Contents

Letters in Drug Design & Discovery, Volume 3 - Number 5

Quality Initiatives in Drug Discovery: Swim Dont Sink

, 3(5): 286 - 288

S. G. Volsen, M. G. Parry and M. Masson


DOI: 10.2174/157018006777574195




Design and Discovery of Novel, Potent Pyrazinone-Based Thrombin Inhibitors with a Solubilizing Amino P1-P2-Linker

, 3(5): 289 - 292

S. Bulat, S. Bosio, M. A. Papadopoulos, S. Cerezo-Galvez, E. Grabowski, C. Rosenbaum, V. G. Matassa, I. Ott, G. Metz, J. Schamberger, R. Sekul and A. Feurer


DOI: 10.2174/157018006777574203




Target Structure-based Modeling of the Glutamate Transporter Pharmacophore

, 3(5): 293 - 297

A. Simon, A. Bencsura and J. Kardos


DOI: 10.2174/157018006777574230




Novel Benzimidazole Derivatives as Selective CB2 Inverse Agonists

, 3(5): 298 - 303

D. Page, M.-C. Brochu, H. Yang, W. Brown, S. St-Onge, E. Martin and D. Salois


DOI: 10.2174/157018006777574177




Design, Synthesis and Biological Evaluation of Novel Curcumin Analogues as Anti-Neoplastic Agents

, 3(5): 304 - 310

Amitabh Jha, Jin Zhao, T. Stanley Cameron, Erik De Clercq, Jan Balzarini, Elias K. Manavathu and James P. Stables


DOI: 10.2174/157018006777574131




Synthesis of Piperazinephen-1-ylethylamines as Potent and Selective Antagonists of the Human Melanocortin-4 Receptor

, 3(5): 311 - 315

Fabio C. Tucci, Joe A. Tran, Wanlong Jiang, Joseph Pontillo, Dragan Marinkovic, Nicole S. White, Melissa Arellano, Beth A. Fleck, Jenny Wen, John Saunders, Alan C. Foster and Chen Chen


DOI: 10.2174/157018006777574249




Cytotoxic and COX-2 Inhibition Properties of Hydroxycinnamic Derivatives

, 3(5): 316 - 320

M. Paula M. Marques, Fernanda Borges, Joana Sousa, Rita Calheiros, Jorge Garrido, Alexandra Gaspar, Carmen Diniz and Paula Fresco


DOI: 10.2174/157018006777574212




Lamotrigine Pharmacokinetics During Anticonception and Pregnancy

, 3(5): 321 - 322

A. Sabers


DOI: 10.2174/157018006777574267




The NK-1 Receptor is Involved in the Antitumoural Action of L-733,060 and in the Mitogenic Action of Substance P on Human Pancreatic Cancer Cell Lines

, 3(5): 323 - 329

Miguel Munoz, Marisa Rosso and Rafael Covenas


DOI: 10.2174/157018006777574168




Synthesis and Radiopharmacological Characterisation of 86Y- and 68Ga-Labelled L-RNA Oligonucleotides as Molecular Probes for Positron Emission Tomography (PET)

, 3(5): 330 - 335

Joern Schlesinger, Ralf Bergmann, Sven Klussmann and Frank Wuest


DOI: 10.2174/157018006777574221




Design, Synthesis and Initial In Vitro Evaluation of Novel Prodrugs for the Treatment of Cystinosis

, 3(5): 336 - 345

R. J. Anderson, D. Cairns, W. A. Cardwell, M. Case, P. W. Groundwater, A. G. Hall, L. Hogarth, A. L. Jones, O. Meth-Cohn and P. Suryadevara


DOI: 10.2174/157018006777574258




The Cardiovascular Properties of Some Amide Derivatives of Pyrimidin-8-on[2,1-f]theophylline-9- Alkylcarboxylic Acids

, 3(5): 346 - 350

A. Zagorska, O. Fhid, M. Pawlowski, B. Filipek and M. Zygmunt


DOI: 10.2174/157018006777574159




Homocysteine and Folate Therapy in Dialysis Patients

, 3(5): 351 - 355

Marco Righetti


DOI: 10.2174/157018006777574140




Erratum

, 3(5): 356


DOI: 10.2174/157018006777574186




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