Contents

Letters in Drug Design & Discovery, Volume 8 - Number 3

Graphical Abstracts

, 8(3): i - iv


DOI: 10.2174/157018011794578268




Alteration of Warfarins Pharmacologic Properties in Clathrates with Glycyrrhizic Acid and Arabinogalactan

, 8(3): 201 - 204

Tatjana G. Tolstikov, Mikhail V. Khvostov, Galina I. Lifshits, Alexander V. Dushkin and Elezaveta S. Meteleva


DOI: 10.2174/157018011794578222




Novel Aglycones of Steroidal Glycoalkaloids as Potent Tyrosine Kinase Inhibitors: Role in VEGF and EGF Receptors Targeted Angiogenesis

, 8(3): 205 - 215

Salman Akhtar, Othman A. Al-Sagair and Jamal M. Arif


DOI: 10.2174/157018011794578187




Molecular Insight into the Inhibitory Mechanism of Galangin Towards Human Cytochrome P450 1A2. A Modeling Study

, 8(3): 216 - 222

Yunyun Chen, Guo-Wen Chen and Hai-Bin Luo


DOI: 10.2174/157018011794578150




Prediction of Specificity and Cross-Reactivity of Kinase Inhibitors

, 8(3): 223 - 228

Nitish Kumar Mishra and Gajendra P.S. Raghava


DOI: 10.2174/157018011794578204




3D-QSAR and Docking Studies on Pyrrolopyrimidine Derivatives as LIM-Kinase 2 Inhibitors

, 8(3): 229 - 240

Jun-Rong Sun, Ping Lan, Ping-Hua Sun and Wei-Min Chen


DOI: 10.2174/157018011794578178




Synthesis and Biological Evaluation of a Range of Thiosemicarbazone - Based Compounds as Potential Inhibitors of Estrone Sulfatase (ES)

, 8(3): 241 - 245

Amit Kumar, Sukriti Singh, Hadi Bordbar, Timothy Cartledge and Sabbir Ahmed


DOI: 10.2174/157018011794578231




Targeting Catechol-O-Methyl Transferase (COMT) Inhibitors for Schizophrenia:An Approach to Target Validation and Rational Drug Design

, 8(3): 246 - 252

Deepak Purushotham, Chaiti Ganguly and Chiranjib Chakraborty


DOI: 10.2174/157018011794578277




Synthesis and Biochemical Evaluation of a Series of Trifluoromethanesulfonate Derivatives of 4 Hydroxyphenyl Ketones – Probes of the Active Site of Type 1 and 3 of the 17β-Hydroxysteroid Dehydrogenase Family of Enzymes

, 8(3): 253 - 259

Moniola S. Olusanjo, Timothy Cartledge, Kruti Shah and Sabbir Ahmed


DOI: 10.2174/157018011794578259




In Silico Studies of (2E,5E)-2,5-bis(3-methoxy-4-hydroxy-benzylidene) Cyclopentanone on Proteins AChE and BChE Involved in Alzheimers disease and Ameliorative Effects on Paraquat Induced Oxidative Stress Markers in Drosophila melanogaster

, 8(3): 260 - 267

Balladka Kunhanna Sarojini, Chenna Govindaraju Darshan Raj, Modalkoppalu Kyathegowda Ramakrishna, Saraf R Ramesh, Basavapattana Rudresh Bharath and Hanumanthappa Manjunatha


DOI: 10.2174/157018011794578213




Microwave-Assisted Synthesis and Evaluation of Substituted Aryl Propyl Acridone-4-Carboxamides as Potential Chemosensitizing Agents for Cancer

, 8(3): 268 - 275

Vinaykumar S. Velingkar and Vikrant D. Dandekar


DOI: 10.2174/157018011794578169




Synthesis, Characterization of Some New Five Membered Heterocycles Based on Imidazole Moiety and their Applications on Therapeutics

, 8(3): 276 - 283

V. S.V. Satyanarayana, A. Sivakumar and Asit Ranjan Ghosh


DOI: 10.2174/157018011794578196




Gallic Acid-Phospholipid Complex: Drug Incorporation and Physicochemical Characterization

, 8(3): 284 - 291

Devendra Singh, Mohan Singh Maniyari Rawat, Ajay Semalty and Mona Semalty


DOI: 10.2174/157018011794578240




THIS ARTICLE HAS BEEN RETRACTED

, 8(3): 292 - 301

Kadria A. Elkhodairy, Nahla S. Barakat and Fars K. Alanazi


DOI: 10.2174/157018011794578141




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