L. Su, W.-N. He and X.-Q. Deng


DOI: 10.2174/157018011796576006




Design, Synthesis and Cytotoxicity of Chalcone Analogs Derived from 2-Phenylimino-3-phenylthiazolidin-4-one

, 8(8): 704 - 708

Vijay Satam, Ravi Kumar Bandi, Ajaya Kumar Behera, Bijay Kumar Mishra, Olivia Brockway, Samuel Tzou, Matthias Zeller, Moses Lee and Hari Pati


DOI: 10.2174/157018011796576033




Aryl and Acyclic Unsaturated Derivatives of Thioguanine and 6- Mercaptopurine: Synthesis and Cytotoxic Activity

, 8(8): 709 - 716

Tien N. Banh, Nageswara R. Kode and Shashikant Phadtare


DOI: 10.2174/157018011796576088




Synthesis and Preliminary In-Vitro Cytotoxic Activity of Novel Substituted diaryl-imidazo [2,1,b]-benzothiazole Derivatives

, 8(8): 717 - 724

Jitender K. Malik, Malleshappa N. Noolvi, Fakkirappa V. Manvi, B.K. Nanjwade, Harun M. Patel, Manjula S. N., Mallikarjuna Rao C. and Ashutosh Barve


DOI: 10.2174/157018011796576015




Synthesis, Biological Evaluation and In Silico Study of β-Chloro Vinyl Chalcones as Inhibitors of the TNF-α, IL-6 With Anticancer and Antioxidant Activity

, 8(8): 725 - 732

Babasaheb P. Bandgar, Baliram S. Hote and Shivraj H Nile


DOI: 10.2174/157018011796576051




Nicotinic Acid Benzylidene/Phenyl-Ethylidene Hydrazides: Synthesis, Antimicrobial Evaluation and QSAR Studies

, 8(8): 733 - 749

Rakesh Narang, Balasubramanian Narasimhan, Sunil Sharma, Dharmarajan Sriram, Perumal Yogeeswari, Erik De Clercq, Christophe Pannecouque and Jan Balzarini


DOI: 10.2174/157018011796575999




Concise and Facile Synthesis of Novel Pyrano[2,3-d]pyrimidine-7- one/thione Derivatives as In Vitro Antimicrobial and Antitubercular Agents

, 8(8): 750 - 757

Prashant T. Mistry, Nimesh R. Kamdar, Dhaval D. Haveliwala and Saurabh K. Patel


DOI: 10.2174/157018011796576060




Synthesis and Antifungal Activities of Some Aryl Naphthofuran Ketoximes

, 8(8): 758 - 762

Ahmet Cagri Karaburun, Nalan Gundogdu-Karaburun, Umit Ucucu and Seref Demirayak


DOI: 10.2174/157018011796576097




Facile Synthesis, Antibacterial Activity and Molecular Properties Prediction of Some New 1,3-dihydroimidazol-2-thione Derivatives

, 8(8): 763 - 768

Julfikar Ali Junejo, Surajit Kumar Ghosh, Mutahar Shaikh, Prashant Gahtori and Udaya Pratap Singh


DOI: 10.2174/157018011796575980




Synthesis and Anticonvulsant Activity Evaluation of 6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazines

, 8(8): 769 - 773

Ming-Xia Song, Chun-Bo Zhang, Xian-Qing Deng, Zhi-Gang Sun and Zhe-Shan Quan


DOI: 10.2174/157018011796575962




Synthesis, Neurotoxicity and Anticonvulsant Study of Some Benzothiazole Analogs

, 8(8): 774 - 777

Kalyan K. Sethi, Saurabh M. Verma, Naru Prasanthi and Mathrusri M. Annapurna


DOI: 10.2174/157018011796575953




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