Letters in Drug Design & Discovery, Volume 5 - Number 1

Evaluation of the Ability of an Organic Derivative of Ruthenium(II) to Reinforce the Cytotoxicity of Fast Neutron Against Malignant Cells in Culture

, 5(1): 1 - 6

P. Bischoff, L. Leyva, F. Malek, S. Benzina, J. M. Denis, J. Gueulette, P. Dufour, C. Gaiddon, J. P. Loeffler, C. Sirlin and M. Pfeffer

DOI: 10.2174/157018008783406714

CoMFA Study, Syntheses, Antitubercular and Anticancer Activity of Some Novel 1,4-Dihydropyridines

, 5(1): 7 - 14

B.R. Prashantha Kumar, S. Yuvaraj, Anil Srivastava, Vanitha Chaturvedi, Y. K. Manju, B. Suresh and M. J. Nanjan

DOI: 10.2174/157018008783406688

Synthesis, In Vitro Evaluations and Structure-Activity Assessment of Pyrrole Hydrazones as Potential Tuberculostatics

, 5(1): 15 - 24

A. Bijev

DOI: 10.2174/157018008783406651

Synthesis and Evaluation of N-Aryl 2-Aminothiazole-4-Carboxamide Derivatives for Activity Against TB

, 5(1): 25 - 28

R. M. Riggs, R. K. Jennings, E. R. Derstine, T. M. Nguyen, T. Trinh and J. M. Riordan

DOI: 10.2174/157018008783406615

Immunomodulation and Anti-Inflammatory Effects of Macrolides: Old Drugs with Fascinating New Perspectives

, 5(1): 29 - 35

I. Starakis

DOI: 10.2174/157018008783406642

Selective Inhibition of Neuronal Nitric Oxide Synthase by L-Arginine Derivatives

, 5(1): 36 - 38

Anna Capasso, Carmela Saturnino and Mariafrancesca Buonerba

DOI: 10.2174/157018008783406660

Design and Synthesis of 2-Azetidinone Cholesterol Absorption Inhibitors

, 5(1): 39 - 42

Huibin Zhang, Yubin Wang, Rui Zhao, Wenlong Huang, Yunman Li and Jinpei Zhou

DOI: 10.2174/157018008783406741

Solution Phase Synthesis of a 3,5,7-Substituted Indolin-2-one Library as Potential CDK2 Inhibitor Isosteres

, 5(1): 43 - 47

Dmytro O. Tymoshenko, Brian T. Gregg, Matthew J. Hirsch and Jennifer L. Butcher

DOI: 10.2174/157018008783406633

Inhibition of 17β -Hydroxysteroid Dehydrogenase (17β -HSD) by Imidazole-Based Compounds

, 5(1): 48 - 51

Sabbir Ahmed, Moniola S. Olusanjo, Imran Shahid and Caroline P. Owen

DOI: 10.2174/157018008783406705

Synthesis and Chymotrypsin Inhibitory Activity of Substituted Oxazolones

, 5(1): 52 - 56

Khalid Mohammed Khan, Uzma Rasool Mughal, Muhammad Arif Lodhi and Muhammad Iqbal Choudhary

DOI: 10.2174/157018008783406624

Classical and Fragment-Based Hologram Structure-Activity Relationships for a Series of Analgesic Cyclic Imides

, 5(1): 57 - 64

A. D. Andricopulo, D. M. Borchhardt and M. S. Castilho

DOI: 10.2174/157018008783406723

Central Administration of L-Ser-L-His and L-Ile-L-His Induced Sedative Effects Under an Acute Stressful Condition in Chicks

, 5(1): 65 - 68

Mitsuhiro Furuse, Yousuke Tsuneyoshi, Shozo Tomonaga, Haruka Yamane, Koji Morishita and D. Michael Denbow

DOI: 10.2174/157018008783406679

Flavylium Salts as Precursors of Biologically Active Chalcones

, 5(1): 69 - 73

Karl A. Werbovetz, Tesmol G. George, Julian Richard, Todd Barszcz and Jeffrey Capers

DOI: 10.2174/157018008783406697

Antifungal Activity of Goniothalamin Enantiomers

, 5(1): 74 - 78

Angelo de Fatima, Cleide Viviane Buzanello Martins, Maria Aparecida de Resende, Thais Furtado Ferreira Magalhaes, Bruno Henrique Santiago Lima, Gisele Almeida Watanabe, Ana Lucia Tasca Gois Ruiz, Joao Ernesto de Carvalho and Ronaldo Aloise Pilli

DOI: 10.2174/157018008783406732

Webmaster Contact:
Copyright © 2018 Bentham Science