Letters in Drug Design & Discovery, Volume 2 - Number 8

Rational Design of the New Antihypertensive I1-Receptor Ligand 2-(2- Biphenyl-2-yl-1-methyl-ethyl)-4,5-dihydro-1H-imidazole

, 2(8): 571 - 578

F. Gentili, P. Bousquet, A. Carrieri, J. Feldman, F. Ghelfi, M. Giannella, A. Piergentili, W. Quaglia, C. Vesprini and M. Pigini

DOI: 10.2174/157018005774717325

Docking Study, Synthesis and SAH-Hydrolase Inhibitory Activity of LAdeninylalanine and Related Analogues

, 2(8): 579 - 583

Nicolas Floquet, Samuel Leroy, Murielle Muzard, Georges Guillerm and Jean-Bernard Behr

DOI: 10.2174/157018005774717262

Anti-tumour Activity of Some Polydentate N-Ligands: N,N-bis-(3- Substituted-5-Methylpyrazol-1yl Methyl) Arylamines and N,N,N,N-Tetra- [(3-Substituted-5-Methylpyrazol-1yl] Para-Phenylenediamines

, 2(8): 584 - 589

T. B. Hadda, A. T. Kotchevar, M. Daoudi, B. Bennani, N. B. Larbi and A. Kerbal

DOI: 10.2174/157018005774717299

Discovery of Thrombin Inhibitor Fragments from Chemical Microarray Screening

, 2(8): 590 - 594

Thomas Neumann, Hans-Dieter Junker, Oliver Keil, Klaus Burkert, Holger Ottleben, Jurgen Gamer, Renate Sekul, Holger Deppe, Achim Feurer, Dirk Tomandl and Gunther Metz

DOI: 10.2174/157018005774717343

Identification of Privileged Scaffolds from a Diversified Chemical Library forβ-Secretase Inhibition

, 2(8): 595 - 600

Nicolas Pietrancosta, Gilles Quelever, Cedrik Garino, Younes Laras, Stephane Burlet and Jean-Louis Kraus

DOI: 10.2174/157018005774717352

Synthesis and Biological Evaluation of 1,2,4-Triazolo[2,3-a]pyrrole Derivatives as Alpha-4 ( α4) Integrin Antagonists

, 2(8): 601 - 605

Edward C. Lawson, William A. Kinney, Rosemary J. Santulli, Carol M. Fisher, Bruce P. Damiano and Bruce E. Maryanoff

DOI: 10.2174/157018005774717280

Szeged Index - Applications for Drug Modeling&#

, 2(8): 606 - 624

Padmakar V. Khadikar, Sneha Karmarkar, Vijay K. Agrawal, Jyoti Singh, Anjali Shrivastava, Istvan Lukovits and Mircea V. Diudea

DOI: 10.2174/157018005774717334

Initial Structure-Activity Relationships for a Caprolactam-based Series of Neutral Factor Xa Inhibitors: Lead Identification

, 2(8): 625 - 630

Gregory S. Bisacchi, Philip D. Stein, Jack Z. Gougoutas, Karen S. Hartl, R. Michael Lawrence, Eddie Liu, Andrew Pudzianowski, William A. Schumacher, Doree Sitkoff, Thomas E. Steinbacher, James Sutton, Zhaoxiao Zhang and Steven M. Seiler

DOI: 10.2174/157018005774717316

Synthesis and Evaluation of p-Nitrophenylβ-D-Glucopyranosiduronic Analogues as New Triggers for β-Glucuronidase Mediated Prodrug Mono- Therapy

, 2(8): 631 - 637

Damien Combaud, Mickael Thomas, Sebastien Papot and Jean-Pierre Gesson

DOI: 10.2174/157018005774717271

Structure Based Design of Inhibitors of Aspartic Protease of HIV-1

, 2(8): 638 - 646

V. Frecer, A. Jedinak, A. Tossi, F. Berti, F. Benedetti, D. Romeo and S. Miertus

DOI: 10.2174/157018005774717307

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