Letters in Drug Design & Discovery, Volume 6 - Number 1

Synthesis of 4-substituted-3-hydroxy-5-oxo-10-oxa-4-azatricyclo[5.2.1]dec- 3-yl Acetic Acid Ethyl Esters as Norcantharidin Analogues

, 6(1): 1 - 7

Benjamin Sauer, Jayne Gilbert, Jennette A. Sakoff and Adam McCluskey

DOI: 10.2174/157018009787158535

Involvement of Serotonin in the Acute Dependence Produced by μ, and K Opioid Agonists

, 6(1): 8 - 12

Anna Capasso

DOI: 10.2174/157018009787158562

Buprenorphine and Methadone Maintenance Treatment - Sexual Behaviour and Dysfunction Prevalence

, 6(1): 13

S. M. Giacomuzzi, A. Khreis, Y. Riemer, K. Garber and M. Ertl

DOI: 10.2174/157018009787158580

Computer-Aided Drug Design for Cancer-Causing H-Ras p21 Mutant Protein

, 6(1): 14 - 20

Mannu Jayakanthan, Gulshan Wadhwa, Thangavel Madhan Mohan, Loganathan Arul, Ponnusamy Balasubramanian and Durai Sundar

DOI: 10.2174/157018009787158526

Synthesis, Antibacterial Activity of 2,4-Disubstituted Oxazoles and Thiazoles as Bioisosteres

, 6(1): 21 - 28

Mohamed Kaspady, Venugopala Katharigatta Narayanaswamy, Mohana Raju and Gopal Krishna Rao

DOI: 10.2174/157018009787158481

Identification of GCP II Inhibitors Based on 4-Arylmethyl-3-(4- carboxyphenyl)-5-hydroxyisoxazole Scaffold

, 6(1): 29 - 32

M. Teus, A. Jirgensons, M. Dambrova, R. Mezhapuke, C. G. Parsons and W. Danysz

DOI: 10.2174/157018009787158544

Structural and Morphological Studies of Cationic Liposomes-DNA Complexes

, 6(1): 33 - 37

Yan Sun, Itziar Migueliz, Gemma Navarro and Conchita Tros de Ilarduya

DOI: 10.2174/157018009787158571

Pharmacophore Searching of Benzofuran Derivatives for Selective CYP19 Aromatase Inhibition

, 6(1): 38 - 45

Shuchi Nagar, Md Ataul Islam, Suvadra Das, Arup Mukherjee and Achintya Saha

DOI: 10.2174/157018009787158607

Evaluation of In-Vivo Anti-Implantation and In-Vitro Anti-Proliferative Activities of Substituted 3-phenyl-4-phenylvinyl Benzopyranone Derivatives

, 6(1): 46 - 50

Atul Gupta, Ramesh Sharma, Anil Kumar Balapure, Govind Keshri, M. M. Singh and Suprabhat Ray

DOI: 10.2174/157018009787158508

Synthesis and Antitumor Activity of Novel 4-Chloro-3-Arylmaleimide Derivatives

, 6(1): 51 - 55

Guiqing Xu, Qiaojun He, Bo Yang and Yongzhou Hu

DOI: 10.2174/157018009787158490

DNA Binders: 1. Evaluation of DNA-Interactive Ability, Design, and Synthesis of Novel Intercalating Agents

, 6(1): 56 - 62

Mario Sechi, Marco Derudas, Roberto Dallocchio, Alessandro Dessì, Alessia Cosseddu and Giuseppe Paglietti

DOI: 10.2174/157018009787158472

Susceptibility of Staphylococcus spp. Isolated from Milk of Goats with Mastitis to Antibiotics and Green Propolis Extracts

, 6(1): 63 - 68

T. M. Santos Neto, R. A. Mota, L. B.G. Silva, D. A. Viana, J. L. Lima-Filho, L. A. Sarubbo, A. Converti and A. L.F. Porto

DOI: 10.2174/157018009787158599

Synthesis and Antibacterial and Antifungal Activity of 5-Substituted Imidazolones

, 6(1): 69 - 77

Khalid Mohammed Khan, Uzma Rasool Mughal, Sadia Khan, Saira Khan, Shahnaz Perveen and M. Iqbal Choudhary

DOI: 10.2174/157018009787158553

Solution-Phase Parallel Synthesis of N-Arylisoquinuclidines

, 6(1): 78 - 81

Ronald F. Borne, Mark S. Levi, M. O. Faruk Khan and Norman H. Wilson

DOI: 10.2174/157018009787158517

Development of an Economical, Single Step Synthesis of FAZA, a Clinical Hypoxia Marker, and Potential Synthons to Prepare its Positional Analogs

, 6(1): 82 - 85

P. Kumar, S. Emami, A. J.B. McEwan and L. I. Wiebe

DOI: 10.2174/157018009787158616

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