Letters in Drug Design & Discovery, Volume 6 - Number 7

Solification with Hydrobromic Acid as a Factor Defining the Antiarrhythmic Effect of Lappaconitine Derivatives

, 6(7): 475 - 477

T. G. Tolstikova, A. O. Bryzgalov, I. V. Sorokina, S. A. Osadchii, E. E. Shults, M. P. Dolgikh and M. V. Khvostov

DOI: 10.2174/157018009789108312

Synthesis and Biological Evaluation of Bridged Analogues of the Platelet Aggregation Inhibitor Trifenagrel

, 6(7): 478 - 486

Magdalena Slusarczyk, Wim M. De Borggraeve, Georges Hoornaert, Koen Robeyns, Luc Van Meervelt, Tongfei Wu, Frederik Deroose and Joannes T.M. Linders

DOI: 10.2174/157018009789108213

Targeting the Peptide Deformylase of Mycobacterium tuberculosis Leads to Drug Discovery

, 6(7): 487 - 493

Vijai Singh and Pallavi Somvanshi

DOI: 10.2174/157018009789108286

In Silico Screening of Novel Inhibitors for HPV: A Rational Structure Based Approach (Docking Versus Pharmacophore Model Generation)

, 6(7): 494 - 501

G. Reshmi and M. Radhakrishna Pillai

DOI: 10.2174/157018009789108321

Microwave-Assisted Solvent-Free Synthesis of N-alkyl Benzotriazole Derivatives: Antimicrobial Studies

, 6(7): 502 - 507

Raghu Ningegowda, C. V. Kavitha, B. S. Priya, S. L. Gaonkar, M. V. Tejesvi, K. S. Rangappa and S. Nanjunda Swamy

DOI: 10.2174/157018009789108222

New Pyrrole Hydrazones Synthesized and Evaluated In Vitro as Potential Tuberculostatics

, 6(7): 508 - 517

A. Bijev, S. Vladimirova and P. Prodanova

DOI: 10.2174/157018009789108268

Synthesis and Biochemical Evaluation of a Series of Methanesulfonate Derivatives of 4-Hydroxyphenyl Ketone as Probes of the Active Site of Type 3 OF 17β-Hydroxysteroid Dehydrogenase Family of Enzymes

, 6(7): 518 - 523

Kruti Shah, Moniola S. Olusanjo, Tim Cartledge, Caroline P. Owen and Sabbir Ahmed

DOI: 10.2174/157018009789108259

Synthesis and Biochemical Evaluation of a Range of 2-, 3- and 4-Substituted Derivatives of Benzyl Imidazole-Based Compounds as Probes of the Active Site of 17α-hydroxylase/17,20-Lyase (P45017α)

, 6(7): 524 - 530

Sabbir Ahmed, Imran Shahid, Kishore K. Bhatti, Wai-Yee Lee and Caroline P. Owen

DOI: 10.2174/157018009789108295

On the Synthesis and Anticancer Testing of α,β-Unsaturated Ketones as Analogs of Combretastatin-A4

, 6(7): 531 - 537

Sameer Chavda, Ryan Davis, Amanda Ferguson, Camille Riddering, Kristin Dittenhafer, Hilary Mackay, Balaji Babu, Moses Lee, Adam Siegfried, William Pennington, Miriam Shadfan, Susan L. Mooberry, Bijay K. Mishra and Hari N. Pati

DOI: 10.2174/157018009789108277

Design, Synthesis, Crystal Structure and Antitumor Activity of A New Ethyl 3-(quinazolin-4-ylamino)-1H-pyrrole-2-carboxylate Derivative

, 6(7): 538 - 541

Youguang Zheng, Xiaoqing Wu, Min Sun, Liuhai Feng, Mingdong Li and Min Ji

DOI: 10.2174/157018009789108240

Enhanced Brain Targeting of Tegafur Using Novel Lactyl Cholesterol Liposome as a Carrier

, 6(7): 542 - 547

Wei Fan, Xiankun Li, Shan Qian, Shan Wang and Yong Wu

DOI: 10.2174/157018009789108303

Synthesis, Anticonvulsant Evaluation of 2,3,4,5-Tetrahydro-7-alkoxy-1H-2-benzazepin-1-ones

, 6(7): 548 - 553

Cheng-Xi Wei, Wei Zhang, Zhe-Shan Quan, Rong-Bi Han, Ri-Shan Jiang and Feng-Yu Piao

DOI: 10.2174/157018009789108231

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