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Letters in Drug Design & Discovery

Volume 17, 12 Issues, 2020
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

In the current pandemic scenario, publication process of all articles related to Coronavirus will be expedited, for timely publication of much needed research


Letters in Drug Design & Discovery, Volume 16 - Number 3

Research Article   Open Access

A Study on the Synthesis of Risedronic Acid: The Role of an Ionic Liquid Additive

, 16(3): 238 - 244

Dávid Illés Nagy, Alajos Grün, Júlia Sinkovicz, Sándor Garadnay, István Greiner and György Keglevich*

DOI: 10.2174/1570180815666180626122630

Research Article

Total Synthesis and Antibacterial Screening of (±)-6,8-Dihydroxy-3- undecyl-3,4-dihydroisochromen-1-one: A Structural Analogue of Metabolites from Ononis natrix

, 16(3): 245 - 248

Hummera Rafique*, Aamer Saeed, Ehsan Ullah Mughal, Muhammad Naveed Zafar, Amara Mumtaz, Naghmana Kausar and Kiran Hina

DOI: 10.2174/1570180815666180502114402

Research Article

Green Synthesis, Characterization, DPPH and Ferrous Ion-chelating (FIC) Activity of Tetrakis-Schiff’s Bases of Terephthalaldehyde

, 16(3): 249 - 255

Momin Khan*, Umar Ali, Anis Ur Rahman, Muhammad Ibrahim, Abdul Hameed, Muhammad Asif, Zahid Hussain, Kanwal, Khalid Mohammed Khan, Shahnaz Perveen and Munir ur Rehman

DOI: 10.2174/1570180815666180531101404

Research Article

Coumarinyl Aryl/Alkyl Sulfonates with Dual Potential: Alkaline Phosphatase and ROS Inhibitory Activities: In-Silico Molecular Modeling and ADME Evaluation

, 16(3): 256 - 272

Uzma Salar, Khalid Mohammed Khan*, Syeda Abida Ejaz, Abdul Hameed, Mariya al-Rashida, Shahnaz Perveen, Muhammad Nawaz Tahir, Jamshed Iqbal* and Muhammad Taha

DOI: 10.2174/1570180815666180327125738

Research Article

Cytotoxicity and Molecular Targeting Study of Novel 2-Chloro-3- substituted Quinoline Derivatives as Antitumor Agents

, 16(3): 273 - 283

Mohammed A.M. Massoud*, Magda A. El-Sayed, Waleed A. Bayoumi and Basem Mansour

DOI: 10.2174/1570180815666180604090924

Research Article

Catalyst Free and Energy Economical Synthesis of Thiazole Derivatives Bearing Azo Imine Linkage with Imidazole as Antimicrobial Agents

, 16(3): 284 - 290

Nayan M. Panchani and Hitendra S. Joshi*

DOI: 10.2174/1570180815666180627155443

Research Article

Assessing the Antimalarial Potentials of Phytochemicals: Virtual Screening, Molecular Dynamics and In-Vitro Investigations

, 16(3): 291 - 300

Saumya K. Patel, Mohd Athar, Prakash C. Jha*, Vijay M. Khedkar, Yogesh Jasrai, Himanshu A. Pandya, Linz-buoy George, Hyacinth Highland and Supriya Sharma

DOI: 10.2174/1570180815666180604085626

Research Article

3D QSAR Based Virtual Screening of Pyrido[1,2-a] Benzimidazoles as Potent Antimalarial Agents

, 16(3): 301 - 312

Kalicharan Sharma, Apeksha Srivastava, Pooja Tiwari, Shweta Sharma, Mohammad Shaquiquzzaman, M. Mumtaz Alam and Mymoona Akhter*

DOI: 10.2174/1570180815666180502115147

Research Article

Synthesis, Structure Elucidation and Biological Activities of Some Novel 4(3H)-Quinazolinones as Anti-Biofilm Agents

, 16(3): 313 - 321

Sevda Türk, Sevgi Karakuş*, Abdulilah Ece, Seyhan Ulusoy and Gülgün Bosgelmez-Tınaz

DOI: 10.2174/1570180815666180621101123

Research Article

Synthesis and Evaluation of Chalcone and its Derivatives as Potential Anticholinergic Agents

, 16(3): 322 - 332

Shahzad Murtaza*, Khoula Zubair Mir, Adina Tatheer and Raja Summe Ullah

DOI: 10.2174/1570180815666180523085436

Research Article

Aurones as New Porcine Pancreatic α-Amylase Inhibitors

, 16(3): 333 - 340

Khashayar Roshanzamir, Elaheh Kashani-Amin, Azadeh Ebrahim-Habibi* and Latifeh Navidpour*

DOI: 10.2174/1570180815666180712150600

Research Article

Investigating the Antidepressant-like Effects of some Benzimidazolepiperidine Derivatives by In-Vivo Experimental Methods

, 16(3): 341 - 346

Nazlı Turan, Ümide Demir Özkay*, Nafiz Öncü Can and Özgür Devrim Can

DOI: 10.2174/1570180815666181004103112

Research Article

N-Acetylserotonin vs Melatonin: In-Vitro Controlled Release from Hydrophilic Matrix Tablets

, 16(3): 347 - 352

M. Vlachou*, G. Stavrou, A. Siamidi, S. Flitouri, V. Ioannidou and S. Mavrokordopoulos

DOI: 10.2174/1570180815666180404125519


Evaluation of a Series of 9,10-Anthraquinones as Antiplasmodial Agents

, 16(3): 353 - 363

Che Puteh Osman*, Nor Hadiani Ismail, Aty Widyawaruyanti, Syahrul Imran, Lidya Tumewu, Chee Yan Choo and Sharinah Ideris

DOI: 10.2174/1570180815666180607085102


Synthesis of 3-furanyl-4,5-dihydroisoxazole Derivatives via Cycloaddition and their Antibacterial Evaluation

, 16(3): 364 - 369

Gabriela de Andrade Danin Barbosa, Alcino Palermo de Aguiar*, Erika Martins de Carvalho and Joseli Maria da Rocha Nogueira

DOI: 10.2174/1570180815666180627115606


K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)

View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 1.05



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