Contents

Letters in Drug Design & Discovery, Volume 6 - Number 7

Solification with Hydrobromic Acid as a Factor Defining the Antiarrhythmic Effect of Lappaconitine Derivatives

, 6(7): 475 - 477

T. G. Tolstikova, A. O. Bryzgalov, I. V. Sorokina, S. A. Osadchii, E. E. Shults, M. P. Dolgikh and M. V. Khvostov


DOI: 10.2174/157018009789108312




Synthesis and Biological Evaluation of Bridged Analogues of the Platelet Aggregation Inhibitor Trifenagrel

, 6(7): 478 - 486

Magdalena Slusarczyk, Wim M. De Borggraeve, Georges Hoornaert, Koen Robeyns, Luc Van Meervelt, Tongfei Wu, Frederik Deroose and Joannes T.M. Linders


DOI: 10.2174/157018009789108213




Targeting the Peptide Deformylase of Mycobacterium tuberculosis Leads to Drug Discovery

, 6(7): 487 - 493

Vijai Singh and Pallavi Somvanshi


DOI: 10.2174/157018009789108286




In Silico Screening of Novel Inhibitors for HPV: A Rational Structure Based Approach (Docking Versus Pharmacophore Model Generation)

, 6(7): 494 - 501

G. Reshmi and M. Radhakrishna Pillai


DOI: 10.2174/157018009789108321




Microwave-Assisted Solvent-Free Synthesis of N-alkyl Benzotriazole Derivatives: Antimicrobial Studies

, 6(7): 502 - 507

Raghu Ningegowda, C. V. Kavitha, B. S. Priya, S. L. Gaonkar, M. V. Tejesvi, K. S. Rangappa and S. Nanjunda Swamy


DOI: 10.2174/157018009789108222




New Pyrrole Hydrazones Synthesized and Evaluated In Vitro as Potential Tuberculostatics

, 6(7): 508 - 517

A. Bijev, S. Vladimirova and P. Prodanova


DOI: 10.2174/157018009789108268




Synthesis and Biochemical Evaluation of a Series of Methanesulfonate Derivatives of 4-Hydroxyphenyl Ketone as Probes of the Active Site of Type 3 OF 17β-Hydroxysteroid Dehydrogenase Family of Enzymes

, 6(7): 518 - 523

Kruti Shah, Moniola S. Olusanjo, Tim Cartledge, Caroline P. Owen and Sabbir Ahmed


DOI: 10.2174/157018009789108259




Synthesis and Biochemical Evaluation of a Range of 2-, 3- and 4-Substituted Derivatives of Benzyl Imidazole-Based Compounds as Probes of the Active Site of 17α-hydroxylase/17,20-Lyase (P45017α)

, 6(7): 524 - 530

Sabbir Ahmed, Imran Shahid, Kishore K. Bhatti, Wai-Yee Lee and Caroline P. Owen


DOI: 10.2174/157018009789108295




On the Synthesis and Anticancer Testing of α,β-Unsaturated Ketones as Analogs of Combretastatin-A4

, 6(7): 531 - 537

Sameer Chavda, Ryan Davis, Amanda Ferguson, Camille Riddering, Kristin Dittenhafer, Hilary Mackay, Balaji Babu, Moses Lee, Adam Siegfried, William Pennington, Miriam Shadfan, Susan L. Mooberry, Bijay K. Mishra and Hari N. Pati


DOI: 10.2174/157018009789108277




Design, Synthesis, Crystal Structure and Antitumor Activity of A New Ethyl 3-(quinazolin-4-ylamino)-1H-pyrrole-2-carboxylate Derivative

, 6(7): 538 - 541

Youguang Zheng, Xiaoqing Wu, Min Sun, Liuhai Feng, Mingdong Li and Min Ji


DOI: 10.2174/157018009789108240




Enhanced Brain Targeting of Tegafur Using Novel Lactyl Cholesterol Liposome as a Carrier

, 6(7): 542 - 547

Wei Fan, Xiankun Li, Shan Qian, Shan Wang and Yong Wu


DOI: 10.2174/157018009789108303




Synthesis, Anticonvulsant Evaluation of 2,3,4,5-Tetrahydro-7-alkoxy-1H-2-benzazepin-1-ones

, 6(7): 548 - 553

Cheng-Xi Wei, Wei Zhang, Zhe-Shan Quan, Rong-Bi Han, Ri-Shan Jiang and Feng-Yu Piao


DOI: 10.2174/157018009789108231




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