Contents

Letters in Drug Design & Discovery, Volume 7 - Number 9

Graphical Abstracts

, 7(9): i - v


DOI: 10.2174/157018010792929531




Exploring QSAR on 4-Cyclohexylmethoxypyrimidines as Antitumor Agents for Their Inhibitory Activity of CDK2

, 7(9): 625 - 631

A. Ece and F. Sevin


DOI: 10.2174/157018010792929612




4-Hydroxy-3-methoxyphenyl Substituted 3-methyl-tetrahydroquinoline Derivatives Obtained Through Imino Diels-Alder Reactions as Potential Antitumoral Agents

, 7(9): 632 - 639

Vladimir V. Kouznetsov, Diego R. Merchan Arenas, Francisco Arvelo, Josue S. Bello Forero, Felipe Sojo and Arturo Munoz


DOI: 10.2174/157018010792929577




Novel 3-(1-acetyl-5-(substituted-phenyl)-4,5-dihydro-1H-pyrazol-3-yl)-7-fluoro-2H-chromen-2-one Derivatives: Synthesis and Anticancer Activity

, 7(9): 640 - 643

Zheng-Yu Cai, Yang Yang, Xin-Hua Liu and Xing-Bao Qi


DOI: 10.2174/157018010792929540




Design, Synthesis and In Vitro Anticancer Activity of a New Class of Bifunctional DNA Intercalators

, 7(9): 644 - 649

Ana Maria V. Zbancioc, Gheorghita N. Zbancioc, Catalin Tanase, Anca Miron, Cornelia Ursu and Ionel I. Mangalagiu


DOI: 10.2174/157018010792929504




Estrone (E1) Based Esters as Potential Inhibitors of Type 3 17β- hydroxysteroid Dehydrogenase (17β-HSD3) in the Treatment of Hormone-Dependent Prostate Cancer

, 7(9): 650 - 656

Moniola S. Olusanjo and Sabbir Ahmed


DOI: 10.2174/157018010792929496




Antioxidant Capacity of 2-(3,5-diaryl-4,5-dihydro-1H-pyrazol-1-yl)-4-phenylthiazoles

, 7(9): 657 - 660

F. A.N. Silva, L. Pizzuti, F. H. Quina, S. P. Souza, P. F. Rosales, G. M. Siqueira, C. M.P. Pereira, S. B.M. Barros and D. P. Rivelli


DOI: 10.2174/157018010792929513




Synthesis and Anticonvulsant Activity of Some Cinnamylpiperazine Derivatives

, 7(9): 661 - 664

Chuan Hu, Zhi-Gang Sun, Cheng-Xi Wei and Zhe-Shan Quan


DOI: 10.2174/157018010792929595




Synthesis of Cyclodextrin Derivatives of Amino-(thiazolyl) Coumarins as Potential Antimicrobial Agents

, 7(9): 665 - 673

Ahmed Kamal, S. F. Adil, Jaki R. Tamboli, B. Siddardha and U. S.N. Murthy


DOI: 10.2174/157018010792929559




3-(1-Adamantylthio)-4-Phenylpyridine as a Potential Therapeutic for Methicillin-Resistant Staphylococcus aureus

, 7(9): 674 - 678

Ratana Lawung, Lertyot Treeratanapiboon, Supaluk Prachayasittikul and Virapong Prachayasittikul


DOI: 10.2174/157018010792929603




In Vitro Antiprotozoal Evaluation of Zinc and Copper Complexes Based on Sulfonamides Containing 8-Aminoquinoline Ligands

, 7(9): 679 - 685

Luiz Everson da Silva, Paulo Teixeira de Sousa Jr., Eduardo Nunes Maciel, Rebeca Korting Nunes, Iriane Eger, Mario Steindel and Ricardo Andrade Rebelo


DOI: 10.2174/157018010792929586




Synthesis and In Vivo Acute Antihyperglycemic Evaluation of Novel Isosteviol Derivatives

, 7(9): 686 - 693

Junqing Chen, Xiaoming Zha, Min Sun, Jin Cai, Wen Zhou and Min Ji


DOI: 10.2174/157018010792929522




Recent Advancement in the Field of Anticonvulsants: A Review

, 7(9): 694 - 706

Shailendra Pandey and Radhey Shyam Srivastava


DOI: 10.2174/157018010792929487




A Tribute to Octavio Antunes: A Brazilian Approach to Protease Inhibitors

, 7(9): 707 - 709

Jose C. Barros, Rodrigo Octavio M.A. de Souza, Joaquim F.M. da Silva, Eloan dos S. Pinheiro and Amilcar Tanuri


DOI: 10.2174/157018010792929568




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