Contents

Letters in Drug Design & Discovery, Volume 7 - Number 1

Graphical Abstracts

, 7(1): v


DOI: 10.2174/157018081100701000v




New Bisquaternary Isoquinolinium Inhibitors of Brain Cholinesterases - Synthesis and Anticholinesterase Activity

, 7(1): 1 - 4

Jiri Binder, Martin Paar, Daniel Jun, Miroslav Pohanka, Martina Hrabinova, Veronika Opletalova and Kamil Kuca


DOI: 10.2174/1570180811007010001




Design, Synthesis, and Biological Evaluation of 7H-thiazolo[3,2-b]-1,2,4-triazin-7-one Derivatives as Acetylcholinesterase Inhibitors

, 7(1): 5 - 8

Si-Jie Liu, Liu Yang, Xiao-Guang Liu, Ying Luo, Zi-Jian Cao, David Chi Cheong Wan, Huang-Quan Lin and Chun Hu


DOI: 10.2174/157018010789869343




Synthesis of the Neurotransmitter 4-Aminobutanoic Acid (GABA) from Diethyl Cyanomalonate

, 7(1): 9 - 13

Matthew C. Cook, Ross D. Witherell and Robert L. White


DOI: 10.2174/157018010789869361




Structure Activity Relationship of Organic Alcohol and Esters for Antidepressant- Like Activity

, 7(1): 14 - 17

Shahnaz Perveen, Arfa Yasmeen, Muhammad Aitmaud Khan, Ahsana Dar, Rehana Jafri and Amir Ahmed


DOI: 10.2174/157018010789869334




Synthesis and Biological Study of 3-Butyl-1-(2,6-dichlorophenyl)-1H-[1,2,4]triazol- 5(4H)-one Derivatives as Anti-hypertension Drugs

, 7(1): 18 - 22

Yanchun Zhang, Jinpei Zhou, Weihong Pan, Xiaoming Wu and Shuai Wang


DOI: 10.2174/157018010789869370




The Antisense Oligonucleotides Decrease Expression of the Cellular Prion

, 7(1): 23 - 26

Vitalii V. Stadnyk, Lyudmyla A. Izyumova, Yuriy A. Rzhepetskiy, Chrystyna Ya Mayor and Vasyl V. Vlizlo


DOI: 10.2174/157018010789869299




Synthesis and Preliminary Biological Activity of Some New Pyrazole Derivatives as Acyclonucleoside Analogues

, 7(1): 27 - 30

Smaail Radi, Souad Salhi and Amal Radi


DOI: 10.2174/157018010789869307




Synergistic Combinations of Chitosans and Antibiotics in Staphylococcus aureus

, 7(1): 31 - 35

San Tin, Chu Sing Lim, Meena Kishore Sakharkar and Kishore Ramaji Sakharkar


DOI: 10.2174/157018010789869406




Structure Function Relationships of KTS Disintegrins and Design of Antiangiogenic Drugs

, 7(1): 36 - 40

Olfa Kallech-Ziri, Jose Luis, Ziad Faljoun, Jean-Marc Sabatier, Maxime Lehmann, Mohamed El Ayeb, Naziha Marrakchi and Erwann Loret


DOI: 10.2174/157018010789869325




Synthesis and Biological Activity of New Triazole Compounds

, 7(1): 41 - 45

Hanane Al Bay, Bouchra Quaddouri, Abdelkarim Guaadaoui, Rachid Touzani, Nour-Eddine Benchat, Abdellah Hamal, Mustafa Taleb, Mohammed Bellaoui and Sghir El Kadiri


DOI: 10.2174/157018010789869352




Synthesis and In Vitro Evaluation of Novel 1, 2, 4-Triazole Derivatives as Antifungal Agents

, 7(1): 46 - 49

Ganesh R. Kokil, Prarthana V. Rewatkar, Sandeep Gosain, Saurabh Aggarwal, Arunima Verma, Atin Kalra and Suresh Thareja


DOI: 10.2174/157018010789869415




Physicochemical Interaction Study of Non-Steroidal Anti-Inflammatory Drugs with Dimyristoylphosphatidylethanolamine Liposomes

, 7(1): 50 - 56

Marcela Manrique-Moreno, Jorg Howe, Mario Suwalsky, Patrick Garidel and Klaus Brandenburg


DOI: 10.2174/157018010789869280




Homology Modelling of Human E1 Ubiquitin Activating Enzyme

, 7(1): 57 - 62

Ghali Brahemi, Angelika M. Burger, Andrew D. Westwell and Andrea Brancale


DOI: 10.2174/157018010789869316




Preparation of Tiagabine HCl/2-HPβCD Complex Pellets by Extrusion-Spheronization Using Glycerol Monostearate as Pellet-Aid

, 7(1): 63 - 69

Abdussalam Sughir, Malika Lahiani-Skiba and Mohamed Skiba


DOI: 10.2174/157018010789869389




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