Contents

Letters in Drug Design & Discovery, Volume 7 - Number 7

Graphical Abstracts

, 7(7): i - iv


DOI: 10.2174/157018010791526331




Synthesis and Evaluation of Haloacetyl, α-Bromoacryloyl and Nitrooxyacetyl Benzo[b]furan and Benzo[b]thiophene Derivatives as Potent Antiproliferative Agents Against Leukemia L1210 and K562 Cells

, 7(7): 476 - 486

Romeo Romagnoli, Pier Giovanni Baraldi, Maria Dora Carrion, Carlota Lopez Cara, Alberto Casolari, Ernest Hamel, Enrica Fabbri and Roberto Gambari


DOI: 10.2174/157018010791526296




Synthesis of Xanthones and Benzophenones as Inhibitors of Tumor Cell Growth

, 7(7): 487 - 493

Elisangela Costa, Emilia Sousa, Nair Nazareth, Maria S.J. Nascimento and Madalena M.M. Pinto


DOI: 10.2174/157018010791526250




Chemometric Evaluation of the Significance of Molecular Structural Descriptors on Binding of Acridinone Derivatives to DNA

, 7(7): 494 - 499

Marcin Koba and Tomasz Baczek


DOI: 10.2174/157018010791526278




Reversion of Multidrug Resistance Using Self-Organized Nanoparticles Holding Both Doxorubicin and Targeting Moiety

, 7(7): 500 - 506

Yu Cao, Ying Gu, Lina Liu, Yi Yang, Peiguang Zhao, Ping Su, Liyan Liu, Chao Qi, Xia Lei and Changjiang Yang


DOI: 10.2174/157018010791526322




Biphenyl-Derivatives Possessing Tertiary Amino Groups as β-Secretase (BACE1) Inhibitors

, 7(7): 507 - 515

Simone Bertini, Elisa Ghilardi, Valentina Asso, Carlotta Granchi, Filippo Minutolo and Marco Macchia


DOI: 10.2174/157018010791526304




Potency of HI-6 to Reactivate Cyclosarin, Soman and Tabun Inhibited Acetylcholinesterase – In Vivo Study

, 7(7): 516 - 520

Jana Zdarova Karasova, Jiri Kassa, Miroslav Pohanka, Kamil Musilek and Kamil Kuca


DOI: 10.2174/157018010791526269




Triterpenes from Gloeophyllum odoratum as Potential Leads Towards Potent Thrombin Inhibitors

, 7(7): 521 - 527

Francesca Cateni, Vittorio Lucchini, Marko Anderluh, Paolo Martinuzzi, Marina Zacchigna, Andrej Piltaver and Bojan Doljak


DOI: 10.2174/157018010791526340




Molecular Modeling Suggests Cruzain Specificity for Peptide Primaquine Prodrugs

, 7(7): 528 - 533

Gustavo Henrique Goulart Trossini, Chung Man Chin, Carla Maria de Souza Menezes and Elizabeth Igne Ferreira


DOI: 10.2174/157018010791526287




Synthesis, Characterization by Means of IR, 1H, 13C - NMR and Biological Investigations on New Diorganotin Carboxylic Acid Derivatives

, 7(7): 534 - 540

Abderrahmane Yahyi, Abdelkader Et-Touhami, Rachid Yahyaoui and Rachid Touzani


DOI: 10.2174/157018010791526241




Inhibition of Pigment Epithelium-Derived Factor (PEDF) Augments Vascular Endothelial Growth Factor (VEGF)-Induced Recovery of Limb Perfusion after Ischemia in Klotho Mouse

, 7(7): 541 - 545

Ken Arima, Sho-ichi Yamagishi, Takanori Matsui, Yutaka Saito, Yoshio Katsuki, Ken-ichiro Sasaki, Yousuke Katsuda, Hisashi Kai and Tsutomu Imaizumi


DOI: 10.2174/157018010791526313




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