Contents

Letters in Drug Design & Discovery, Volume 4 - Number 7

Effect of the Metal Center on the Antitumor Activity of the Analogous Dinuclear Spermine Chelates (PdCl2)2(Spermine) and (PtCl2)2(Spermine)

, 4(7): 460 - 463

Ana S. Soares, Sonia M. Fiuza, M. Joao Goncalves, Luis A.E. Batista de Carvalho, M. Paula M. Marques and Ana M. Urbano


DOI: 10.2174/157018007781788516




Microwave-Assisted Synthesis of Substituted 2,4-Diarylthiazoles and their Evaluation as Anticancer Agents

, 4(7): 464 - 466

Romeo Romagnoli, Pier Giovanni Baraldi, Olga Cruz Lopez, Maria Dora Carrion, Carlota Lopez Cara, Delia Preti, Mojgan Aghazadeh Tabrizi and Jan Balzarini


DOI: 10.2174/157018007781788507




In Vitro Cytotoxicity Evaluation of Some Substituted Indazole Derivatives

, 4(7): 467 - 470

El Mostapha Rakib, Bassou Oulemda, Said Abouricha, Latifa Bouissane, Hassan Ait Mouse and Abdelmajid Zyad


DOI: 10.2174/157018007781788589




Synthesis and Anti-HIV Activity of Bi-Functional Triterpene Derivatives

, 4(7): 471 - 478

Li Huang, Donglei Yu, Phong Ho, Kuo-Hsiung Lee and Chin-Ho Chen


DOI: 10.2174/157018007781788561




Synthesis, Biochemical Evaluation and Rationalisation of the Inhibitory Activity of a Series of 4-Substituted Phenyl Alkyl Triazole-Based Compounds as Potential Inhibitors of 17α-Hydroxylase/17,20-Lyase (P45017α)

, 4(7): 479 - 483

Caroline P. Owen, Sachin Dhanani, Chirag H. Patel and Sabbir Ahmed


DOI: 10.2174/157018007781788471




Synthesis and Biological Activity of a New Class of Azetidinones Compounds as Potential HLE Inhibitors

, 4(7): 484 - 486

Carmela Saturnino, Mariafrancesca Buonerba and Anna Capasso


DOI: 10.2174/157018007781788543




Caveats Regarding the Use of IL-10 and IL-10 Antagonist as Immunotherapeutic Factors

, 4(7): 487 - 495

Jesus Colino


DOI: 10.2174/157018007781788552




A Quantitative Structure-Activity Relationship Study on Some Aryl Sulfonyl Amido and Ureido Derivatives Acting as Matrix Metalloproteinase and Clostridium histolyticum Collagenase Inhibitors

, 4(7): 496 - 501

Satya P. Gupta, Priyanka Bagaria and Venkata Satya Ashok Kumar Satuluri


DOI: 10.2174/157018007781788598




In Silico Prediction of Human Plasma Protein Binding Using Hologram QSAR

, 4(7): 502 - 509

Tiago L. Moda, Carlos A. Montanari and Adriano D. Andricopulo


DOI: 10.2174/157018007781788480




Twelve Different HI-6 Salts and their Potency to Reactivate Cyclosarin Inhibited AChE In Vitro

, 4(7): 510 - 512

Kamil Kuca, Kamil Musilek, Petr Stodulka, Jan Marek, Petra Hanusova, Daniel Jun, Martina Hrabinova, Jiri Kassa and Bohuslav Dolezal


DOI: 10.2174/157018007781788462




Antibacterial Activity of 3-Substituted Pyrrole-2,5-diones Against Pseudomonas Aeruginosa

, 4(7): 513 - 519

Eric Lattmann, Simon Dunn, Suwanna Niamsanit, Jintana Sattayasai and Nison Sattayasai


DOI: 10.2174/157018007781788570




First In Vivo Evaluation of a New Morpholine Analog

, 4(7): 520 - 523

M. Altamura, A. Guidi, F. Pasqui, M. Tramontana and K. Worm-Leonhard


DOI: 10.2174/157018007781788534




Artemisinin Delays Sphingolipid Biosynthesis in Plasmodium falciparum

, 4(7): 524 - 526

Francoise Debierre-Grockiego, Jorg Schmidt, Eliezer Flescher and Ralph T. Schwarz


DOI: 10.2174/157018007781788499




The Derivation of a Potential Transition-State for the Reduction Reaction Catalysed by 17β -Hydroxysteroid Dehydrogenase Type 3 (17β -HSD) - An Approximate Representation of its Active Site for Use in Drug Design and Discovery

, 4(7): 527 - 531

Moniola S. Olusanjo and Sabbir Ahmed


DOI: 10.2174/157018007781788525




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