Contents

Letters in Drug Design & Discovery, Volume 3 - Number 6

Targeting the Epidermal Growth Factor Receptor Family in Radionuclide Therapy of Tumors – Signal Transduction and DNA Repair

, 3(6): 357 - 368

Johan Lennartsson, Jorgen Carlsson and Bo Stenerlow


DOI: 10.2174/157018006777805503




MDR Reversal by Deprenylated Tetracyclic and Hexacyclic Analogues of N-Acetylardeemin: Confirmation of the Ardeemin Pharmacophore

, 3(6): 369 - 377

Carmen Avendano, Esmeralda Caballero, Cristina Mendez-Vidal, Ana R. de Quesada and J. Carlos Menendez


DOI: 10.2174/157018006777805558




Coenzyme Q10 and Neurological Diseases: An Update

, 3(6): 378 - 382

Michelangelo Mancuso, Anna Choub, Massimiliano Filosto, Lucia Petrozzi, Gianfranco Cafforio, Gabriele Siciliano and Luigi Murri


DOI: 10.2174/157018006777805495




Lead Optimisation: Improving the Affinity of the Antiretrovirals Nelfinavir and Amprenavir for HIV-1 Protease

, 3(6): 383 - 389

P. A. Fernandes, M.L. A.C. Araujo, A. J.M. Barbosa, C. N. Alves, Z. Q. Ferreira, C. R.-N. Gonzalez, C.F. R.A. C. Lima, S. I.E. Loureiro, J. M.T. Magalhaes, F. C. Maia, S. A. Moura, E.M. M. Peredo, M.A. S. Perez, T.A. Q. Rodrigues, A.M. Pessoa, C.A. M. da Silva, J.P. A. da Silva and M. J. Ramos


DOI: 10.2174/157018006777805576




Utilization of Ribozymes as Antiviral Agents

, 3(6): 390 - 404

M. L. Benitez-Hess and L. M. Alvarez-Salas


DOI: 10.2174/157018006777805521




Non-Classical Drug Metabolism Enzymes: The Curious Case of Phenylalanine 4-Monooxygenase

, 3(6): 405 - 412

G. B. Steventon and S. C. Mitchell


DOI: 10.2174/157018006777805512




High-Throughput Lipophilicity Screening of Opioid-Like Analgesics: Validation of Computational Methods by Means of RP-HPLC Analysis

, 3(6): 413 - 418

O. Azzolina, S. Collina, D. Rossi, A. Carnevale Baraglia, S. Alcaro and A. Artese


DOI: 10.2174/157018006777805530




Antitubercular Properties of Substituted Hydroxycyclohexadienones

, 3(6): 419 - 423

Manish Shah, Geoffrey Wells, Tracey D. Bradshaw, Charles A. Laughton, Malcolm F.G. Stevens and Andrew D. Westwell


DOI: 10.2174/157018006777805486




Synthesis and In Vitro Anti-Tubercular Activity of a Series of N- (Disubstitutedbenzoyl)Isoniazid Derivatives

, 3(6): 424 - 428

Ivan Neves Junior, Maria C.S. Lourenco, Guilherme de B.P. de Miranda, Thatyana R.A. Vasconcelos, Karla C. Pais, Jose dos P. de A. Junior, M. S.V. Wardell, James L. Wardell and V. N. de Souza


DOI: 10.2174/157018006777805549




Replacement of Cyclosporin A from its Binding to Hepatocyte Plasma Membrane by Silymarin Flavonoids

, 3(6): 429 - 435

Vladimira Moulisova, Jiri Sebestian, Olga Jedlickova, Alexandr Jegorov and Stepanka B. Sebestianova


DOI: 10.2174/157018006777805567




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