Contents

Letters in Drug Design & Discovery, Volume 4 - Number 4

Inhibitory Effect of Acetogenins on Mammalian DNA Polymerase and Human Cancer Cell Growth

, 4(4): 239 - 245

Chisato Ishimaru, Toshifumi Takeuchi, Yuko Yonezawa, Isoko Kuriyama, Msasaharu Takemura, Ikuo Kato, Fumio Sugawara, Hiromi Yoshida and Yoshiyuki Mizushina


DOI: 10.2174/157018007784619961




Synthesis and Evaluation of 2-Substituted Fendiline Analogues as Antileukemics

, 4(4): 246 - 248

James A. Wilkinson, Steven B. Rossington, Nicholas A. Coe, Nicholas Hirst, Alan T. McGown, John Leonard and Nigel Hussain


DOI: 10.2174/157018007784620068




Synthesis and Antitumor Properties of N1-(Hydroxymethyl Phenylmethyl) Pyrimidine Derivatives and their Intermediates

, 4(4): 249 - 256

Liying Chen, Nageswara Kode, Devangachinta Murthy and Shashikant Phadtare


DOI: 10.2174/157018007784620022




Copper Complexes of Henna-Sulforaphane Conjugates as Potent Antiproliferative Agents Against Human Myeloma KBM-5 Cells Through Blockade of Transcription Factor NF-κB

, 4(4): 257 - 262

K. Shirisha, J. Patole, S. Padhye, E. Sinn, S. Shishodia and B. B. Aggarwal


DOI: 10.2174/157018007784620059




Novel, Acidic CCR2 Receptor Antagonists: Lead Optimization

, 4(4): 263 - 271

O. A. Dasse, J. L. Evans, H.-X. Zhai, D. Zou, J. T. Kintigh, F. Chan, K. Hamilton, E. Hill, J. B. Eckman, P. J. Higgins, A. Volosov, P. Collart, J.-M. Nicolas, R.K. Kondru and C.E. Schwartz


DOI: 10.2174/157018007784619989




An Alternative Method for the Synthesis of Tetraketones and their Lipoxygenase Inhibiting and Antioxidant Properties

, 4(4): 272 - 278

Khalid Mohammed Khan, Ghulam Murtaza Maharvi, Sarfraz Ahmed Nawaz, Shahnaz Perveen and Muhammad Iqbal Choudhary


DOI: 10.2174/157018007784620004




Synthesis of 18F-labeled Neurotensin(8-13) via Copper-Mediated 1,3-Dipolar [3+2]Cycloaddition Reaction

, 4(4): 279 - 285

Theres Ramenda, Ralf Bergmann and Frank Wuest


DOI: 10.2174/157018007784619998




A Novel Descriptor Histogram Filtering Method for Database Mining and the Identification of Active Molecules

, 4(4): 286 - 292

Yuan Wang, Jeffrey W. Godden and Jurgen Bajorath


DOI: 10.2174/157018007784619970




Target-Oriented Synthesis of Antiparasitic 2-Hetaryl Substituted Quinolines Based on Imino Diels-Alder Reactions

, 4(4): 293 - 296

Vladimir V. Kouznetsov, Leonor Y. Vargas Mendez, Sandra Milena Leal, Uriel Mora Cruz, Carlos Andres Coronado, Carlos M. Melendez Gomez, Arnold R. Romero Bohorquez and Patricia Escobar Rivero


DOI: 10.2174/157018007784620031




In vitro Antimicrobial Activity of Liposomes Containing Ciprofloxacin,Meropenem and Gentamicin Against Gram-Negative Clinical Bacterial Strains

, 4(4): 297 - 304

Jerzy Gubernator, Zuzanna Drulis-Kawa, Agata Dorotkiewicz-Jach, Wlodzimierz Doroszkiewicz and Arkadiusz Kozubek


DOI: 10.2174/157018007784620040




Effect of Fluoxetine on Brain Oxidative Stress, Neuronal Damage and Behavioural Induced in the Olfactory Bulbectomy Model of Depression

, 4(4): 305 - 310

Isaac Tunez, Francisco J. Medina, Ignacio Jimena and María del C. Munoz


DOI: 10.2174/157018007784620013




Webmaster Contact: info@benthamscience.org
Copyright © 2018 Bentham Science