Contents

Letters in Drug Design & Discovery, Volume 8 - Number 1

Graphical Abstracts

, 8(1): i - v


DOI: 10.2174/157018011793663895




Binding Modes of 2-Phenylamino-6-oxopurines to Herpes Simplex Virus Thymidine Kinases

, 8(1): 1 - 8

Federico Focher, Andrea Lossani, Andrea Torti, Joseph Gambino and George E. Wright


DOI: 10.2174/157018011793663877




Design, Synthesis and Pharmacokinetic Evaluation of a Novel Series of Triazole-Based Src Kinase Inhibitors with Anti-proliferative Activity

, 8(1): 9 - 13

Shaojun Chen, Chuansheng Guo, Shiting Shi, Yanyan Shi, Du Fang and Houxing Fan


DOI: 10.2174/157018011793663930




QSAR Analysis of Isosteviol Derivatives as α-Glucosidase Inhibitors with Element Count and Other Descriptors

, 8(1): 14 - 25

N. S. Hari Narayana Moorthy, Maria J. Ramos and Pedro A. Fernandes


DOI: 10.2174/157018011793663859




Synthesis and In Vitro Biochemical Evaluation of a Series of Alkyl 6- Aminosulfonyl Naphthanoates as Potential Inhibitors of Human Placental Estrone Sulfatase (ES)

, 8(1): 26 - 31

Chirag K. Patel and Sabbir Ahmed


DOI: 10.2174/157018011793663967




QSAR Study on 5-Lipoxygenase Activating Protein (FLAP) Inhibitors: The Derivatives of 2,2-Bisaryl-Bicycloheptane

, 8(1): 32 - 43

Brij Kishore Sharma, Pradeep Pilania and Prithvi Singh


DOI: 10.2174/157018011793663903




Volsurf Descriptors to Analyse Anti-HCV and Cytotoxic Activities of Sesquiterpene Lactones from Asteraceae Family

, 8(1): 44 - 58

Mariane Ballerini Fernandes, Michelle Rossini, Ricardo Stefani, Leoberto Tavares, Vicente de Paulo Emerenciano, Luciana Scotti, Marcelo Sobral da Silva and Marcus Tullius Scotti


DOI: 10.2174/157018011793663868




Design, Synthesis and Anti Colon Cancer Activity Evaluation of Phosphorylated Derivatives of Lamivudine (3TC)

, 8(1): 59 - 64

Valasani Koteswara Rao, Sanapalli S. Reddy, Balam S. Krishna, Cirandur S. Reddy, Nimmanapalli P. Reddy, Tamatam C.M. Reddy, Chamarthi N. Raju and S. K. Ghosh


DOI: 10.2174/157018011793663921




Ethyl Gallate as a Combination Drug Can Overcome Resistance in MRSA

, 8(1): 65 - 68

Win Mar Soe, Nyan Lin Myint, Lim Chu Sing, Meena K. Sakharkar, Thean Hock Tang and Kishore R. Sakharkar


DOI: 10.2174/157018011793663949




Effects of Honey Against the Accumulation of Adipose Tissue and the Increased Blood Pressure on Carbohydrate-Induced Obesity in Rat

, 8(1): 69 - 75

Samanta Romero-Silva, Miguel Angel Martinez R, Laura P. Romero-Romero, Oralia Rodriguez, C. Gerardo Salas G, Nicole Morel, Francisco Javier Lopez-Munoz, Luis Angel Lima-Mendoza and Guadalupe Bravo


DOI: 10.2174/157018011793663912




Synthesis and Biological Evaluation of Nitric Oxide-releasing Derivatives of Capsaicin as Analgesia Drugs

, 8(1): 76 - 81

Liang Ge, jingjie Wang, Xiaoyan Zhang, Huibin Zhang, Hai Qian, Wenlong Huang and Jinpei Zhou


DOI: 10.2174/157018011793663831




Synthesis and Evaluation of Antimicrobial Activity of Thiazolidinone Derivatives

, 8(1): 82 - 86

Ravichandran Veerasamy, Harish Rajak, Krishnan Suresh Kumar and Ram Kishore Agrawal


DOI: 10.2174/157018011793663958




Enhancing Oral Bioavailability of Methylnaltrexone Using an Emulsion Formulation

, 8(1): 87 - 92

Li-Fang Yu, Wei-Gen Lu, Ping Xiang, Li-Li Wang, Li Chen, Ting-Ting Chen, Michael Maojian Gu, Chong-Zhi Wang and Chun-Su Yuan


DOI: 10.2174/157018011793663886




Discovery of BRM Targeted Therapies: Novel Reactivation of an Anticancer Gene

, 8(1): 93 - 99

Sarah Gramling and David Reisman


DOI: 10.2174/157018011793663840




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