Contents

Letters in Drug Design & Discovery, Volume 6 - Number 2

Structure-Based Drug Design of Peptide Mimetics Containing Large P3 Moieties as Inhibitors of Factor VIIa

, 6(2): 86 - 92

Takuya Shiraishi, Shojiro Kadono, Masayuki Haramura, Hirofumi Kodama, Yoshiyuki Ono, Hitoshi Iikura, Tohru Esaki, Takaki Koga, Kunihiro Hattori, Yoshiaki Watanabe, Akihisa Sakamoto, Kazutaka Yoshihashi, Takehisa Kitazawa, Keiko Esaki, Masateru Ohta, Haruhiko Sato and Toshiro Kozono


DOI: 10.2174/157018009787582606




Prediction of Binding Affinities for Hydroxamic Acid Derivatives as Urease Inhibitors by Molecular Docking and 3D-QSAR Studies

, 6(2): 93 - 100

Zaheer-ul-Haq and Abdul Wadood


DOI: 10.2174/157018009787582598




Novel N-Substituted Thiazolidinones as Proton Pump Inhibitors and Potent Anti-Ulcer Agents: SAR Study

, 6(2): 101 - 106

S. Chandrappa, K. Vinaya, B. M. Srikanta, C.S. Ananda Kumar, N. R. Thimmegowda, S. R. Ranganatha, Shylaja M. Dharmesh and K. S. Rangappa


DOI: 10.2174/157018009787582697




Synthesis of Substituted 1H-Pyrrol-2(5H)-ones and 2(5H)-Furanones as Inhibitors of P. aeruginosa Biofilm

, 6(2): 107 - 113

Jia-Liang Guo, Bing-Zhou Li, Wei-Min Chen, Ping-Hua Sun and Yuqiang Wang


DOI: 10.2174/157018009787582642




Investigation of the Structural Requirement for Blocking the Human CCR5 Chemokine Receptor. An Insight from Quantitative Structure Activity Relationships Study

, 6(2): 114 - 124

Nigus Dessalew


DOI: 10.2174/157018009787582615




Physical Stability of PLGA Microparticles for DNA Encapsulation

, 6(2): 125 - 128

Itziar Migueliz, Sonsoles Diez, Gemma Navarro and Conchita Tros de ILarduya


DOI: 10.2174/157018009787582679




A Novel Synthesis Method of Apogossypolone and its Antitumor Activity

, 6(2): 129 - 132

Yonghua Zhan and Guangfeng Jia


DOI: 10.2174/157018009787582589




Synthesis and Antiproliferative Activity of Coumarin-Estrogen Conjugates against Breast Cancer Cell Lines

, 6(2): 133 - 138

Musiliyu A. Musa, M. Omar F. Khan and John S. Cooperwood


DOI: 10.2174/157018009787582624




Presentation of the β -Carboxamidophosphonate Arrangement in Substrate Structures Targeting HIV-1 PR

, 6(2): 139 - 145

N. J. Wardle, H. R. Hudson, R. W. Matthews, C. Nunn, C. Vella and S.W. A. Bligh


DOI: 10.2174/157018009787582660




Synthesis and In Vitro Antimicrobial Activity of Medicinally Important Novel N-alkyl, N-aryl and Urea Derivatives of 1-benzhydryl Piperizine: A Structure-Activity Relationship Study

, 6(2): 146 - 154

Channapillekoppal Siddegowda Ananda Kumar, Karunakara Murthy, Marlinganadoddi Panchegowda Sadashiva, Mallappanahally Kambappa Vinaya, Naraganahalli Ramegowda Thimmegowda, Salekoppal Boregowda Benaka Prasad, Siddappa Chandrappa and Kanchugarakoppal Subbegowda Rangappa


DOI: 10.2174/157018009787582570




Complex of Nifedipine with Glycyrrhizic Acid as a Novel Water-Soluble Antihypertensive and Antiarrhythmic Agent

, 6(2): 155 - 158

T. G. Tolstikova, M. V. Khvostov, A. O. Bryzgalov, A. V. Dushkin and E. S. Meteleva


DOI: 10.2174/157018009787582688




α 2-Adrenoceptor Antagonist SL84.0418 Involvement in the Development of Opioid Withdrawal

, 6(2): 159 - 162

Anna Capasso and Chiara Gallo


DOI: 10.2174/157018009787582651




3-Aminosterol Compounds as a New Class of Anti-Malarial Agents against Chloroquine-Susceptible and -Resistant Plasmodium falciparum

, 6(2): 163 - 166

Chanaz Salmi, Celine Loncle, Nicolas Vidal, Christophe Rogier, Yves Letourneux, Bruno Pradines and Jean Michel Brunel


DOI: 10.2174/157018009787582633




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