Contents

Letters in Drug Design & Discovery, Volume 5 - Number 1

Evaluation of the Ability of an Organic Derivative of Ruthenium(II) to Reinforce the Cytotoxicity of Fast Neutron Against Malignant Cells in Culture

, 5(1): 1 - 6

P. Bischoff, L. Leyva, F. Malek, S. Benzina, J. M. Denis, J. Gueulette, P. Dufour, C. Gaiddon, J. P. Loeffler, C. Sirlin and M. Pfeffer


DOI: 10.2174/157018008783406714




CoMFA Study, Syntheses, Antitubercular and Anticancer Activity of Some Novel 1,4-Dihydropyridines

, 5(1): 7 - 14

B.R. Prashantha Kumar, S. Yuvaraj, Anil Srivastava, Vanitha Chaturvedi, Y. K. Manju, B. Suresh and M. J. Nanjan


DOI: 10.2174/157018008783406688




Synthesis, In Vitro Evaluations and Structure-Activity Assessment of Pyrrole Hydrazones as Potential Tuberculostatics

, 5(1): 15 - 24

A. Bijev


DOI: 10.2174/157018008783406651




Synthesis and Evaluation of N-Aryl 2-Aminothiazole-4-Carboxamide Derivatives for Activity Against TB

, 5(1): 25 - 28

R. M. Riggs, R. K. Jennings, E. R. Derstine, T. M. Nguyen, T. Trinh and J. M. Riordan


DOI: 10.2174/157018008783406615




Immunomodulation and Anti-Inflammatory Effects of Macrolides: Old Drugs with Fascinating New Perspectives

, 5(1): 29 - 35

I. Starakis


DOI: 10.2174/157018008783406642




Selective Inhibition of Neuronal Nitric Oxide Synthase by L-Arginine Derivatives

, 5(1): 36 - 38

Anna Capasso, Carmela Saturnino and Mariafrancesca Buonerba


DOI: 10.2174/157018008783406660




Design and Synthesis of 2-Azetidinone Cholesterol Absorption Inhibitors

, 5(1): 39 - 42

Huibin Zhang, Yubin Wang, Rui Zhao, Wenlong Huang, Yunman Li and Jinpei Zhou


DOI: 10.2174/157018008783406741




Solution Phase Synthesis of a 3,5,7-Substituted Indolin-2-one Library as Potential CDK2 Inhibitor Isosteres

, 5(1): 43 - 47

Dmytro O. Tymoshenko, Brian T. Gregg, Matthew J. Hirsch and Jennifer L. Butcher


DOI: 10.2174/157018008783406633




Inhibition of 17β -Hydroxysteroid Dehydrogenase (17β -HSD) by Imidazole-Based Compounds

, 5(1): 48 - 51

Sabbir Ahmed, Moniola S. Olusanjo, Imran Shahid and Caroline P. Owen


DOI: 10.2174/157018008783406705




Synthesis and Chymotrypsin Inhibitory Activity of Substituted Oxazolones

, 5(1): 52 - 56

Khalid Mohammed Khan, Uzma Rasool Mughal, Muhammad Arif Lodhi and Muhammad Iqbal Choudhary


DOI: 10.2174/157018008783406624




Classical and Fragment-Based Hologram Structure-Activity Relationships for a Series of Analgesic Cyclic Imides

, 5(1): 57 - 64

A. D. Andricopulo, D. M. Borchhardt and M. S. Castilho


DOI: 10.2174/157018008783406723




Central Administration of L-Ser-L-His and L-Ile-L-His Induced Sedative Effects Under an Acute Stressful Condition in Chicks

, 5(1): 65 - 68

Mitsuhiro Furuse, Yousuke Tsuneyoshi, Shozo Tomonaga, Haruka Yamane, Koji Morishita and D. Michael Denbow


DOI: 10.2174/157018008783406679




Flavylium Salts as Precursors of Biologically Active Chalcones

, 5(1): 69 - 73

Karl A. Werbovetz, Tesmol G. George, Julian Richard, Todd Barszcz and Jeffrey Capers


DOI: 10.2174/157018008783406697




Antifungal Activity of Goniothalamin Enantiomers

, 5(1): 74 - 78

Angelo de Fatima, Cleide Viviane Buzanello Martins, Maria Aparecida de Resende, Thais Furtado Ferreira Magalhaes, Bruno Henrique Santiago Lima, Gisele Almeida Watanabe, Ana Lucia Tasca Gois Ruiz, Joao Ernesto de Carvalho and Ronaldo Aloise Pilli


DOI: 10.2174/157018008783406732




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