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Letters in Drug Design & Discovery

Volume 16, 12 Issues, 2019
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

Contents

Letters in Drug Design & Discovery, Volume 16 - Number 1



Research Article

Copper-catalyzed Convenient Synthesis and SAR Studies of Substituted- 1,2,3-triazole as Antimicrobial Agents

, 16(1): 3 - 10

Aniket P. Sarkate*, Kshipra S. Karnik, Pravin S. Wakte, Ajinkya P. Sarkate, Ashwini V. Izankar and Devanand B. Shinde


DOI: 10.2174/1570180815666180326153322



Research Article

Development and Validation of a Robust QSAR Model for Benzothiazole Hydrazone Derivatives as Bcl-XL Inhibitors

, 16(1): 11 - 20

Pawan Gupta* and Aleksandrs Gutcaits


DOI: 10.2174/1570180815666180502093039



Research Article

Discovery of Hybrid Purine-quinoline Molecules and Their Cytotoxic Evaluation

, 16(1): 21 - 28

Khushal M. Kapadiya and Ranjan C. Khunt*


DOI: 10.2174/1570180815666180419151742



Research Article

Synthesis, Nematicidal Activity and Docking Study of Novel Pyrazole-4- Carboxamide Derivatives Against Meloidogyne incognita

, 16(1): 29 - 35

Long Cheng, Wen Zhao, Zhong-Hua Shen, Tian-Ming Xu, Hong-Ke Wu, Wei-Li Peng* and Xing-Hai Liu*


DOI: 10.2174/1570180815666180326150827



Research Article

Novel Piperazine Amides of Cinnamic Acid Derivatives as Tyrosinase Inhibitors

, 16(1): 36 - 44

Zehra Tuğçe Gür, Fatma Sezer Şenol, Suhaib Shekfeh, İlkay Erdoğan Orhan , Erden Banoğlu and Burcu Çalişkan*


DOI: 10.2174/1570180815666180420105652



Research Article

Synthesis and Cytotoxicity Studies on Novel Piperazinylacetamides

, 16(1): 45 - 51

Eman Bobtaina, Enise Ece Gurdal*, Irem Durmaz, Rengul Cetin Atalay and Mine Yarim


DOI: 10.2174/1570180815666180501124009



Research Article

Genoprotective Effect of New Triazine Derivatives in Endosulfan Mediated Toxicity, an In vivo and In vitro Study

, 16(1): 52 - 57

Nima Naderi, Seyed Mostafa Ghasemi Najarkolaee, Mona Modanlookordi, Mohammad Shokrzadeh and Hamid Irannejad*


DOI: 10.2174/1570180815666180420095446



Research Article

Synthesis of 1,3-benzoxazines Based on 2,4,4-trimethyl-7,2’,4’-trihydroxy Flavan: Antibacterial, Anti-inflammatory, Cyclooxygenase-2 Inhibition and Molecular Modelling Studies

, 16(1): 58 - 65

Issam A. Mohammed, Mahmood Ahmed*, Rabia Ikram, Muhammad Muddassar, Muhammad Abdul Qadir and Khalijah Binti Awang


DOI: 10.2174/1570180815666180420100922



Research Article

A New Class of Pure Estrogen Alpha Receptor Antagonists; Design, Synthesis and in-vitro Screening

, 16(1): 66 - 81

Akbar John Jameera Begam, Katike Ahamed Basheer, Selvaraj Jubie*, Srikanth Jupudi, Mohammed Afzal Azam and Palanisamy Dhanabal


DOI: 10.2174/1570180815666180327124634



Research Article

New Benzodioxole-based Pyrazoline Derivatives: Synthesis and Anticandidal, In silico ADME, Molecular Docking Studies

, 16(1): 82 - 92

Ahmet Özdemir*, Belgin Sever and Mehlika Dilek Altıntop


DOI: 10.2174/1570180815666180326152726



Letter

Synthesis of a Series of Chalcones and Related Flavones and Evaluation of their Antibacterial and Antifungal Activities

, 16(1): 93 - 100

Hind Benouda, Btissam Bouchal, Allal Challioui, Abdelkader Oulmidi, Tarik Harit, Fouad Malek, Abdelkhalek Riahi, Mohammed Bellaoui and Boufelja Bouammali *


DOI: 10.2174/1570180815666180404130430




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