Letters in Drug Design & Discovery, Volume 3 - Number 5

Quality Initiatives in Drug Discovery: Swim Dont Sink

, 3(5): 286 - 288

S. G. Volsen, M. G. Parry and M. Masson

DOI: 10.2174/157018006777574195

Design and Discovery of Novel, Potent Pyrazinone-Based Thrombin Inhibitors with a Solubilizing Amino P1-P2-Linker

, 3(5): 289 - 292

S. Bulat, S. Bosio, M. A. Papadopoulos, S. Cerezo-Galvez, E. Grabowski, C. Rosenbaum, V. G. Matassa, I. Ott, G. Metz, J. Schamberger, R. Sekul and A. Feurer

DOI: 10.2174/157018006777574203

Target Structure-based Modeling of the Glutamate Transporter Pharmacophore

, 3(5): 293 - 297

A. Simon, A. Bencsura and J. Kardos

DOI: 10.2174/157018006777574230

Novel Benzimidazole Derivatives as Selective CB2 Inverse Agonists

, 3(5): 298 - 303

D. Page, M.-C. Brochu, H. Yang, W. Brown, S. St-Onge, E. Martin and D. Salois

DOI: 10.2174/157018006777574177

Design, Synthesis and Biological Evaluation of Novel Curcumin Analogues as Anti-Neoplastic Agents

, 3(5): 304 - 310

Amitabh Jha, Jin Zhao, T. Stanley Cameron, Erik De Clercq, Jan Balzarini, Elias K. Manavathu and James P. Stables

DOI: 10.2174/157018006777574131

Synthesis of Piperazinephen-1-ylethylamines as Potent and Selective Antagonists of the Human Melanocortin-4 Receptor

, 3(5): 311 - 315

Fabio C. Tucci, Joe A. Tran, Wanlong Jiang, Joseph Pontillo, Dragan Marinkovic, Nicole S. White, Melissa Arellano, Beth A. Fleck, Jenny Wen, John Saunders, Alan C. Foster and Chen Chen

DOI: 10.2174/157018006777574249

Cytotoxic and COX-2 Inhibition Properties of Hydroxycinnamic Derivatives

, 3(5): 316 - 320

M. Paula M. Marques, Fernanda Borges, Joana Sousa, Rita Calheiros, Jorge Garrido, Alexandra Gaspar, Carmen Diniz and Paula Fresco

DOI: 10.2174/157018006777574212

Lamotrigine Pharmacokinetics During Anticonception and Pregnancy

, 3(5): 321 - 322

A. Sabers

DOI: 10.2174/157018006777574267

The NK-1 Receptor is Involved in the Antitumoural Action of L-733,060 and in the Mitogenic Action of Substance P on Human Pancreatic Cancer Cell Lines

, 3(5): 323 - 329

Miguel Munoz, Marisa Rosso and Rafael Covenas

DOI: 10.2174/157018006777574168

Synthesis and Radiopharmacological Characterisation of 86Y- and 68Ga-Labelled L-RNA Oligonucleotides as Molecular Probes for Positron Emission Tomography (PET)

, 3(5): 330 - 335

Joern Schlesinger, Ralf Bergmann, Sven Klussmann and Frank Wuest

DOI: 10.2174/157018006777574221

Design, Synthesis and Initial In Vitro Evaluation of Novel Prodrugs for the Treatment of Cystinosis

, 3(5): 336 - 345

R. J. Anderson, D. Cairns, W. A. Cardwell, M. Case, P. W. Groundwater, A. G. Hall, L. Hogarth, A. L. Jones, O. Meth-Cohn and P. Suryadevara

DOI: 10.2174/157018006777574258

The Cardiovascular Properties of Some Amide Derivatives of Pyrimidin-8-on[2,1-f]theophylline-9- Alkylcarboxylic Acids

, 3(5): 346 - 350

A. Zagorska, O. Fhid, M. Pawlowski, B. Filipek and M. Zygmunt

DOI: 10.2174/157018006777574159

Homocysteine and Folate Therapy in Dialysis Patients

, 3(5): 351 - 355

Marco Righetti

DOI: 10.2174/157018006777574140


, 3(5): 356

DOI: 10.2174/157018006777574186

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