Contents

Letters in Drug Design & Discovery, Volume 4 - Number 6

Inhibition of Human Leucocyte Elastase by Novel Thieno-1,3-oxazin-4-ones and Thieno-1,3-thioxazin-4-ones

, 4(6): 386 - 393

N.A. Santagati, L. Salerno, C. Di Giacomo, L. Vanella and S. Ronsisvalle


DOI: 10.2174/157018007781387764




Synthesis and In Vitro Biochemical Evaluation of a Series of Compounds as Potential Inhibitors of Estrone Sulfatase (ES) and the Role of pKa in both the Synthesis and the Inhibitory Activity of the Potential Inhibitors

, 4(6): 394 - 398

Caroline P. Owen, Mijal Patel, Chirag K Patel, Tim Cartledge and Sabbir Ahmed


DOI: 10.2174/157018007781387773




Synthesis and In Vitro Biochemical Evaluation of a Series of Cycloalkyl Esters of 4-Sulfamoylated Benzoic Acid as Inhibitors of Estrone Sulfatase (ES)

, 4(6): 399 - 403

Caroline P. Owen, Chirag K. Patel, Tim Cartledge and Sabbir Ahmed


DOI: 10.2174/157018007781387845




Synthesis and Anti-HSV-1 Activity of 1,4-dihydro-4-oxoquinoline Ribonucleosides

, 4(6): 404 - 409

Carla Veronica B. dos S. Canuto, Claudia R. B. Gomes, Isakelly P. Marques, Leticia V. Faro, Fernanda da Costa Santos, Izabel Christina de P. P. Frugulhetti, Thiago M. L. e Souza, Anna C.Cunha, Gilberto A. Romeiro, Vitor F. Ferreira and Maria Cecilia B.V.de Souza


DOI: 10.2174/157018007781387818




Classification and Prediction of Tripeptides Inhibiting HIV-1 Tat/TAR-RNA Interaction Using a Self-Organizing Map

, 4(6): 410 - 416

A. Givehchi, V. Ludwig, O. Boden, A. Krebs, U. Scheffer, M. Gobel and G. Schneider


DOI: 10.2174/157018007781387791




Structure-Based Quantitative Structure Activity Relationship Analysis of Omuralide Analogs in the 20S Proteasome: A Covalent Inhibitor COMBINE Study

, 4(6): 417 - 421

Jenna L. Wang, Apurba Datta and Gerald H. Lushington


DOI: 10.2174/157018007781387809




The Molecular Basis of COX-2 Versus COX-1 Selectivity of Lumiracoxib by Molecular Docking Studies

, 4(6): 422 - 425

Celia M. Correa, Andre F. de Paula, Gilberto M.S. da Silva, Carlos M.R. Sant'Anna, Carlos A. M. Fraga and Eliezer J. Barreiro


DOI: 10.2174/157018007781387737




A Cationic Liposomal Vincristine Formulation with Improved Vincristine Retention, Extended Circulation Lifetime and Increased Anti-Tumor Activity

, 4(6): 426 - 433

Murray S. Webb, Nancy L. Boman, Dana Masin, Donald Yapp, Euan Ramsay, Gigi N.C. Chiu, Pieter R. Cullis and Marcel B. Bally


DOI: 10.2174/157018007781387782




Isoform-Selective Regulation of Adenylyl Cyclase by Forskolin Derivatives:Prediction of Selectivity by Computer-Based Analysis

, 4(6): 434 - 441

Haruki Eguchi, Kousaku Iwatsubo and Yoshihiro Ishikawa


DOI: 10.2174/157018007781387755




Preparation and Biological Activities of Heteroarotinoids

, 4(6): 442 - 445

Akimori Wada, Yukari Mizuguchi, Hiromi Miyake, Miki Niihara, Masayoshi Ito, Kimie Nakagawa and Toshio Okano


DOI: 10.2174/157018007781387827




Lamotrigine as an Effective Treatment for Behavioral Disorders

, 4(6): 446 - 452

Rita Moretti, Paola Torre, Cristina Vilotti and Rodolfo M. Antonello


DOI: 10.2174/157018007781387836




Release Kinetics of Ampicillin, Biocompatibility Tests with a Fibroblast Strain of a Zirconia Gel Glass

, 4(6): 453 - 459

M. Catauro, M.G. Raucci and M.A. Continenza


DOI: 10.2174/157018007781387746




Webmaster Contact: info@benthamscience.org
Copyright © 2018 Bentham Science