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Letters in Drug Design & Discovery

Volume 17, 12 Issues, 2020
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

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    Chemistry, Medicinal

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Contents

Letters in Drug Design & Discovery, Volume 17 - Number 2


Review Article

Progress in Synthesis and Bioactivity Evaluation of Pyrazoloquinazolines

, 17(2): 104 - 113

Hui Zhao, Xiaoxia Hu, Yue Zhang, Chunlei Tang* and Bainian Feng*


DOI: 10.2174/1570180815666181017120100



Research Article

Desirability Based Optimization of New Mesalazine Modified Release Formulations: Compression Coated Tablets and Mini Tablets in Capsules

, 17(2): 114 - 123

Marilena Vlachou*, Angeliki Siamidi and Yannis Dotsikas


DOI: 10.2174/1570180816666190110125812



Research Article

New 2-Oxopyridine/2-Thiopyridine Derivatives Tethered to a Benzotriazole with Cytotoxicity on MCF7 Cell Lines and with Antiviral Activities

, 17(2): 124 - 137

Adel Mahmoud Attia, Ahmed Ibrahin Khodair*, Eman Abdelnasser Gendy, Mohammed Abu El-Magd and Yaseen Ali Mosa Mohamed Elshaier*


DOI: 10.2174/1570180816666190220123547



Research Article

An Environment-friendly Synthesis of Piperonal Chalcones and Their Cytotoxic and Antioxidant Evaluation

, 17(2): 138 - 144

Sanal Dev, Della Grace Thomas Parambi, Bency Baby, Githa Elizabeth Mathew, Hendawy Omnia Magdy, Monu Joy, Shine Sudev and Bijo Mathew*


DOI: 10.2174/1570180815666181016155934



Research Article

Synthesis, Antiproliferative, and Antioxidant Activities of Substituted N-[(1,3,4-Oxadiazol-2-yl) Methyl] Benzamines

, 17(2): 145 - 154

Mohamed Jawed Ahsan*, Lakshya Bhandari, Shally Makkar, Rajan Singh, Mohd. Zaheen Hassan, Mohammed H. Geesi, Mohamed Afroz Bakht, Surender Singh Jadav, Tuniki Balaraju, Yassine Riadi , Sandhya Rani, Habibullah Khalilullah, Vasubabu Gorantla and Afzal Hussain


DOI: 10.2174/1570180816666181113110033



Research Article

3D-QSAR Assisted Design of Novel 7-Deazapurine Derivatives as TNNI3K Kinase Inhibitors Using Molecular Docking and Molecular Dynamics Simulation

, 17(2): 155 - 168

Pavithra K. Balasubramanian, Anand Balupuri, Swapnil P. Bhujbal and Seung Joo Cho*


DOI: 10.2174/1570180816666190110121300



Research Article

p-Trifluoroacetophenone Oxime Ester Derivatives: Synthesis, Antimicrobial and Cytotoxic Evaluation and Molecular Modeling Studies

, 17(2): 169 - 183

İrem Bozbey, Suat Sari, Emine Şalva, Didem Kart and Arzu Karakurt*


DOI: 10.2174/1570180816666181128112249



Research Article

Anti-Trypanosoma cruzi Activity and Molecular Docking Studies of 1Hpyrazolo[ 3, 4-b]pyridine Derivatives

, 17(2): 184 - 191

Camilo Henrique da Silva Lima, Júlio César de Araújo Vanelis Soares, Joana Lucius de Sousa Ribeiro, Estela Maris Freitas Muri, Sérgio de Albuquerque and Luiza Rosaria Sousa Dias*


DOI: 10.2174/1570180816666190305141733



Research Article

Synthesis and Herbicidal Activities of Novel Thiazole PPO Inhibitors

, 17(2): 192 - 198

Shu Chen, Guihua Ren, Dan Pei, Fan Zhang, Jie Liu, Donglin Zhang, Ren Yang, Jianjun Shi, Tianming Xu and Chengxia Tan*


DOI: 10.2174/1570180816666190329221521



Research Article

Novel 3-{4-[2-Amino-4-(Substitutedphenyl)-2H-[1, 3] Oxazin/Thiazin-6-Yl} -2-Phenyl-3H-Quinazolin-4-One Derivatives as Enhancer of GABA Mediated Inhibition: Synthesis, Molecular Modeling and Pharmacological Studies

, 17(2): 199 - 213

Nimisha Jain and Pradeep Kumar Singour*


DOI: 10.2174/1570180816666190222155404



Research Article

QSAR Analysis of Selected Antimicrobial Structures Belonging to Nitro-derivatives of Heterocyclic Compounds

, 17(2): 214 - 225

Piotr Kawczak*, Leszek Bober and Tomasz Bączek


DOI: 10.2174/1570180815666181004112947






Editor-in-Chief

K. Kuca
University of Hradec Kralove
Hradec Kralove
Czech Republic

Biography View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
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Scopus CiteScore Metrics: 1.05

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