Contents

Letters in Drug Design & Discovery, Volume 3 - Number 5


Design and Discovery of Novel, Potent Pyrazinone-Based Thrombin Inhibitors with a Solubilizing Amino P1-P2-Linker

, 3(5): 289 - 292

S. Bulat, S. Bosio, M. A. Papadopoulos, S. Cerezo-Galvez, E. Grabowski, C. Rosenbaum, V. G. Matassa, I. Ott, G. Metz, J. Schamberger, R. Sekul and A. Feurer


DOI: 10.2174/157018006777574203




Design, Synthesis and Biological Evaluation of Novel Curcumin Analogues as Anti-Neoplastic Agents

, 3(5): 304 - 310

Amitabh Jha, Jin Zhao, T. Stanley Cameron, Erik De Clercq, Jan Balzarini, Elias K. Manavathu and James P. Stables


DOI: 10.2174/157018006777574131


Synthesis of Piperazinephen-1-ylethylamines as Potent and Selective Antagonists of the Human Melanocortin-4 Receptor

, 3(5): 311 - 315

Fabio C. Tucci, Joe A. Tran, Wanlong Jiang, Joseph Pontillo, Dragan Marinkovic, Nicole S. White, Melissa Arellano, Beth A. Fleck, Jenny Wen, John Saunders, Alan C. Foster and Chen Chen


DOI: 10.2174/157018006777574249


Cytotoxic and COX-2 Inhibition Properties of Hydroxycinnamic Derivatives

, 3(5): 316 - 320

M. Paula M. Marques, Fernanda Borges, Joana Sousa, Rita Calheiros, Jorge Garrido, Alexandra Gaspar, Carmen Diniz and Paula Fresco


DOI: 10.2174/157018006777574212





Design, Synthesis and Initial In Vitro Evaluation of Novel Prodrugs for the Treatment of Cystinosis

, 3(5): 336 - 345

R. J. Anderson, D. Cairns, W. A. Cardwell, M. Case, P. W. Groundwater, A. G. Hall, L. Hogarth, A. L. Jones, O. Meth-Cohn and P. Suryadevara


DOI: 10.2174/157018006777574258






Webmaster Contact: info@benthamscience.org
Copyright © 2018 Bentham Science