Letters in Drug Design & Discovery
Volume 18, 12 Issues, 2021
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access
Contents
Letters in Drug Design & Discovery, Volume 8 - Number 10
MGBG in Combined Anticancer Chemotherapy
, 8(10): 897 - 903R. F. Goncalves, G. Kriechammer and M. P.M. Marques
DOI: 10.2174/157018011797655197
Titanocene Y and Vanadocene Y: Platinum Resistance-Breaking Cytotoxic and DNA-Targeting Anticancer Drug Candidates
, 8(10): 904 - 910Ralf A. Hilger, Dennis Alex, Anthony Deally, Brendan Gleeson and Matthias Tacke
DOI: 10.2174/157018011797655241
Synthesis and Biological Evaluation of Licofelone Derivatives as Anticancer and Anti-inflammatory Agents
, 8(10): 911 - 917Wukun Liu, Jinpei Zhou, Huibin Zhang, Hai Qian, Jiahan Yin, Kerstin Bensdorf and Ronald Gust
DOI: 10.2174/157018011797655223
A QSAR Study on a Series of Indolin-2-Ones Acting as Non-Receptor Src Tyrosine Kinase Inhibitors
, 8(10): 918 - 925Zaihra Anwer and Satya P. Gupta
DOI: 10.2174/157018011797655250
3D-QSAR Studies of VEGFR-2 Kinase Inhibitors Based on Docking
, 8(10): 926 - 942Xiaoping Jiang, Guangchuan Ou, Depeng Yan, Min Zhang and Xianyou Yuan
DOI: 10.2174/157018011797655296
Synthesis and Preliminary Screening of Novel A- and D-Ring Modified Steroids as Aromatase Inhibitors
, 8(10): 943 - 950Mange Ram Yadav, Prafulla M. Sabale, Rajani Giridhar, Dharmendra Baria, Christina Zimmer and Rolf W. Hartmann
DOI: 10.2174/157018011797655322
A Novel Bromomelatonin Derivative Suppresses Apoptosis with Regulating the Expression of Bcl-2 Family Genes
, 8(10): 951 - 956Yoshikazu Mikami, Masanori Somei, Eri Watanabe, Nobukazu Watanabe, Tomihisa Takahashi and Masaki J. Honda
DOI: 10.2174/157018011797655287
Synthesis of Cinnamide Dimers as Potential Antibacterial and Antifungal Agents
, 8(10): 957 - 965Ahmed Kamal, G. Ramakrishna, P. Raju, A. V. Subba Rao, Joveeta Joseph, B. Siddhardha and U. S.N. Murty
DOI: 10.2174/157018011797655205
Novel Clarithromycin Analogs with C-4” 2-arylbenzimidazolyl Bishydrazide Side Chain: Synthesis and Antibacterial Evaluation
, 8(10): 966 - 971Yunkun Qi, Ruixin Ma, Xin Li, Yue Hu, Siti Ma, Chao Cong, Xiaodong Ma, Wenping Cui and Shutao Ma
DOI: 10.2174/157018011797655269
Synthesis and Antibacterial Activity of 6-Substituted Anacardic Acid Derivatives
, 8(10): 972 - 979Subhakara Reddy Nallamilli, Ravi Kumar V, Himabindu V, B. Ram and Srinivas Rao Aalapati
DOI: 10.2174/157018011797655278
Antimicrobial Efficacy of Metal-Barbiturate Conjugates Against Pathogenic Strains of Escherichia coli and Staphylococcus aureus
, 8(10): 980 - 987Ashfaq Mahmood Qureshi, Mehmood Qadir, Abdul Rauf, Muhammad Idrees, Siara Mumtaz, Muhammad Najam-ul-Haq, Muhammad Ismail, Muhammad Athar, Rashid Khushal, Sara Riaz and Habib Bokhari
DOI: 10.2174/157018011797655232
Synthesis of 2-methyl-3-(2-(piperazin-1-yl)ethyl)-6,7,8,9-tetrahydro-4Hpyrido[ 1,2-a]pyrimidin-4-one Derivatives as Antimicrobial Agents
, 8(10): 988 - 995Byregowda Krishnamurthy, Kambappa Vinaya, Doddakunche S. Prasanna, Byregowda Raghava and Kanchugarakoppal S. Rangappa
DOI: 10.2174/157018011797655304
Molecular Mapping and Docking Interactions for Selective Anti-Fertility Potency of Estrogen Analogs
, 8(10): 996 - 1003Ria Pal, Md Ataul Islam, Tabassum Hossain and Achintya Saha
DOI: 10.2174/157018011797655214
Antioxidant Evaluation of Some Semicarbazide, 1,2,4-Triazolone and Pyrazolone Derivatives
, 8(10): 1004 - 1008Monika Pitucha and Renata Nowak
DOI: 10.2174/157018011797655188
A New Practice: Study on the Molecular Mechanism of Traditional Chinese Medicine by Computational Pharmacology Methods: Part 2: Pharmacodynamic Modeling and Distribution on Ligand-Target Space of Effective Components
, 8(10): 1009 - 1014Ding-Hong Wu, Xiao-Jie Xu, Min-Zhou Zhang and Lei Wang
DOI: 10.2174/157018011797655331
Editor-in-Chief
K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
Biography
University of Hradec Kralove
Hradec Kralove
Biography
Biography of K. Kuca
Kamil Kuca is working for several academic institutes (University of Hradec Kralove, Czech Republic; University Hospital Hradec Kralove, Czech republic; Florida International University, USA; Yangtze University, China; etc.). He is recently rector of the University of Hradec Kralove. He was also technology scout focused on biomedicine in the past. His research interests are toxicology, pharmacology, drug design, technology transfer, pharmacoeconomy, chemical and biological terrorism, etc. He was/is principal investigator on numerous national and international projects (EU, NATO, GACR, IGA MZ, MSMT etc.). He has published more than 350 IF research papers. He is working with several companies as a scientific consultant. He has lots of cooperators throughout the world (e.g. Korea, Croatia, United Arab Emirates, USA, France, Turkey, China, Singapore, Sweden, and Brazil). His Hindex is 36, number of citation in WoS is over 3000.
About the Journal
For Authors
For Librarians & Readers
Quick Links
Journal History
Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 2.0
Webmaster Contact: info@benthamscience.net