Contents

Letters in Drug Design & Discovery, Volume 8 - Number 6

Graphical Abstracts

, 8(6): i - v


DOI: 10.2174/157018011795906767




High-Density Lipoprotein Cholesterol-Elevating Effect of a Novel Peroxisome Proliferator-Activated Receptor δ Agonist

, 8(6): 496 - 499

Shogo Sakuma, Tsuyoshi Endo, Takashi Kanda, Hideki Nakamura, Satomi Yamasaki and Tomio Yamakawa


DOI: 10.2174/157018011795906802




Synthesis and Biological Evaluation of Ezetimibe Analogs as Possible Cholesterol Absorption Inhibitors

, 8(6): 500 - 505

Yubin Wang, Haiqian, Wenlong Huang, Huibin Zhang and Jinpei Zhou


DOI: 10.2174/157018011795906776




Exploring the Structure Activity Relationships of Imidazole Containing Tetrahydrobenzodiazepines as Farnesyltransferase Inhibitors: A QSAR Study

, 8(6): 506 - 515

Anand Gaurav, Vertika Gautam and Ranjit Singh


DOI: 10.2174/157018011795906758




Synthesis, Biochemical Evaluation and Rationalisation of the Inhibitory Activity of a Range of Derivatives of 2-imidazol-1-yl-1-phenyl-ethanone as Potential Novel Inhibitors of 17α-hydroxylase/17,20-lyase (P-45017α)

, 8(6): 516 - 522

Kruti Shah, Baljeet Jandu, Ammara Abdullah and Sabbir Ahmed


DOI: 10.2174/157018011795906749




Synthesis and SAR Study of Prenylated Xanthone Analogues as HeLa and MDA-MB-231 Cancer Cell Inhibitors

, 8(6): 523 - 528

Chan Kiang Lim, Lai-Yeng Tho, Cheng Hoe Lim, Yang Mooi Lim, Syed Adnan Ali Shah and Jean-Frederic Faizal Weber


DOI: 10.2174/157018011795906820




Specificity of Three Vasopressin Receptor Antagonists

, 8(6): 529 - 535

Jeremy T. Saks, Barbara Truitt and Menachem Shoham


DOI: 10.2174/157018011795906794




Anticancer Activity of the Bioreductive and Non-Bioreductive Zerumbone Derivatives

, 8(6): 536 - 543

Siripit Pitchuanchom, Uraiwan Songsiang, Natthida Weerapreeyakul and Chavi Yenjai


DOI: 10.2174/157018011795906811




Lipid-Lowering Effects of Polymers Derived from Halophenyl Pyrroles

, 8(6): 544 - 549

Bruce S. Burnham, Joshua D. Berkowitz, Zachary Orr, Bryan McCranor, Mardel Cooper, Kurt McCann, Kyle Pillitteri, Jodi Hallback, Lisa-Marie Bergh, Larisa Gofman, Melissa Melendez, Justin M. Holub, Kenzo Morie and Charles E. Carraher


DOI: 10.2174/157018011795906839




Design, Synthesis and Biological Study of Novel NO-Donor-Caffeic Acid Hybrids as Potential Anti-Atherosclerotic Drug Candidates

, 8(6): 550 - 557

Nian-Guang Li, Rong Wang, Yu-Ping Tang, Zhi-Hao Shi, Bao-Quan Li, Wei Li, Jian-Ping Yang, Zhen-Jiang Wang, Shu-Lin Song, Li-Hua Qian, Li-Juan Yao, Jun-Zuan Xia, Jia Xu, Feng Feng, Da-Wei Qian and Jin-Ao Duan


DOI: 10.2174/157018011795906848




Novel Coumarin and 4H-Chromene Derivatives Containing 4,5- Dihydropyrazole Moiety: Synthesis and Antibacterial Activity

, 8(6): 558 - 561

Qian-Zhu Li, Xiao-Yan Nie and Jie Liang


DOI: 10.2174/157018011795906857




New Small-Size Antifungal Peptides: Design, Synthesis and Antifungal Activity

, 8(6): 562 - 567

Adriana D. Garro, Francisco M. Garibotto, Ana M. Rodriguez, Marcela Raimondi, Susana A. Zacchino, Andras Perczel, Csaba Somlai, Botond Penke and Ricardo D. Enriz


DOI: 10.2174/157018011795906785




A Flow Chemistry Approach to Norcantharidin Analogues

, 8(6): 568 - 574

Mark Tarleton, Kelly A. Young, Elli Unicomb, Siobhann N. McCluskey, Mark J. Robertson, Christopher P. Gordon and Adam McCluskey


DOI: 10.2174/157018011795906730




Synthesis, Characterization of (E)-N'-(substituted-benzylidene)isonicotinohydrazide Derivatives as Potent Antitubercular Agents

, 8(6): 575 - 579

Manav Malhotra, Rajiv Sharma, Vikramdeep Monga, Aakash Deep, Kapendra Sahu and Abdul Samad


DOI: 10.2174/157018011795906866




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