Letters in Drug Design & Discovery
Volume 16, 12 Issues, 2019
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access
Contents
Letters in Drug Design & Discovery, Volume 16 - Number 1
Biography Open Access
Preface Open Access
Research Article
Copper-catalyzed Convenient Synthesis and SAR Studies of Substituted- 1,2,3-triazole as Antimicrobial Agents
, 16(1): 3 - 10Aniket P. Sarkate*, Kshipra S. Karnik, Pravin S. Wakte, Ajinkya P. Sarkate, Ashwini V. Izankar and Devanand B. Shinde
DOI: 10.2174/1570180815666180326153322
Copper-catalyzed Convenient Synthesis and SAR Studies of Substituted- 1,2,3-triazole as Antimicrobial Agents
Research Article
Development and Validation of a Robust QSAR Model for Benzothiazole Hydrazone Derivatives as Bcl-XL Inhibitors
, 16(1): 11 - 20Pawan Gupta* and Aleksandrs Gutcaits
DOI: 10.2174/1570180815666180502093039
Development and Validation of a Robust QSAR Model for Benzothiazole Hydrazone Derivatives as Bcl-XL Inhibitors
Research Article
Discovery of Hybrid Purine-quinoline Molecules and Their Cytotoxic Evaluation
, 16(1): 21 - 28Khushal M. Kapadiya and Ranjan C. Khunt*
DOI: 10.2174/1570180815666180419151742
Discovery of Hybrid Purine-quinoline Molecules and Their Cytotoxic Evaluation
Research Article
Synthesis, Nematicidal Activity and Docking Study of Novel Pyrazole-4- Carboxamide Derivatives Against Meloidogyne incognita
, 16(1): 29 - 35Long Cheng, Wen Zhao, Zhong-Hua Shen, Tian-Ming Xu, Hong-Ke Wu, Wei-Li Peng* and Xing-Hai Liu*
DOI: 10.2174/1570180815666180326150827
Synthesis, Nematicidal Activity and Docking Study of Novel Pyrazole-4- Carboxamide Derivatives Against Meloidogyne incognita
Research Article
Novel Piperazine Amides of Cinnamic Acid Derivatives as Tyrosinase Inhibitors
, 16(1): 36 - 44Zehra Tuğçe Gür, Fatma Sezer Şenol, Suhaib Shekfeh, İlkay Erdoğan Orhan , Erden Banoğlu and Burcu Çalişkan*
DOI: 10.2174/1570180815666180420105652
Novel Piperazine Amides of Cinnamic Acid Derivatives as Tyrosinase Inhibitors
Research Article
Synthesis and Cytotoxicity Studies on Novel Piperazinylacetamides
, 16(1): 45 - 51Eman Bobtaina, Enise Ece Gurdal*, Irem Durmaz, Rengul Cetin Atalay and Mine Yarim
DOI: 10.2174/1570180815666180501124009
Synthesis and Cytotoxicity Studies on Novel Piperazinylacetamides
Research Article
Genoprotective Effect of New Triazine Derivatives in Endosulfan Mediated Toxicity, an In vivo and In vitro Study
, 16(1): 52 - 57Nima Naderi, Seyed Mostafa Ghasemi Najarkolaee, Mona Modanlookordi, Mohammad Shokrzadeh and Hamid Irannejad*
DOI: 10.2174/1570180815666180420095446
Genoprotective Effect of New Triazine Derivatives in Endosulfan Mediated Toxicity, an In vivo and In vitro Study
Research Article
Synthesis of 1,3-benzoxazines Based on 2,4,4-trimethyl-7,2’,4’-trihydroxy Flavan: Antibacterial, Anti-inflammatory, Cyclooxygenase-2 Inhibition and Molecular Modelling Studies
, 16(1): 58 - 65Issam A. Mohammed, Mahmood Ahmed*, Rabia Ikram, Muhammad Muddassar, Muhammad Abdul Qadir and Khalijah Binti Awang
DOI: 10.2174/1570180815666180420100922
Synthesis of 1,3-benzoxazines Based on 2,4,4-trimethyl-7,2’,4’-trihydroxy Flavan: Antibacterial, Anti-inflammatory, Cyclooxygenase-2 Inhibition and Molecular Modelling Studies
Research Article
A New Class of Pure Estrogen Alpha Receptor Antagonists; Design, Synthesis and in-vitro Screening
, 16(1): 66 - 81Akbar John Jameera Begam, Katike Ahamed Basheer, Selvaraj Jubie*, Srikanth Jupudi, Mohammed Afzal Azam and Palanisamy Dhanabal
DOI: 10.2174/1570180815666180327124634
A New Class of Pure Estrogen Alpha Receptor Antagonists; Design, Synthesis and in-vitro Screening
Research Article
New Benzodioxole-based Pyrazoline Derivatives: Synthesis and Anticandidal, In silico ADME, Molecular Docking Studies
, 16(1): 82 - 92Ahmet Özdemir*, Belgin Sever and Mehlika Dilek Altıntop
DOI: 10.2174/1570180815666180326152726
New Benzodioxole-based Pyrazoline Derivatives: Synthesis and Anticandidal, In silico ADME, Molecular Docking Studies
Letter
Synthesis of a Series of Chalcones and Related Flavones and Evaluation of their Antibacterial and Antifungal Activities
, 16(1): 93 - 100Hind Benouda, Btissam Bouchal, Allal Challioui, Abdelkader Oulmidi, Tarik Harit, Fouad Malek, Abdelkhalek Riahi, Mohammed Bellaoui and Boufelja Bouammali *
DOI: 10.2174/1570180815666180404130430
Synthesis of a Series of Chalcones and Related Flavones and Evaluation of their Antibacterial and Antifungal Activities
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Editor-in-Chief
George Perry
University of Texas
San Antonio, TX
USA
University of Texas
San Antonio, TX
USA
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Journal History
Letters in Drug Design & Discovery was introduced in 2004 with the assistance of Dr. George Perry, who is the current Editor-in-Chief serving since 2004.
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