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Letters in Drug Design & Discovery

Volume 18, 12 Issues, 2021
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

Contents

Letters in Drug Design & Discovery, Volume 17 - Number 11


Letter Article

Design, Synthesis and Biological Evaluation: 5-amino-1H-pyrazole-1- carbonyl derivatives as FGFR Inhibitors

, 17(11): 1330 - 1341

Yan Zhang and Niefang Yu*


DOI: 10.2174/1570180817999200608140628



Research Article

Design, Synthesis, Docking and Computational Pharmacokinetic Profiling of New Pyrazolinyl Thiazolinone Biheterocycles as Potent Antimicrobial Agents

, 17(11): 1342 - 1354

Vinutha Vittala Salian, Badiadka Narayana*, Balladka Kunhanna Sarojini, Sharath Chandra Kodandoor and Anupam Glorious Lobo


DOI: 10.2174/1570180817999200623115049



Research Article

Evaluating Phenyl Propanoids Isolated from Citrus medica as Potential Inhibitors for Mitotic kinesin Eg5

, 17(11): 1355 - 1363

Himesh Makala, Venkatasubramanian Ulaganathan*, Aravind Sivasubramanian, Narendran Rajendran and Shankar Subramanian


DOI: 10.2174/1570180817999200630125449



Research Article

QSAR Studies of Sulfonamide Hydroxamates Derivatives as MMP-2 Inhibitors Topomer CoMFA and Molecular Docking

, 17(11): 1364 - 1371

Jian-Bo Tong*, Feng Yi, Ding Luo and Tian-Hao Wang


DOI: 10.2174/1570180817999200630124920



Research Article

Synthesis, Characterization and Antimicrobial Activity of Some Novel 1- substituted Benzimidazole Derivatives

, 17(11): 1372 - 1379

Erkut Isik, Demet Astley, Seda Yuksekdanaci* and Ihsan Yasa


DOI: 10.2174/1570180817999200531164230



Research Article

Design, Synthesis, In vitro and In silico Evaluation of New Hydrazonebased Antitumor Agents as Potent Akt Inhibitors

, 17(11): 1380 - 1392

Emine Merve Güngör, Mehlika Dilek Altıntop*, Belgin Sever and Gülşen Akalın Çiftçi


DOI: 10.2174/1570180817999200618163507



Research Article

Computational Analysis of Dynamical Fluctuations of Oncoprotein E7 (HPV 16) for the Hot Spot Residue Identification Using Elastic Network Model

, 17(11): 1393 - 1400

Rabbiah Malik*, Sahar Fazal and Mohammad Amjad Kamal


DOI: 10.2174/1570180817999200606225735



Research Article

Evaluation of Kaempferol as AKT Dependent mTOR Regulator via Targeting FKBP-12 in Hepatocellular Carcinoma: An In silico Approach

, 17(11): 1401 - 1408

Pooja Siniprasad, Bhagyalakshmi Nair, Vaisali Balasubramaniam, Prashanth Sadanandan, Puliyapally Krishnan Namboori* and Lekshmi Reghu Nath*


DOI: 10.2174/1570180817999200623115703



Research Article

Synthesis and Evaluation of Dapagliflozin Ester Prodrugs with Improved Hygroscopicity and Thermal Stability

, 17(11): 1409 - 1421

Si Young Sung, Yu Na Chae, Dae Young Lee, Kyeong Min Kim, Eun Jung Kim, Ji Hye Han, Wook Kim and Sung-Hwa Yoon*


DOI: 10.2174/1570180817999200618162949



Research Article

Comparative Proteome Analysis of Mycobacterium Tuberculosis Strains - H37Ra, H37Rv, CCDC5180, and CAS/NITR204: A Step Forward to Identify Novel Drug Targets

, 17(11): 1422 - 1431

Shradheya R.R. Gupta, Ekta Gupta, Avnam Ohri, Sandeep Kumar Shrivastava, Sumita Kachhwaha, Vinay Sharma, Rupesh Kumar Mishra and Ravi Ranjan Kumar Niraj*


DOI: 10.2174/1570180817999200531165148



Research Article

Novel 2-(5-Aryl)thiophen-2-yl)benzimidazoles; Design, Synthesis and In vitro Evaluation Against Cercarial Phase of Schistosoma mansoni

, 17(11): 1432 - 1438

Serry Atta El Bialy, Basem Mansour*, Waleed Abdelhakeem Bayoumi, Amira Taman and Hassan Mohammed Eissa


DOI: 10.2174/1570180817999200523181211



Research Article

High Anti-cancer Activity, Low Animal Toxicity, and Structure Activity Relationships of Curcumin Analogs

, 17(11): 1439 - 1455

Sen-Chuan Song, Yu-Liang Mai, Hua-Hong Shi, Bing Liao* and Fei Wang*


DOI: 10.2174/2352096513999200714103641




Editor-in-Chief

K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
Biography
View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 2.0

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