Contents

Letters in Drug Design & Discovery, Volume 8 - Number 10

Graphical Abstracts

, 8(10): i - v


DOI: 10.2174/157018011797655313




MGBG in Combined Anticancer Chemotherapy

, 8(10): 897 - 903

R. F. Goncalves, G. Kriechammer and M. P.M. Marques


DOI: 10.2174/157018011797655197




Titanocene Y and Vanadocene Y: Platinum Resistance-Breaking Cytotoxic and DNA-Targeting Anticancer Drug Candidates

, 8(10): 904 - 910

Ralf A. Hilger, Dennis Alex, Anthony Deally, Brendan Gleeson and Matthias Tacke


DOI: 10.2174/157018011797655241




Synthesis and Biological Evaluation of Licofelone Derivatives as Anticancer and Anti-inflammatory Agents

, 8(10): 911 - 917

Wukun Liu, Jinpei Zhou, Huibin Zhang, Hai Qian, Jiahan Yin, Kerstin Bensdorf and Ronald Gust


DOI: 10.2174/157018011797655223




A QSAR Study on a Series of Indolin-2-Ones Acting as Non-Receptor Src Tyrosine Kinase Inhibitors

, 8(10): 918 - 925

Zaihra Anwer and Satya P. Gupta


DOI: 10.2174/157018011797655250




3D-QSAR Studies of VEGFR-2 Kinase Inhibitors Based on Docking

, 8(10): 926 - 942

Xiaoping Jiang, Guangchuan Ou, Depeng Yan, Min Zhang and Xianyou Yuan


DOI: 10.2174/157018011797655296




Synthesis and Preliminary Screening of Novel A- and D-Ring Modified Steroids as Aromatase Inhibitors

, 8(10): 943 - 950

Mange Ram Yadav, Prafulla M. Sabale, Rajani Giridhar, Dharmendra Baria, Christina Zimmer and Rolf W. Hartmann


DOI: 10.2174/157018011797655322




A Novel Bromomelatonin Derivative Suppresses Apoptosis with Regulating the Expression of Bcl-2 Family Genes

, 8(10): 951 - 956

Yoshikazu Mikami, Masanori Somei, Eri Watanabe, Nobukazu Watanabe, Tomihisa Takahashi and Masaki J. Honda


DOI: 10.2174/157018011797655287




Synthesis of Cinnamide Dimers as Potential Antibacterial and Antifungal Agents

, 8(10): 957 - 965

Ahmed Kamal, G. Ramakrishna, P. Raju, A. V. Subba Rao, Joveeta Joseph, B. Siddhardha and U. S.N. Murty


DOI: 10.2174/157018011797655205




Novel Clarithromycin Analogs with C-4” 2-arylbenzimidazolyl Bishydrazide Side Chain: Synthesis and Antibacterial Evaluation

, 8(10): 966 - 971

Yunkun Qi, Ruixin Ma, Xin Li, Yue Hu, Siti Ma, Chao Cong, Xiaodong Ma, Wenping Cui and Shutao Ma


DOI: 10.2174/157018011797655269




Synthesis and Antibacterial Activity of 6-Substituted Anacardic Acid Derivatives

, 8(10): 972 - 979

Subhakara Reddy Nallamilli, Ravi Kumar V, Himabindu V, B. Ram and Srinivas Rao Aalapati


DOI: 10.2174/157018011797655278




Antimicrobial Efficacy of Metal-Barbiturate Conjugates Against Pathogenic Strains of Escherichia coli and Staphylococcus aureus

, 8(10): 980 - 987

Ashfaq Mahmood Qureshi, Mehmood Qadir, Abdul Rauf, Muhammad Idrees, Siara Mumtaz, Muhammad Najam-ul-Haq, Muhammad Ismail, Muhammad Athar, Rashid Khushal, Sara Riaz and Habib Bokhari


DOI: 10.2174/157018011797655232




Synthesis of 2-methyl-3-(2-(piperazin-1-yl)ethyl)-6,7,8,9-tetrahydro-4Hpyrido[ 1,2-a]pyrimidin-4-one Derivatives as Antimicrobial Agents

, 8(10): 988 - 995

Byregowda Krishnamurthy, Kambappa Vinaya, Doddakunche S. Prasanna, Byregowda Raghava and Kanchugarakoppal S. Rangappa


DOI: 10.2174/157018011797655304




Molecular Mapping and Docking Interactions for Selective Anti-Fertility Potency of Estrogen Analogs

, 8(10): 996 - 1003

Ria Pal, Md Ataul Islam, Tabassum Hossain and Achintya Saha


DOI: 10.2174/157018011797655214




Antioxidant Evaluation of Some Semicarbazide, 1,2,4-Triazolone and Pyrazolone Derivatives

, 8(10): 1004 - 1008

Monika Pitucha and Renata Nowak


DOI: 10.2174/157018011797655188




A New Practice: Study on the Molecular Mechanism of Traditional Chinese Medicine by Computational Pharmacology Methods: Part 2: Pharmacodynamic Modeling and Distribution on Ligand-Target Space of Effective Components

, 8(10): 1009 - 1014

Ding-Hong Wu, Xiao-Jie Xu, Min-Zhou Zhang and Lei Wang


DOI: 10.2174/157018011797655331




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