Contents

Letters in Drug Design & Discovery, Volume 2 - Number 1

Graphical Abstracts

, 2(1): v


DOI: 10.2174/157018081050201000v




RNA Silencing Technologies in Drug Discovery and Target Validation

, 2(1): 1 - 18

Elizabeth Rayburn, Hui Wang, Jie He and Ruiwen Zhang


DOI: 10.2174/1570180053398325




Inhibition of Transforming Growth Factor- βActivation is a Novel Effect of Chymase Inactivation

, 2(1): 19 - 22

S. Takai and M. Miyazaki


DOI: 10.2174/1570180053398433




In-Vitro Searching for a New Potent Reactivator of Acetylcholinesterase Inhibited by Nerve Agent VX

, 2(1): 23 - 25

K. Kuca, J. Cabal, J. Bajgar and D. Jun


DOI: 10.2174/1570180053398398




Farnesyltransferase Inhibitors: Overview of their Action and Role in Solid Malignancy Therapy

, 2(1): 26 - 35

Stefano Margaritora, Alfredo Cesario, Venanzio Porziella, Pierluigi Granone, Alessia Catassi and Patrizia Russo


DOI: 10.2174/1570180053398361




2,3,4,5- Tetrahydro- 1-Benzoxepines a Novel Class of Anti-Implantation Agents

, 2(1): 36 - 39

Vishnu K. Tandon and Sanjay Rai


DOI: 10.2174/1570180053398253




Design of a Heteroaryl Modified, 1,5-Disubstituted Pyrazole Cyclooxygenase-2 (COX-2) Selective Inhibitor

, 2(1): 40 - 43

M. Ezawa, D. S. Garvey, D. R. Janero, S. P. Khanapure, L. G. Letts, A. Martino, R. R. Ranatunge, D. J. Schwalb and D. V. Young


DOI: 10.2174/1570180053398451




L-Carnitine Effect upon Iron Growth Inhibition on Saccharomyces cerevisiae

, 2(1): 44 - 47

C. A. Stella, H. I. Burgos, M. Salellas, M. L. Cristaldo, E. H. Ramos and N. Kriguer


DOI: 10.2174/1570180053398415




Design and Synthesis of Combinatorial Scaffolds-Diazepinone and Homopiperazine

, 2(1): 48 - 50

Chung-Ming Sun


DOI: 10.2174/1570180053398280




Solution-Phase Parallel Synthesis of N,6-Disubstituted Isoquinuclidines as Ibogaine Analogs

, 2(1): 51 - 54

M. S. Levi, M. O.F. Khan and R. F. Borne


DOI: 10.2174/1570180053398217




Synthesis and Biological Activity of C-8 Fluoroaryl Substituted Pyrimidine Linked-Pyrrolobenzodiazepine Conjugates

, 2(1): 55 - 61

Ahmed Kamal, K. Laxma Reddy, V. Devaiah, N. Shankaraiah, M. Shiva Kumar and G. Suresh Kumar Reddy


DOI: 10.2174/1570180053398343




Design, Synthesis and Pharmacological Evaluation of New Nonsteroidal Antiinflammatory 1,3,4-Thiadiazole Derivatives

, 2(1): 62 - 67

L. S. Varandas, C. A.M. Fraga, A. L.P. Miranda and E. J. Barreiro


DOI: 10.2174/1570180053398235




Pharmacological Profile of New Deamino Analogues of Sabarubicin (MEN 10755)

, 2(1): 68 - 73

M. Bigioni, C. Salvatore, A. Cipollone, M. Berettoni, C. A. Maggi and M. Binaschi


DOI: 10.2174/1570180053398307




Exploiting the Ubiquitin-Proteasome Pathway for Anticancer Drug Discovery: Unanswered Questions and Future Directions

, 2(1): 74 - 81

D. M. Smith, K. G. Daniel and Q. P. Dou


DOI: 10.2174/1570180053398406




Author Index to Volume 1

, 2(1): 82 - 85

Bentham Science Publishers


DOI: 10.2174/1570180053398479




Subject Index to Volume 1

, 2(1): 86 - 91

Bentham Science Publishers


DOI: 10.2174/1570180053398299




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