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Letters in Drug Design & Discovery

Volume 17, 12 Issues, 2020
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

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  • 57th of 61 in

    Chemistry, Medicinal

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Letters in Drug Design & Discovery, Volume 16 - Number 3

Research Article   Open Access

A Study on the Synthesis of Risedronic Acid: The Role of an Ionic Liquid Additive

, 16(3): 238 - 244

Dávid Illés Nagy, Alajos Grün, Júlia Sinkovicz, Sándor Garadnay, István Greiner and György Keglevich*

DOI: 10.2174/1570180815666180626122630

Research Article

Total Synthesis and Antibacterial Screening of (±)-6,8-Dihydroxy-3- undecyl-3,4-dihydroisochromen-1-one: A Structural Analogue of Metabolites from Ononis natrix

, 16(3): 245 - 248

Hummera Rafique*, Aamer Saeed, Ehsan Ullah Mughal, Muhammad Naveed Zafar, Amara Mumtaz, Naghmana Kausar and Kiran Hina

DOI: 10.2174/1570180815666180502114402

Research Article

Green Synthesis, Characterization, DPPH and Ferrous Ion-chelating (FIC) Activity of Tetrakis-Schiff’s Bases of Terephthalaldehyde

, 16(3): 249 - 255

Momin Khan*, Umar Ali, Anis Ur Rahman, Muhammad Ibrahim, Abdul Hameed, Muhammad Asif, Zahid Hussain, Kanwal, Khalid Mohammed Khan, Shahnaz Perveen and Munir ur Rehman

DOI: 10.2174/1570180815666180531101404

Research Article

Coumarinyl Aryl/Alkyl Sulfonates with Dual Potential: Alkaline Phosphatase and ROS Inhibitory Activities: In-Silico Molecular Modeling and ADME Evaluation

, 16(3): 256 - 272

Uzma Salar, Khalid Mohammed Khan*, Syeda Abida Ejaz, Abdul Hameed, Mariya al-Rashida, Shahnaz Perveen, Muhammad Nawaz Tahir, Jamshed Iqbal* and Muhammad Taha

DOI: 10.2174/1570180815666180327125738

Research Article

Cytotoxicity and Molecular Targeting Study of Novel 2-Chloro-3- substituted Quinoline Derivatives as Antitumor Agents

, 16(3): 273 - 283

Mohammed A.M. Massoud*, Magda A. El-Sayed, Waleed A. Bayoumi and Basem Mansour

DOI: 10.2174/1570180815666180604090924

Research Article

Catalyst Free and Energy Economical Synthesis of Thiazole Derivatives Bearing Azo Imine Linkage with Imidazole as Antimicrobial Agents

, 16(3): 284 - 290

Nayan M. Panchani and Hitendra S. Joshi*

DOI: 10.2174/1570180815666180627155443

Research Article

Assessing the Antimalarial Potentials of Phytochemicals: Virtual Screening, Molecular Dynamics and In-Vitro Investigations

, 16(3): 291 - 300

Saumya K. Patel, Mohd Athar, Prakash C. Jha*, Vijay M. Khedkar, Yogesh Jasrai, Himanshu A. Pandya, Linz-buoy George, Hyacinth Highland and Supriya Sharma

DOI: 10.2174/1570180815666180604085626

Research Article

3D QSAR Based Virtual Screening of Pyrido[1,2-a] Benzimidazoles as Potent Antimalarial Agents

, 16(3): 301 - 312

Kalicharan Sharma, Apeksha Srivastava, Pooja Tiwari, Shweta Sharma, Mohammad Shaquiquzzaman, M. Mumtaz Alam and Mymoona Akhter*

DOI: 10.2174/1570180815666180502115147

Research Article

Synthesis, Structure Elucidation and Biological Activities of Some Novel 4(3H)-Quinazolinones as Anti-Biofilm Agents

, 16(3): 313 - 321

Sevda Türk, Sevgi Karakuş*, Abdulilah Ece, Seyhan Ulusoy and Gülgün Bosgelmez-Tınaz

DOI: 10.2174/1570180815666180621101123

Research Article

Synthesis and Evaluation of Chalcone and its Derivatives as Potential Anticholinergic Agents

, 16(3): 322 - 332

Shahzad Murtaza*, Khoula Zubair Mir, Adina Tatheer and Raja Summe Ullah

DOI: 10.2174/1570180815666180523085436

Research Article

Aurones as New Porcine Pancreatic α-Amylase Inhibitors

, 16(3): 333 - 340

Khashayar Roshanzamir, Elaheh Kashani-Amin, Azadeh Ebrahim-Habibi* and Latifeh Navidpour*

DOI: 10.2174/1570180815666180712150600

Research Article

Investigating the Antidepressant-like Effects of some Benzimidazolepiperidine Derivatives by In-Vivo Experimental Methods

, 16(3): 341 - 346

Nazlı Turan, Ümide Demir Özkay*, Nafiz Öncü Can and Özgür Devrim Can

DOI: 10.2174/1570180815666181004103112

Research Article

N-Acetylserotonin vs Melatonin: In-Vitro Controlled Release from Hydrophilic Matrix Tablets

, 16(3): 347 - 352

M. Vlachou*, G. Stavrou, A. Siamidi, S. Flitouri, V. Ioannidou and S. Mavrokordopoulos

DOI: 10.2174/1570180815666180404125519


Evaluation of a Series of 9,10-Anthraquinones as Antiplasmodial Agents

, 16(3): 353 - 363

Che Puteh Osman*, Nor Hadiani Ismail, Aty Widyawaruyanti, Syahrul Imran, Lidya Tumewu, Chee Yan Choo and Sharinah Ideris

DOI: 10.2174/1570180815666180607085102


Synthesis of 3-furanyl-4,5-dihydroisoxazole Derivatives via Cycloaddition and their Antibacterial Evaluation

, 16(3): 364 - 369

Gabriela de Andrade Danin Barbosa, Alcino Palermo de Aguiar*, Erika Martins de Carvalho and Joseli Maria da Rocha Nogueira

DOI: 10.2174/1570180815666180627115606


K. Kuca
University of Hradec Kralove
Hradec Kralove
Czech Republic

Biography View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
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Scopus CiteScore Metrics: 1.02


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