Contents

Letters in Drug Design & Discovery, Volume 8 - Number 5

Graphical Abstracts

, 8(5): i - iv


DOI: 10.2174/157018011795514177




Novel RGD Peptidomimetics Embedding 1,2,3-Triazole as Central Scaffold; Synthesis and αvβ3 Integrin Affinity

, 8(5): 401 - 405

Ming Hong Ni, Emiliano Esposito, Massimo Castorina and Alma Dal Pozzo


DOI: 10.2174/157018011795514258




Synthesis and Biological Evaluation of Spiro-δ-lactones as Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 2 (17β-HSD2)

, 8(5): 406 - 421

Kuiying Xu, Marie Wetzel, Rolf W. Hartmann and Sandrine Marchais-Oberwinkler


DOI: 10.2174/157018011795514230




Quantitative Structure Activity Relationship Studies on a Novel Indolediones as Long Chain Fatty Acid Elongase 6 (ELOVL6) Inhibitors

, 8(5): 422 - 429

Junxia Zheng, Zhiwei Wu, Mibei Dai, Zhihui Xu, Xiaomei Li, Shanshan Zhu, Chuyun Lin, Peijian Hu, Luo Zhang, Huarong Huang, Suqing Zhao, Kun Zhang and Pinghua Sun


DOI: 10.2174/157018011795514168




CoMFA and CoMSIA Analyses of Highly Selective Pipecolic Acid Based TNF-α Converting Enzyme (TACE) Inhibitors Using Docked Conformations for Molecular Alignment

, 8(5): 430 - 439

Malkeet Singh Bahia, Sukhvir Chand, Shravan Kumar Gunda, Shwetha Reddy Gade, Saikh Mahmood and Om Silakari


DOI: 10.2174/157018011795514195




Homology Modeling of α-Glucosidase and its Interactions with Andrograpolide Derivatives

, 8(5): 440 - 451

Jun Xu, Yijing Lu, Weizai Shen, Haibin Luo, Sichao Huang, Jiaolin Bao, Shaohui Cai and Yuqiang Wang


DOI: 10.2174/157018011795514203




Synthesis, Cytotoxic and Phytotoxic Effects of Some New N4-Aryl Substituted Isatin-3-thiosemicarbazones

, 8(5): 452 - 458

Humayun Pervez, Muhammad Ramzan, Muhammad Yaqub and Khalid Mohammed Khan


DOI: 10.2174/157018011795514159




Novel 2-(benzo[d]thiazol-2-yl)-1-(3-methyl-5-substituted-phenyl-4,5-dihydropyrazol-1-yl)ethanone Derivatives: Synthesis and Antibacterial Activity

, 8(5): 459 - 463

Chun-Xiu Pan, Jun Li and Xin-Hua Liu


DOI: 10.2174/157018011795514212




Synthesis and Antimicrobial Activity of 8-Alkylpalmatine Derivatives

, 8(5): 464 - 468

Teng-Wen Ma, Xiao-Li Ye, Xue-Gang Li, Bao-Shun Zhang, Xiao-Fei Jiang and Zu Chen


DOI: 10.2174/157018011795514186




Modern Methods & Web Resources in Drug Design & Discovery

, 8(5): 469 - 490

Feroz Khan, Dharmendra Kumar Yadav, Anupam Maurya and Santosh Kumar Srivastava


DOI: 10.2174/157018011795514249




Evaluation of N-(2-Thienylidene)amines, N-(2-Hydroxybenzylidene)amines and 3-Iminoindolin-2-ones as Antileishmanial Agents

, 8(5): 491 - 495

Yasser M.S.A. Al-Kahraman, Girija S. Singh and Masoom Yasinzai


DOI: 10.2174/157018011795514221




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