Contents

Letters in Drug Design & Discovery, Volume 7 - Number 4

Graphical Abstracts

, 7(4): i - iv


DOI: 10.2174/157018010790945850




Novel Thiazolidinone Derivatives with an Uncommon Mechanism of Inhibition Towards HIV-1 Reverse Transcriptase

, 7(4): 228 - 234

Eleni Pitta, Emmanuele Crespan, Athina Geronikaki, Giovanni Maga and Alberta Samuele


DOI: 10.2174/157018010790945869




Synthesis and Biological Evaluation of Dihydroisoquinoline-2(1H)- Carbothioamide Derivatives as TRPV1 Antagonists

, 7(4): 235 - 237

Hai Qian, Wei Chen, Xiaoyan Zhang, Huibin Zhang, Jinpei Zhou, Wenlong Huang, Jing Jin and Dongyan Dai


DOI: 10.2174/157018010790945797




Novel 5-Methyl-2,4-Disubstitued-Oxazole Derivatives: Synthesis and Anticancer Activity

, 7(4): 238 - 243

Xin-Hua Liu, Hui-Feng Liu, Chun-Xiou Pan, Jin-Xin Li, Lin-Shan bai, Bao-An Song and Xiang-Feng Chu


DOI: 10.2174/157018010790945878




A Novel Trypsin and α-Chymotrypsin Inhibitor from Maclura pomifera Seeds

, 7(4): 244 - 249

C. M. Lazza, S. A. Trejo, W. D. Obregon, L. G. Pistaccio, N. O. Caffini and L. M.I. Lopez


DOI: 10.2174/157018010790945832




Synthesis, Characterization and Evaluation of Cytotoxicity of New Aminophosphonic Acid Diesters in Human Leukemia Cells

, 7(4): 250 - 259

Avula Balakrishna, Kishore K. Chiruvella, Mudumala V.N. Reddy, Rajesh Reddy, Sandip K. Nayak, Sathees C. Raghavan and Cirandur S. Reddy


DOI: 10.2174/157018010790945841




Novel Nucleophilic Compounds with Oxime Group as Reactivators of Paraoxon-Inhibited Cholinesterases

, 7(4): 260 - 264

Lucie Musilova, Daniel Jun, Jiri Palecek, Vladimir Cirkva, Kamil Musilek, Martin Paar, Martina Hrabinova, Miroslav Pohanka and Kamil Kuca


DOI: 10.2174/157018010790945823




3-Substituted Isocoumarins as Thymidine Phosphorylase Inhibitors

, 7(4): 265 - 268

Khalid Mohammed Khan, Sumbul Ahmed, Sajjad Hussain, Nida Ambreen, Shahnaz Perveen and M. Iqbal Choudhary


DOI: 10.2174/157018010790945805




Three Dimensional Molecular Field Analysis of Thiomorpholine Analogs of TACE Inhibitors Using Receptor Based Alignment

, 7(4): 269 - 274

Malkeet Singh Bahia, Neha Bagga, Rambabu Gundla and Om Silakari


DOI: 10.2174/157018010790945779




Synthesis and Cytotoxic Evaluation of Disubstituted N-Acylhydrazones Pyrazinecarbohydrazide Derivatives

, 7(4): 275 - 280

Marcelle de L. Ferreira, Andre L.P. Candea, Maria das Gracas M. de O. Henriques, Carlos R. Kaiser, Camilo H. da S. Lima and Marcus V.N. de Souza


DOI: 10.2174/157018010790945814




Design, Synthesis and In Vivo Evaluation of Sulfhydryl β-D-Glucose Cholesterols as Ligands for Brain Targeting Liposomes

, 7(4): 281 - 289

Wei Fan, Chengyi Yan, Shan Qian, Nian Yao, Lei Tang and Yong Wu


DOI: 10.2174/157018010790945788




The Development of PDGF Receptor Inhibitors for the Treatment of Glioma: A Review

, 7(4): 290 - 299

Michael A. Badruddoja, Emad Elquza, James Welsh, Laurence Cooke, Abhay Sanan, Baldassrre Stea and Daruka Mahadavan


DOI: 10.2174/157018010790945887




Making Drops in Microencapsulation Processes

, 7(4): 300 - 309

L. Martin-Banderas, A. M. Ganan-Calvo and M. Fernandez-Arevalo


DOI: 10.2174/157018010790945760




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